메뉴 건너뛰기




Volumn 34, Issue 1, 2011, Pages 51-57

Solubility enhancement and physicochemical characterization of carvedilol solid dispersion with Gelucire 50/13

Author keywords

Carvedilol; Dissolution; Gelucire; Solid dispersion

Indexed keywords

CARVEDILOL; GELUCIRE;

EID: 79955055728     PISSN: 02536269     EISSN: 19763786     Source Type: Journal    
DOI: 10.1007/s12272-011-0106-3     Document Type: Article
Times cited : (52)

References (28)
  • 2
    • 0030016875 scopus 로고    scopus 로고
    • Characterization of glyburide-polyethylene glycol solid dispersions
    • G. V. Betageri K. R. Makarla 1996 Characterization of glyburide-polyethylene glycol solid dispersion Drug Dev. Ind. Pharm. 22 731 734 10.3109/03639049609063230 1:CAS:528:DyaK28XktVars7c%3D (Pubitemid 26245761)
    • (1996) Drug Development and Industrial Pharmacy , vol.22 , Issue.7 , pp. 731-734
    • Betageri, G.V.1    Makarla, K.R.2
  • 3
    • 27744532687 scopus 로고    scopus 로고
    • Preparation and characterization of etoricoxib solid dispersions using lipid carriers by spray drying technique
    • DOI 10.1208/pt060350
    • B. Chauhan S. Shimpi A. Paradkar 2005 Preparation and characterization of etoricoxib solid dispersions using lipid carriers by spray drying technique AAPS PharmSciTech 6 E405 E412 16353998 10.1208/pt060350 (Pubitemid 41631777)
    • (2005) AAPS PharmSciTech , vol.6 , Issue.3 , pp. 50
    • Chauhan, B.1    Shimpi, S.2    Paradkar, A.3
  • 4
    • 0015124656 scopus 로고
    • Pharmaceutical applications of solid dispersion system
    • 4935981 10.1002/jps.2600600902 1:STN:280:DyaE3M3otFersQ%3D%3D
    • W. L. Chiou S. Riegelman 1971 Pharmaceutical applications of solid dispersion system J. Pharm. Sci. 60 1281 1302 4935981 10.1002/jps.2600600902 1:STN:280:DyaE3M3otFersQ%3D%3D
    • (1971) J. Pharm. Sci. , vol.60 , pp. 1281-1302
    • Chiou, W.L.1    Riegelman, S.2
  • 5
    • 0034032146 scopus 로고    scopus 로고
    • Physicochemical characterization of solid dispersions of the antiviral agent UC-781 with polyethylene glycol 6000 and Gelucire 44/14
    • DOI 10.1016/S0928-0987(00)00084-1, PII S0928098700000841
    • F. Damian N. Blaton L. Naesens J. Balzarini R. Kinget P. Augustijns G. Van den Mooter 2000 Physicochemical characterization of solid dispersions of the antiviral agent UC-781 with polyethylene glycol 6000 and Gelucire 44/14 Eur. J. Pharm. Sci. 10 311 322 10838021 10.1016/S0928-0987(00)00084-1 1:CAS:528:DC%2BD3cXjs1Cgs78%3D (Pubitemid 30317467)
    • (2000) European Journal of Pharmaceutical Sciences , vol.10 , Issue.4 , pp. 311-322
    • Damian, F.1    Blaton, N.2    Naesens, L.3    Balzarini, J.4    Kinget, R.5    Augustijns, P.6    Van Den Mooter, G.7
  • 6
    • 0030843847 scopus 로고    scopus 로고
    • Carvedilol. A reappraisal of its pharmacological properties and therapeutic use in cardiovascular disorders
    • C. J. Dunn A. P. Lea A. J. Wagstaff 1997 Carvedilol-a reappraisal of its pharmacological properties and therapeutic use in cardiovascular disorders Drugs. 54 161 185 9211087 10.2165/00003495-199754010-00015 1:CAS:528: DyaK2sXks1eisbc%3D (Pubitemid 27300048)
    • (1997) Drugs , vol.54 , Issue.1 , pp. 161-185
    • Dunn, C.J.1    Lea, A.P.2    Wagstaff, A.J.3
  • 8
