메뉴 건너뛰기




Volumn 70, Issue 1-2, 2011, Pages 49-58

Nasal in situ gel containing hydroxy propyl β-cyclodextrin inclusion complex of artemether: Development and in vitro evaluation

Author keywords

In situ gel; Inclusion mode; Mucoadhesion; Phase solubility; Temperature induced gelation

Indexed keywords


EID: 79956057329     PISSN: 09230750     EISSN: None     Source Type: Journal    
DOI: 10.1007/s10847-010-9861-x     Document Type: Article
Times cited : (36)

References (33)
  • 1
    • 0034813570 scopus 로고    scopus 로고
    • Artemisinin and its derivatives: An important new class of antimalarial agents
    • DOI 10.1016/S0163-7258(01)00140-1, PII S0163725801001401
    • GA Balint 2001 Artemisinin and its derivatives: an important new class of antimalarial agents Pharmacol. Ther. 90 261 265 10.1016/S0163-7258(01)00140-1 1:CAS:528:DC%2BD3MXntV2hurw%3D (Pubitemid 32913479)
    • (2001) Pharmacology and Therapeutics , vol.90 , Issue.2-3 , pp. 261-265
    • Balint, G.A.1
  • 2
    • 0024512810 scopus 로고
    • Thermospray mass spectroscopy/high performance liquid chromatographic identification of the metabolites formed from arteether using a rat liver microsome preparation
    • JK Baker RH Yarber CD Hufford IS Lee HN Elsohly JD McChesney 1988 Thermospray mass spectroscopy/high performance liquid chromatographic identification of the metabolites formed from arteether using a rat liver microsome preparation Biomed. Environ. Mass. Spectrom. 18 337 351 10.1002/bms.1200180509 (Pubitemid 19116520)
    • (1989) Biomedical and Environmental Mass Spectrometry , vol.18 , Issue.5 , pp. 337-351
    • Baker, J.K.1    Yarber, R.H.2    Hufford, C.D.3    Lee, I.-S.4    ElSohly, H.N.5    McChesney, J.D.6
  • 3
    • 0345827826 scopus 로고    scopus 로고
    • In vitro and in vivo evaluation of the Gelrite® gellan gum-based ocular delivery system for indomethacin
    • J Balasubramaniam S Kant JK Pandit 2003 In vitro and in vivo evaluation of the Gelrite® gellan gum-based ocular delivery system for indomethacin Acta Pharm. 53 251 261 1:CAS:528:DC%2BD2cXlvFSntA%3D%3D (Pubitemid 38083940)
    • (2003) Acta Pharmaceutica , vol.53 , Issue.4 , pp. 251-261
    • Balasubramaniam, J.1    Kant, S.2    Pandit, J.K.3
  • 4
    • 70350650218 scopus 로고
    • A general method of accessing skin permeatin enhancement mechanisms and optimization
    • Hsies, D.S., (eds.). New York, NY: Marcel Dekker Inc
    • Behl, C.R., Harper, N.J., Pei, J.Y.: A general method of accessing skin permeatin enhancement mechanisms and optimization. In: Hsies, D.S., (eds.) Drug permeation enhancement: theory and applications, 1st edn, p. 115. New York, NY: Marcel Dekker Inc (1994)
    • (1994) Drug Permeation Enhancement: Theory and Applications, 1st Edn , pp. 115
    • Behl, C.R.1    Harper, N.J.2    Pei, J.Y.3
  • 5
    • 68649127581 scopus 로고    scopus 로고
    • Artemether/hydroxypropyl-b cyclodextrin host-guest system: Characterization, phase-solubility and inclusion mode
    • 10.1016/j.bmc.2009.07.060 1:CAS:528:DC%2BD1MXhtVenurzN
