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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 14, 2011, Pages 4306-4309

Pyrrolo[2,3-c]azepine derivatives: A new class of potent protein tyrosine phosphatase 1B inhibitors

(7) Xie, Jianwei a,c,d Tian, Jinying b Su, Li a Huang, Manna a Zhu, Xinhai a Ye, Fei b Wan, Yiqian a

a SUN YAT SEN UNIVERSITY (China)

b INSTITUTE OF MATERIA MEDICA (China)

c SHIHEZI UNIVERSITY (China)

d Xinjiang Bingtuan Key Laboratory for Green Processing of Chemical Engineering (China)

Author keywords

Aldisin; Inhibitor; Marine natural product; Protein tyrosine phosphatase 1B; Synthesis

Indexed keywords

6,7 DIHYDROPYRROLO[2,3 C]AZEPINE 4,8(1H,5H) DIONE; AZEPINE DERIVATIVE; PROTEIN TYROSINE PHOSPHATASE 1B INHIBITOR; PYRROLO[2,3 C]AZEPINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; IC 50; IN VITRO STUDY;

AZEPINES; BIPHENYL COMPOUNDS; ENZYME INHIBITORS; HUMANS; INDOLES; PROTEIN TYROSINE PHOSPHATASE, NON-RECEPTOR TYPE 1; PYRROLES; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 79959906648 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.05.052 Document Type: Article

Times cited : (27)

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