    • 0035964448 scopus 로고    scopus 로고
    • Dissolution properties and anticonvulsant activity of phenytoin-polyethylene glycol 6000 and -polyvinylpyrrolidone K-30 solid dispersions
    • DOI 10.1016/S0378-5173(01)00751-7, PII S0378517301007517
    • M. Franco G. Trapani A. Latrofa C. Tullio M. R. Provenzano M. Serra M. Muggironi G. Biggio G. Liso 2001 Dissolution properties and anticonvulsant activity of phenytoin polyethylene glycol 6000 and -polyvinylpyrrolidone K-30 solid dispersions Int. J. Pharm. 225 63 73 11489555 10.1016/S0378-5173(01)00751- 7 1:CAS:528:DC%2BD3MXlslant7g%3D (Pubitemid 32728200)
    • (2001) International Journal of Pharmaceutics , vol.225 , Issue.1-2 , pp. 63-73
    • Franco, M.1    Trapani, G.2    Latrofa, A.3    Tullio, C.4    Provenzano, M.R.5    Serra, M.6    Muggironi, M.7    Biggio, G.8    Liso, G.9
  • 9
    • 0034928006 scopus 로고    scopus 로고
    • Enhancement of ibuprofen dissolution via wet granulation with β-cyclodextrin
    • DOI 10.1081/PDT-100002611
    • M. K. Ghorab M. C. Adeyeye 2001 Enhancement of ibuprofen, dissolution via wet granulation with beta-cyclodextrin Pharm. Dev. Technol. 6 305 314 11485172 10.1081/PDT-100002611 1:CAS:528:DC%2BD3MXls1Wms7o%3D (Pubitemid 32678236)
    • (2001) Pharmaceutical Development and Technology , vol.6 , Issue.3 , pp. 305-314
    • Ghorab, M.K.1    Adeyeye, M.C.2
  • 10
    • 0030638567 scopus 로고    scopus 로고
    • Characteristics and significance of the amorphous state in pharmaceutical systems
    • 9002452 10.1021/js9601896 1:CAS:528:DyaK28XntlOqt7k%3D
    • B. C. Hancock G. Zografi 1997 Characteristics and significance of the amorphous state in pharmaceutical systems J. Pharm. Sci. 86 1 12 9002452 10.1021/js9601896 1:CAS:528:DyaK28XntlOqt7k%3D
    • (1997) J. Pharm. Sci. , vol.86 , pp. 1-12
    • Hancock, B.C.1    Zografi, G.2
  • 11
    • 23844542459 scopus 로고    scopus 로고
    • Effect of solubilizing and microemulsifying excipients in polyethylene glycol 6000 solid dispersion on enhanced dissolution and bioavailability of ketoconazole
    • M. Y. Heo Z. Z. Piao T. W. Kim Q. R. Cao A. Kim B. J. Lee 2005 Effect of solubilizing and microemulsifying excipients in polyethylene glycol 6000 solid dispersion on enhanced dissolution and bioavailability of ketoconazole Arch. Pharm. Res. 28 604 611 15974450 10.1007/BF02977766 1:CAS:528: DC%2BD2MXltVamtbw%3D (Pubitemid 44698739)
    • (2005) Archives of Pharmacal Research , vol.28 , Issue.5 , pp. 604-611
    • Heo, M.-Y.1    Piao, Z.-Z.2    Kim, T.-W.3    Cao, Q.-R.4    Kim, A.5    Lee, B.-J.6
  • 13
    • 0028326530 scopus 로고
    • Effect of polyvinylpyrrolidone on the crystallinity and dissolution rate of solid dispersions of the antiinflammatory CI-987
    • DOI 10.1016/0378-5173(94)90192-9
    • A. S. Kearney D. L. Gabriel S. C. Mehta G. W. Radebaugh 1994 Effect of polyvinyl pyrrolidone on the crystallinity and dissolution rate of solid dispersions of the anti-inflammatory Ci-987 Int. J. Pharm. 104 169 174 10.1016/0378-5173(94)90192-9 1:CAS:528:DyaK2cXisFeitbg%3D (Pubitemid 24073701)
    • (1994) International Journal of Pharmaceutics , vol.104 , Issue.2 , pp. 169-174
    • Kearney, A.S.1    Gabriel, D.L.2    Mehta, S.C.3    Radebaugh, G.W.4
  • 14
    • 0031748005 scopus 로고    scopus 로고