    • B Yang J Lin Y Chen Y Liu 2009 Artemether/hydroxypropyl-b cyclodextrin host-guest system: characterization, phase-solubility and inclusion mode Bioorg. Med. Chem. 17 6311 6317 10.1016/j.bmc.2009.07.060 1:CAS:528:DC%2BD1MXhtVenurzN
    • (2009) Bioorg. Med. Chem. , vol.17 , pp. 6311-6317
    • Yang, B.1    Lin, J.2    Chen, Y.3    Liu, Y.4
  • 6
    • 0036182021 scopus 로고    scopus 로고
    • The use of chemically modified cyclodextrins in the development of formulations for chemical delivery systems
    • 1:CAS:528:DC%2BD38XhsFCnu74%3D
    • ME Brewster T Loftsson 2002 The use of chemically modified cyclodextrins in the development of formulations for chemical delivery systems Pharmazie 57 94 1:CAS:528:DC%2BD38XhsFCnu74%3D
    • (2002) Pharmazie , vol.57 , pp. 94
    • Brewster, M.E.1    Loftsson, T.2
  • 7
    • 0032482152 scopus 로고    scopus 로고
    • Temperature-responsive gels and thermogelling polymer matrices for protein and peptide delivery
    • DOI 10.1016/S0169-409X(97)00121-X, PII S0169409X9700121X
    • LE Bromberg ES Ron 1998 Protein and peptide release from temperature responsive gels and thermogelling polymer matrices Adv. Drug Deliv. Rev. 31 197 221 10.1016/S0169-409X(97)00121-X 1:CAS:528:DyaK1cXhvVSjsLg%3D (Pubitemid 28191866)
    • (1998) Advanced Drug Delivery Reviews , vol.31 , Issue.3 , pp. 197-221
    • Bromberg, L.E.1    Ron, E.S.2
  • 8
    • 33747036480 scopus 로고    scopus 로고
    • Thermodynamics of inclusion complexes of natural and modified cyclodextrins with propranolol in aqueous solution at 298 K
    • DOI 10.1016/j.bmc.2006.01.052, PII S096808960600085X
    • G Castronuovo M Niccoli 2006 Thermodynamics of inclusion complexes of natural and modified cyclodextrins with propanolol in aqueous solution at 298 K Bioorg. Med. Chem. 14 3883 3887 10.1016/j.bmc.2006.01.052 1:CAS:528: DC%2BD28XjvFWmsLY%3D (Pubitemid 44316610)
    • (2006) Bioorganic and Medicinal Chemistry , vol.14 , Issue.11 , pp. 3883-3887
    • Castronuovo, G.1    Niccoli, M.2
  • 9
    • 10444279209 scopus 로고    scopus 로고
    • Cyclodextrin-based pharmaceutics: Past, present and future
    • DOI 10.1038/nrd1576
    • ME Davis ME Brewster 2004 Cyclodextrin-based pharmaceutics: past, present, future Nat. Rev. Drug Discov. 3 1023 10.1038/nrd1576 1:CAS:528:DC%2BD2cXhtVarsL3P (Pubitemid 39642365)
    • (2004) Nature Reviews Drug Discovery , vol.3 , Issue.12 , pp. 1023-1035
    • Davis, M.E.1    Brewster, M.E.2
  • 10
    • 30744442534 scopus 로고    scopus 로고
    • Characterization of polymeric dispersions of dimenhydrinate in ethyl cellulose for controlled release
    • DOI 10.1016/j.ijpharm.2005.10.034, PII S0378517305007180
    • J Desai K Alexander A Riga 2006 Characterization of polymeric dispersions of dimenhydrinate in ethyl cellulose for controlled release Int. J. Pharm. 308 115 123 10.1016/j.ijpharm.2005.10.034 1:CAS:528:DC%2BD28Xls1Srsg%3D%3D (Pubitemid 43097242)
    • (2006) International Journal of Pharmaceutics , vol.308 , Issue.1-2 , pp. 115-123
    • Desai, J.1    Alexander, K.2    Riga, A.3
  • 11
    • 0141732678 scopus 로고    scopus 로고
