Docking study, in vitro anticancer screening and radiosensitizing evaluation of some new fluorine-containing quinoline and pyrimidoquinoline derivatives bearing a sulfonamide moiety
ANTINEOPLASTIC ACTIVITY;
ARTICLE;
BINDING AFFINITY;
CANCER CELL CULTURE;
CELL KILLING;
CONTROLLED STUDY;
DRUG SCREENING;
DRUG SYNTHESIS;
GAMMA RADIATION;
HUMAN;
HUMAN CELL;
IC 50;
IN VITRO STUDY;
MOLECULAR DOCKING;
Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX
DOI 10.1016/j.bmcl.2003.09.062
Abbate F, Casini A, Owa T, Scozzafava A, Supuran CT (2004) Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agents, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX. Bioorg Med Chem Lett 14:217-223 (Pubitemid 38010223)
Sulfonamides and sulfonylated derivatives as anticancer agents
DOI 10.2174/1568009023334060
Casini A, Scozzafava A, Mastrolorenzo A, Supuran CT (2002) Sulfonamides and sulfonylated derivatives as anticancer agents. Curr Cancer Drug Targets 2:55-75 (Pubitemid 34627379)
Novel antitumor and radioprotective sulfonamides containing pyrrolo[2,3-d]pyrimidines
Ghorab MM, Noaman E, Ismail MM, Heiba HI, Ammar YA, Sayed MY (2006) Novel antitumor and radioprotective sulfonamides containing pyrrolo[2,3-d] pyrimidines. Arzneimittelforschung 56:405-413 (Pubitemid 44047519)
Synthesis of some novel quinolines and pyrimido[4,5-b]quinolines bearing a sulfonamide moiety as potential anticancer and radioprotective agents
Ghorab MM, Ragab FA, Noaman E, Heiba HI, El-Hossary EM (2007) Synthesis of some novel quinolines and pyrimido[4,5-b]quinolines bearing a sulfonamide moiety as potential anticancer and radioprotective agents. Arzneimittelforschung 57:795-803
Design, synthesis and anticancer evaluation of novel tetrahydroquinoline derivatives containing sulfonamide moiety
Ghorab MM, Ragab FA, Hamed MM (2009) Design, synthesis and anticancer evaluation of novel tetrahydroquinoline derivatives containing sulfonamide moiety. Eur J Med Chem 44:4211-4217
Antitumor activity of 4-amino and 8-methyl-4-(3diethylamino propylamino)pyrimido[40, 50:4, 5]thieno (2, 3-b) quinolines
DOI 10.1016/j.jphotobiol.2003.09.003
Gopal M, Shenoy S, Doddamani LS (2003) Antitumor activity of 4-amino and 8-methyl-4-(3diethylamino propylamino)pyrimido[ 40,50:4,5]thieno (2, 3-b) quinolines. J Photochem Photobiol B 72:69-78 (Pubitemid 37509037)
Novel synthesis of pyrrolo[2,3-d]pyrimidines bearing sulfonamide moieties as potential antitumor and radioprotective agents
Ismail MM, Ghorab MM, Noaman E, Ammar YA, Heiba HI, Sayed MY (2006) Novel synthesis of pyrrolo[2,3-d]pyrimidines bearing sulfonamide moieties as potential antitumor and radioprotective agents. Arzneimittelforschung 56:301-308
G2 arrest and apoptosis by 2-amino-N-quinoline-8-yl-benzene-sulfonamide (QBS), a novel cytotoxic compound
Kim YH, Shin KJ, Lee TG, Kim E, Lee MS, Ryu SH, Suh PG (2005) G2 arrest and apoptosis by 2-amino-N-quinoline-8-yl-benzene-sulfonamide (QBS), a novel cytotoxic compound. Biochem Pharmacol 69:1333-1341
Discovery of 4-amino and 4-hydroxy-1- Aroylindoles as potent tubulin polymerization inhibitors
Liou JP, Wu ZY, Kuo CC, Chang CY, Lu PY, Chen CM, Hsieh HP, Chang JY (2008) Discovery of 4-amino and 4-hydroxy-1- aroylindoles as potent tubulin polymerization inhibitors. J Med Chem 51:4351-4355
Carbonic anhydrases: Current state of the art, therapeutic applications and future prospects
DOI 10.1080/14756360410001689540
Pastorekova S, Parkkila S, Pastorek J, Supuran CT (2004) Carbonic anhydrases: current state of the art, therapeutic applications and future prospects. J Enzym Inhib Med Chem 19:199-229 (Pubitemid 39004275)
Synthesis and in vitro antitumor evaluation of some indeno[1,2-c] pyrazol(in)es substituted with sulfonamide, sulfonylurea(-thiourea) pharmacophores, and some derived thiazole ring systems
Rostom SA (2006) Synthesis and in vitro antitumor evaluation of some indeno[1,2-c]pyrazol(in)es substituted with sulfonamide, sulfonylurea(-thiourea) pharmacophores, and some derived thiazole ring systems. Bioorg Med Chem 14:6475-6485
COX-2 selective inhibitors, carbonic anhydrase inhibition and anticancer properties of sulfonamides belonging to this class of pharmacological agents
Supuran CT, Casini A, Mastrolorenzo A, Scozzafava A (2004) COX-2 selective inhibitors, carbonic anhydrase inhibition and anticancer properties of sulfonamides belonging to this class of pharmacological agents. Mini-Rev Med Chem 4:625-632 (Pubitemid 38961227)
Indanesulfonamides as carbonic anhydrase inhibitors. Toward structure-based design of selective inhibitors of the tumor-associated isozyme CA IX
Thiry A, Ledecq M, Cecchi A, Dogne JM, Wouters J, Supuran CT, Masereel B (2006) Indanesulfonamides as carbonic anhydrase inhibitors. Toward structure-based design of selective inhibitors of the tumor-associated isozyme CA IX. J Med Chem 49:2743-2749
Synthesis and cytotoxic evaluation of certain 4-anilino-2-phenylquinoline derivatives
Zhao YL, Chen YL, Chang FS, Tzeng CC (2005) Synthesis and cytotoxic evaluation of certain 4-anilino-2-phenylquinoline derivatives. Eur J Med Chem 40:792-797
