Development of a phosphatase-resistant, l-tyrosine derived LPA1/LPA3 dual antagonist

MedChemComm

Volumn 2, Issue 4, 2011, Pages 325-330

  East, James E ^a   Carter, Karen M ^a   Kennedy, Perry C ^b   Schulte, Nancy A ^c   Toews, Myron L ^c   Lynch, Kevin R ^b   MacDonald, Timothy L ^a  

^a UNIVERSITY OF VIRGINIA   (United States)

^b UNIVERSITY OF VIRGINIA   (United States)

^c NEBRASKA MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA FLUOROMETHYLENE; ALPHA FLUOROVINYL PHOSPHONIC ACID DERIVATIVE; ALPHA HYDROXYMETHYLENE; LYSOPHOSPHATIDIC ACID RECEPTOR; LYSOPHOSPHATIDIC ACID RECEPTOR 1; LYSOPHOSPHATIDIC ACID RECEPTOR 3; PHOSPHATASE; PHOSPHONIC ACID DERIVATIVE; UNCLASSIFIED DRUG; VINYL PHOSPHONIC ACID DERIVATIVE; VPC 51098; VPC 51299;

ANIMAL EXPERIMENT; ARTICLE; CALCIUM MOBILIZATION; CALCIUM TRANSPORT; CONCENTRATION RESPONSE; DRUG HALF LIFE; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; NONHUMAN; PRIORITY JOURNAL; RAT;

RATTUS;

EID: 79953905199     PISSN: 20402503     EISSN: 20402511     Source Type: Journal    
DOI: 10.1039/c0md00273a     Document Type: Article

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