Synthesis and biological evaluation of phosphonic and thiophosphoric acid derivatives of lysophosphatidic acid

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 13, 2004, Pages 3473-3476

  Santos, Webster L ^c   Heasley, Brian H ^a   Jarosz, Renata ^b   Carter, Karen M ^a   Lynch, Kevin R ^b   Macdonald, Timothy L ^a  

^a UNIVERSITY OF VIRGINIA   (United States)

^b UNIVERSITY OF VIRGINIA   (United States)

^c HARVARD UNIVERSITY   (United States)

Author keywords

Lysophosphatidic acid; Phosphatase; Phosphonic acid; Thiophosphoric acid

Indexed keywords

ALPHA METHYLENE PHOSPHONATE; AMIDE; GUANOSINE TRIPHOSPHATE; LYSOPHOSPHATIDIC ACID; LYSOPHOSPHATIDIC ACID DERIVATIVE; N ACYLETHANOLAMIDE PHOSPHORIC ACID; N OLEOYLETHANOLAMIDE; PHOSPHONIC ACID DERIVATIVE; PHOSPHORIC ACID DERIVATIVE; PHOSPHOROTHIOIC ACID DERIVATIVE; SULFUR 35; UNCLASSIFIED DRUG;

ARTICLE; BINDING ASSAY; CELL PROLIFERATION; DRUG ACTIVITY; DRUG SCREENING; DRUG SYNTHESIS; ENDOTHELIUM CELL; MULTIGENE FAMILY; SUBSTITUTION REACTION;

AMIDES; ANIMALS; CELLS, CULTURED; LYSOPHOSPHOLIPIDS; OLEIC ACIDS; PHOSPHATES; PHOSPHORIC ACIDS; RADIOLIGAND ASSAY; RECEPTORS, LYSOPHOSPHATIDIC ACID; STEARIC ACIDS;

EID: 2942532893     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.04.061     Document Type: Article

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