    • Cyclodextrins and carrier systems
    • DOI 10.1016/S0168-3659(99)00046-2, PII S0168365999000462
    • D Duchene D Wouessidjewe G Poncel 1999 Cyclodextrins and carrier systems J. Control. Release 62 263 268 10.1016/S0168-3659(99)00046-2 1:CAS:528:DyaK1MXmsV2qs7k%3D (Pubitemid 29486506)
    • (1999) Journal of Controlled Release , vol.62 , Issue.1-2 , pp. 263-268
    • Duchene, D.1    Wouessidjewe, D.2    Ponchel, G.3
  • 12
    • 0032055148 scopus 로고    scopus 로고
    • Rheological evaluation of poloxamer as an in situ gel for ophthalmic use
    • DOI 10.1016/S0928-0987(97)00075-4, PII S0928098797000754
    • K Edsman J Carlfors R Petersson 1998 Rheological evaluation of poloxamer as an in situ gel for ophthalmic use Eur. J. Pharm. Sci. 6 105 112 10.1016/S0928-0987(97)00075-4 1:CAS:528:DyaK1cXhsFejt74%3D (Pubitemid 28164280)
    • (1998) European Journal of Pharmaceutical Sciences , vol.6 , Issue.2 , pp. 105-112
    • Edsman, K.1    Carlfors, J.2    Petersson, R.3
  • 13
    • 0031080653 scopus 로고    scopus 로고
    • Quinoline antimalarials: Mechanisms of action and resistance
    • DOI 10.1016/S0020-7519(96)00152-X, PII S002075199600152X
    • M Foley L Tilley 1997 Qinghaosu (artemisinin): an antimalarial drug from China Int. J. Parasitol. 27 213 10.1016/S0020-7519(96)00152-X (Pubitemid 27139713)
    • (1997) International Journal for Parasitology , vol.27 , Issue.2 , pp. 231-240
    • Foley, M.1    Tilley, L.2
  • 14
    • 21344453274 scopus 로고    scopus 로고
    • Nasal drug administration: Potential for targeted central nervous system delivery
    • DOI 10.1002/jps.20318
    • CL Graff GM Pollack 2005 Nasal drug administration: potential for targeted central nervous system delivery J. Pharm. Sci. 94 1187 1195 10.1002/jps.20318 1:CAS:528:DC%2BD2MXkvF2qt7Y%3D (Pubitemid 40904183)
    • (2005) Journal of Pharmaceutical Sciences , vol.94 , Issue.6 , pp. 1187-1195
    • Graff, C.L.1    Pollack, G.M.2
  • 15
    • 0037033989 scopus 로고    scopus 로고
    • Malaria in 2002
    • DOI 10.1038/415670a
    • B Greenwood T Mutabingwa 2002 Malaria in 2002 Nature 415 670 672 10.1038/415670a 1:CAS:528:DC%2BD38XhsVCjtrg%3D (Pubitemid 34136399)
    • (2002) Nature , vol.415 , Issue.6872 , pp. 670-672
    • Greenwood, B.1    Mutabingwa, T.2
  • 16
    • 79956006640 scopus 로고    scopus 로고
    • Temperature induced in situ mucoadhesive gel of Tramadol hydrochlioride for nasal drug delivery
    • 1:CAS:528:DC%2BD2sXhtFOnsbjF
    • ID Gonjari PV Kasture 2007 Temperature induced in situ mucoadhesive gel of Tramadol hydrochlioride for nasal drug delivery J. Pharm. Res. 6 2 89 93 1:CAS:528:DC%2BD2sXhtFOnsbjF
    • (2007) J. Pharm. Res. , vol.6 , Issue.2 , pp. 89-93
    • Gonjari, I.D.1    Kasture, P.V.2
  • 17
    • 21844459973 scopus 로고    scopus 로고
    • 2-Hydroxypropyl-β-cyclodextrin (HP-β-CD): A toxicology review
    • DOI 10.1016/j.fct.2005.03.007, PII S0278691505001006
    • S Gould RC Scott 2005 2-Hydroxypropyl-β-cyclodextrin (HP-β-CD): a toxicology review Food Chem. Toxicol. 43 1451 10.1016/j.fct.2005.03.007 1:CAS:528:DC%2BD2MXmt1eiu78%3D (Pubitemid 40961909)