    • Preparation, characterization, and dissolution studies of ibuprofen solid dispersions using polyethylene glycol (PEG), talc, and PEG-talc as dispersion carriers
    • G. M. Khan Z. Jiabi 1998 Preparation, characterization, and dissolution studies of ibuprofen solid dispersions using polyethylene glycol (PEG), talc, and PEG-talc as dispersion carriers Drug Dev. Ind. Pharm. 24 455 462 9876608 10.3109/03639049809085643 1:CAS:528:DyaK1cXjt1eqsrs%3D (Pubitemid 28273136)
    • (1998) Drug Development and Industrial Pharmacy , vol.24 , Issue.5 , pp. 455-462
    • Khan, G.M.1    Jiabi, Z.2
  • 15
    • 0016422844 scopus 로고
    • The concept of dissolution efficiency
    • 235616 1:CAS:528:DyaE2MXhsVCru7o%3D
    • K. A. Khan 1975 The concept of dissolution efficiency J. Pharm. Pharmacol. 27 48 49 235616 1:CAS:528:DyaE2MXhsVCru7o%3D
    • (1975) J. Pharm. Pharmacol. , vol.27 , pp. 48-49
    • Khan, K.A.1
  • 16
    • 0344440911 scopus 로고    scopus 로고
    • The influence of drug incorporation on the structure and release properties of solid dispersions in lipid matrices
    • DOI 10.1016/j.jconrel.2003.09.006
    • N. Khan D. Q. Craig 2003 The influence of drug incorporation on the structure and release properties of solid dispersions in the lipid matrices J. Control. Release 93 355 368 14644585 10.1016/j.jconrel.2003.09.006 1:CAS:528:DC%2BD3sXptlCmsLg%3D (Pubitemid 37485957)
    • (2003) Journal of Controlled Release , vol.93 , Issue.3 , pp. 355-368
    • Khan, N.1    Craig, D.Q.M.2
  • 17
    • 0035966510 scopus 로고    scopus 로고
    • Preparation and evaluation of biphenyl dimethyl dicarboxylate microemulsions for oral delivery
    • DOI 10.1016/S0168-3659(00)00343-6, PII S0168365900003436
    • C. K. Kim Y. J. Cho Z. G. Gao 2001 Preparation and evaluation of biphenyl dimethyl dicarboxylate microemulsions for oral delivery J. Control. Release 70 149 155 11166415 10.1016/S0168-3659(00)00343-6 1:CAS:528:DC%2BD3MXovV2quw%3D%3D (Pubitemid 32144799)
    • (2001) Journal of Controlled Release , vol.70 , Issue.1-2 , pp. 149-155
    • Kim, C.-K.1    Cho, Y.-J.2    Gao, Z.-G.3
  • 18
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • DOI 10.1016/S0939-6411(00)00076-X, PII S093964110000076X
    • C. Leuner J. Dressman 2000 Improving drug solubility for oral delivery using solid dispersions Eur. J. Pharm. Biopharm. 50 47 60 10840192 10.1016/S0939-6411(00)00076-X 1:CAS:528:DC%2BD3cXjslyju7c%3D (Pubitemid 30326688)
    • (2000) European Journal of Pharmaceutics and Biopharmaceutics , vol.50 , Issue.1 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 20
    • 27444438012 scopus 로고    scopus 로고
    • The effect of type and concentration of vehicles on the dissolution rate of a poorly soluble drug (indomethacin) from liquisolid compacts
    • A. Nokhodchi Y. Javadzadeh M. R. Siahi-Shadbad M. Barzegar-Jalali 2005 The effect of type and concentration of vehicles on dissolution rates of a poorly water soluble drug (indomethacin) from liquisolid compacts J. Pharm. Pharm. Sci. 8 18 25 15946594 1:CAS:528:DC%2BD2MXivVCgsb8%3D (Pubitemid 41528866)
    • (2005) Journal of Pharmacy and Pharmaceutical Sciences , vol.8 , Issue.1 , pp. 18-25
    • Nokhodchi, A.1    Javadzadeh, Y.2    Siahi-Shadbad, M.R.3    Barzegar-Jalali, M.4