    • (2005) Food and Chemical Toxicology , vol.43 , Issue.10 , pp. 1451-1459
    • Gould, S.1    Scott, R.C.2
  • 19
    • 0031054513 scopus 로고    scopus 로고
    • Pharmaceutical applications of cyclodextrins. III. Toxicological issues and safety evaluation
    • DOI 10.1021/js960213f
    • T Irie K Uekama 1997 Pharmaceutical applications of cyclodextrins. III. Toxicological issues and safety evaluation J. Pharm. Sci. 86 147 10.1021/js960213f 1:CAS:528:DyaK2sXhtVOgsLY%3D (Pubitemid 27078377)
    • (1997) Journal of Pharmaceutical Sciences , vol.86 , Issue.2 , pp. 147-162
    • Irie, T.1    Uekama, K.2
  • 20
    • 34548725661 scopus 로고    scopus 로고
    • A novel nasal delivery system of a Chinese traditional medicine, Radix Bupleuri, based on the concept of ion-activated in situ gel
    • Jiang, X., et al.: A novel nasal delivery system of a Chinese traditional medicine, Radix Bupleuri, based on the concept of ion-activated in situ gel. Arch. Pharm. Res. 30(8), 1014-1019 (2007). http://apr.psk.or.kr
    • (2007) Arch. Pharm. Res. , vol.30 , Issue.8 , pp. 1014-1019
    • Jiang, X.1
  • 22
    • 79956009474 scopus 로고
    • Nasal compositions
    • US Patent: 4,885,305
    • Kiechel, J. R., Malmison, R.: Nasal compositions. US Patent: 4,885,305 (1989)
    • (1989)
    • Kiechel, J.R.1    Malmison, R.2
  • 23
    • 0021948029 scopus 로고
    • Qinghaosu (artemisinin). An antimalarial drug from China
    • Klayman, D.: Qinghaosu (artemisinin). An antimalarial drug from China. Science 228, 1049-1055 (1989)
    • (1989) Science , vol.228 , pp. 1049-1055
    • Klayman, D.1
  • 24
    • 0029819323 scopus 로고    scopus 로고
    • Pharmaceutical applications of cyclodextrins. 1. Drug solubilization and stabilization
    • DOI 10.1021/js950534b
    • T Loftsson ME Brewster 1996 Pharmaceutical applications of cyclodextrins. 1. Drug solubilization and stabilization J. Pharm. Sci. 85 1017 1025 10.1021/js950534b 1:CAS:528:DyaK28XlsFSrsr4%3D (Pubitemid 26338912)
    • (1996) Journal of Pharmaceutical Sciences , vol.85 , Issue.10 , pp. 1017-1025
    • Loftsson, T.1    Brewster, M.E.2
  • 25
    • 0344286485 scopus 로고    scopus 로고
    • Cyclodextrins in ophthalmic drug delivery
    • DOI 10.1016/S0169-409X(98)00055-6, PII S0169409X98000556
    • T Loftsson T Järvinen 1999 Cyclodextrins in ophthalmic drug delivery Adv. Drug Deliv. Rev. 36 59 10.1016/S0169-409X(98)00055-6 (Pubitemid 29074477)
    • (1999) Advanced Drug Delivery Reviews , vol.36 , Issue.1 , pp. 59-79
    • Loftssona, T.1    Jarvinen, T.2
  • 26
    • 0037218147 scopus 로고    scopus 로고
    • Cerebral malaria: Optimising management
    • DOI 10.2165/00023210-200317030-00002
    • JL Maggs LPD Bishop G Edwards PM O'Neill SA Ward PA Winstanley N Mturi CO Musumba BM Wamola BR Ogutu CR Newton 2003 Cerebral malaria: optimising management CNS Drugs 17 153 165 10.2165/00023210-200317030-00002 (Pubitemid 36286532)
    • (2003) CNS Drugs , vol.17 , Issue.3 , pp. 153-165
    • Mturi, N.1    Musumba, C.O.2    Wamola, B.M.3    Ogutu, B.R.4    Newton, C.R.J.C.5
  • 27