  • 23
    • 0034495414 scopus 로고    scopus 로고
    • Solid dispersions of carbamazepine with Gelucire 44/14 and 50/13
    • B. Perissutti F. Rubessa F. Princivalle 2000 Solid dispersions of carbamazepine with Gelucire 44/14 and 50/13 STP Pharma Sci. 10 479 484 1:CAS:528:DC%2BD3MXot1Wjug%3D%3D (Pubitemid 32103932)
    • (2000) S.T.P. Pharma Sciences , vol.10 , Issue.6 , pp. 479-484
    • Perissutti, B.1    Rubessa, F.2    Princivalle, F.3
  • 24
    • 63049125218 scopus 로고    scopus 로고
    • Preparation and characterization of inclusion complexes of carvedilol with methyl-bcyclodextrin
    • 10.1007/s10847-008-9506-5
    • H. Rajashree K. Vilasrao 2009 Preparation and characterization of inclusion complexes of carvedilol with methyl-bcyclodextrin J. Incl. Phenom. Macrocyclic Chem. 63 219 224 10.1007/s10847-008-9506-5
    • (2009) J. Incl. Phenom. Macrocyclic Chem. , vol.63 , pp. 219-224
    • Rajashree, H.1    Vilasrao, K.2
  • 25
    • 0026754564 scopus 로고
    • Carvedilol: A novel cardiovascular drug with multiple actions
    • 10.1111/j.1527-3466.1992.tb00242.x 1:CAS:528:DyaK3sXksw%3D%3D
    • R. R. Ruffolo D. A. Boyle D. P. Brooks 1992 Carvedilol: a novel cardiovascular drug with multiple actions Cardiovasc. Drug Rev. 10 127 157 10.1111/j.1527-3466.1992.tb00242.x 1:CAS:528:DyaK3sXksw%3D%3D
    • (1992) Cardiovasc. Drug Rev. , vol.10 , pp. 127-157
    • Ruffolo, R.R.1    Boyle, D.A.2    Brooks, D.P.3
  • 26
    • 46349099994 scopus 로고    scopus 로고
    • Effect of hydroxylpropyl-β-cyclodextrin on solubility of carvedilol
    • DOI 10.4103/0250-474X.41470
    • B. D. Shewale N. P. Sapkal N. A. Raut N. J. Gaikwad H. R. Fursule 2008 Effect of hydroxyl propyl-β-cyclodextrinon solubility of carvedilol Indian J. Pharm. Sci. 70 255 257 20046727 10.4103/0250-474X.41470 1:STN:280: DC%2BC3c%2FgtlGltw%3D%3D (Pubitemid 351920211)
    • (2008) Indian Journal of Pharmaceutical Sciences , vol.70 , Issue.2 , pp. 255-257
    • Shewale, B.1    Sapkal, N.2    Raut, N.3    Gaikwad, N.4    Fursule, R.5
  • 27
    • 25144511900 scopus 로고    scopus 로고
    • Stabilization and improved in vivo performance of amorphous etoricoxib using Gelucire 50/13
    • DOI 10.1007/s11095-005-6694-1
    • S. L. Shimpi B. Chauhan K. R. Mahadik A. Paradkar 2005 Stabilization and improved in vivo performance of amorphous Etoricoxib using Gelucire 50/13 Pharm. Res. 22 1727 1734 16180131 10.1007/s11095-005-6694-1 1:CAS:528: DC%2BD2MXhtVent7vJ (Pubitemid 41355913)
    • (2005) Pharmaceutical Research , vol.22 , Issue.10 , pp. 1727-1734
    • Shimpi, S.L.1    Chauhan, B.2    Mahadik, K.R.3    Paradkar, A.4
  • 28
    • 0842346346 scopus 로고    scopus 로고
    • Preparation and study the 1:2 inclusion complex of carvedilol with β-cyclodextrin
    • DOI 10.1016/S0731-7085(03)00576-4
    • X. Wen F. Tan Z. Jing Z. Liu 2004 Preparation and study the 1:2 inclusion complex of carvedilol with cyclodextrin J. Pharm. Biomed. Anal. 34 517 523 15127807 10.1016/S0731-7085(03)00576-4 1:CAS:528:DC%2BD2cXptFehuw%3D%3D (Pubitemid 38177341)
    • (2004) Journal of Pharmaceutical and Biomedical Analysis , vol.34 , Issue.3 , pp. 517-523
    • Wen, X.1    Tan, F.2    Jing, Z.3    Liu, Z.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.