    • 33747670237 scopus 로고    scopus 로고
    • Thermoreversible-mucoadhesive gel for nasal delivery of Sumatriptan
    • Murthy, R. S. R., Majithiya, R. J., Ghosh P. K.: Thermoreversible- mucoadhesive gel for nasal delivery of Sumatriptan. AAPS PharmSciTech. 7(3), E1-E7 (2006). ( http://www.aapspharmscitech.org )
    • (2006) AAPS PharmSciTech. , vol.7 , Issue.3
    • Murthy, R.S.R.1    Majithiya, R.J.2    Ghosh, P.K.3
  • 29
    • 3843071010 scopus 로고    scopus 로고
    • In situ-forming hydrogels - Review of temperature-sensitive systems
    • DOI 10.1016/j.ejpb.2004.03.019, PII S0939641104000876
    • E Ruel-Gariepy JC Leroux 2004 In situ forming hydrogels-review of temperature- sensitive systems Eur. J. Pharm. Biopharm. 58 409 426 10.1016/j.ejpb.2004.03.019 1:CAS:528:DC%2BD2cXmsVGnsL8%3D (Pubitemid 39037244)
    • (2004) European Journal of Pharmaceutics and Biopharmaceutics , vol.58 , Issue.2 , pp. 409-426
    • Ruel-Gariepy, E.1    Leroux, J.-C.2
  • 30
    • 77957939117 scopus 로고    scopus 로고
    • New simple and economical spectrophotometric method for estimation of artemether in pharmaceutical dosage forms
    • Shrivastava A., Nagori B.P., Saini P, Issarani R., Gaur S.S.: New simple and economical spectrophotometric method for estimation of artemether in pharmaceutical dosage forms. Asian J. Res. Chem. 1, 19-21 (2008)
    • (2008) Asian J. Res. Chem. , vol.1 , pp. 19-21
    • Shrivastava, A.1    Nagori, B.P.2    Saini, P.3    Issarani, R.4    Gaur, S.S.5
  • 31
    • 3542998669 scopus 로고    scopus 로고
    • Nasal route and drug delivery systems
    • DOI 10.1023/B:PHAR.0000026823.82950.ff
    • S Türker E Onur Y Ö zur 2004 Nasal route and drug delivery systems Pharm. World Sci. 26 137 142 10.1023/B:PHAR.0000026823.82950.ff (Pubitemid 39012580)
    • (2004) Pharmacy World and Science , vol.26 , Issue.3 , pp. 137-142
    • Turker, S.1    Onur, E.2    Ozer, Y.3
  • 32
    • 0032119526 scopus 로고    scopus 로고
    • Cyclodextrin drug carrier systems
    • 10.1021/cr970025p 1:CAS:528:DyaK1cXksV2itr0%3D
    • K Uekama F Hirayama T Irie 1998 Cyclodextrin drug carrier systems Chem. Rev. 98 2045 10.1021/cr970025p 1:CAS:528:DyaK1cXksV2itr0%3D
    • (1998) Chem. Rev. , vol.98 , pp. 2045
    • Uekama, K.1    Hirayama, F.2    Irie, T.3
  • 33
    • 0035845756 scopus 로고    scopus 로고
    • Effect of sodium chloride on the gelation temperature, gel strength and bioadhesive force of poloxamer gels containing diclofenac sodium
    • DOI 10.1016/S0378-5173(01)00809-2, PII S0378517301008092
    • CS Yong JS Choi JD Rhee 2001 Effect of sodium chloride on the gelation temperature, gel strength, and bioadhesive force of poloxamer gels containing diclofenac sodium Int. J. Pharm. 226 195 205 10.1016/S0378-5173(01)00809-2 1:CAS:528:DC%2BD3MXmsV2jtrw%3D (Pubitemid 32800794)
    • (2001) International Journal of Pharmaceutics , vol.226 , Issue.1-2 , pp. 195-205
    • Yong, C.S.1    Choi, J.S.2    Quan, Q.-Z.3    Rhee, J.-D.4    Kim, C.-K.5    Lim, S.-J.6    Kim, K.-M.7    Oh, P.-S.8    Choi, H.-G.9


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.