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ChemMedChem

Volumn 6, Issue 4, 2011, Pages 725-736

Discovery of Benzamide Analogues as a Novel Class of 5-HT3 Receptor Agonists

(4) Jørgensen, Charlotte G a Frølund, Bente a Kehler, Jan b Jensen, Anders A a

a UNIVERSITY OF COPENHAGEN (Denmark)

b H LUNDBECK A S (Denmark)

Author keywords

Agonists; Allosterism; Benzamides; Ion channels; Serotonin type 3 receptors

Indexed keywords

BENZAMIDE DERIVATIVE; METOCLOPRAMIDE; SEROTONIN 3 AGONIST; SEROTONIN 3 RECEPTOR; TROPISETRON; ZACOPRIDE;

ALLOSTERISM; ARTICLE; CONCENTRATION RESPONSE; DRUG BINDING; DRUG DESIGN; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ALLOSTERIC SITE; BENZAMIDES; HEK293 CELLS; HUMANS; LIGANDS; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN RECEPTOR AGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 79953030312 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000444 Document Type: Article

Times cited : (13)

References (28)

1
- 44849104847
- D. E. Nichols, C. D. Nichols, Chem. Rev. 2008, 108, 1614-1641;
- (2008) Chem. Rev. , vol.108 , pp. 1614-1641
- Nichols, D.E.¹ Nichols, C.D.²

2
- 64549158645
- M. Berger, J. A. Gray, B. L. Roth, Annu. Rev. Med. 2009, 60, 355-366;
- (2009) Annu. Rev. Med. , vol.60 , pp. 355-366
- Berger, M.¹ Gray, J.A.² Roth, B.L.³

3
- 78650661080
- J. Walstab, G. Rappold, B. Niesler, Pharmacol. Ther. 2010, 128, 146-169.
- (2010) Pharmacol. Ther. , vol.128 , pp. 146-169
- Walstab, J.¹ Rappold, G.² Niesler, B.³

4
- 58049215463
- N. M. Barnes, T. G. Hales, S. C. R. Lummis, J. A. Peters, Neuropharmacology 2009, 56, 273-284;
- (2009) Neuropharmacology , vol.56 , pp. 273-284
- Barnes, N.M.¹ Hales, T.G.² Lummis, S.C.R.³ Peters, J.A.⁴

5
- 33947677144
- A. J. Thompson, S. C. R. Lummis, Expert Opin. Ther. Targets 2007, 11, 527-540;
- (2007) Expert Opin. Ther. Targets , vol.11 , pp. 527-540
- Thompson, A.J.¹ Lummis, S.C.R.²

6
- 50249105158
- A. A. Jensen, P. A. Davies, H. Bräuner-Osborne, K. Krzywkowski, Trends Pharmacol. Sci. 2008, 29, 437-444;
- (2008) Trends Pharmacol. Sci. , vol.29 , pp. 437-444
- Jensen, A.A.¹ Davies, P.A.² Bräuner-Osborne, H.³ Krzywkowski, K.⁴

7
- 33846245154
- W. Sieghart, Adv. Pharmacol. 2006, 54, 231-263;
- (2006) Adv. Pharmacol. , vol.54 , pp. 231-263
- Sieghart, W.¹

8
- 69949159308
- A. Taly, P. J. Corringer, D. Guedin, P. Lestage, J. P. Changeux, Nat. Rev. Drug Discovery 2009, 8, 733-750;
- (2009) Nat. Rev. Drug Discovery , vol.8 , pp. 733-750
- Taly, A.¹ Corringer, P.J.² Guedin, D.³ Lestage, P.⁴ Changeux, J.P.⁵

9
- 4644265039
- J. W. Lynch, Physiol. Rev. 2004, 84, 1051-1095.
- (2004) Physiol. Rev. , vol.84 , pp. 1051-1095
- Lynch, J.W.¹

10
- 34548677767
- D. Bertrand, M. Gopalakrishnan, Biochem. Pharmacol. 2007, 74, 1155-1163.
- (2007) Biochem. Pharmacol. , vol.74 , pp. 1155-1163
- Bertrand, D.¹ Gopalakrishnan, M.²

11
- 7744243992
- G. A. Patani, E. J. LaVoie, Chem. Rev. 1996, 96, 3147-3176.
- (1996) Chem. Rev. , vol.96 , pp. 3147-3176
- Patani, G.A.¹ LaVoie, E.J.²

12
- 0032697489
- A. E. Dubin, R. Huvar, M. R. D'Andrea, J. Pyati, J. Y. Zhu, K. C. Joy, S. J. Wilson, J. E. Galindo, C. A. Glass, L. Luo, M. R. Jackson, T. W. Lovenberg, M. G. Erlander, J. Biol. Chem. 1999, 274, 30799-30810;
- (1999) J. Biol. Chem. , vol.274 , pp. 30799-30810
- Dubin, A.E.¹ Huvar, R.² D'Andrea, M.R.³ Pyati, J.⁴ Zhu, J.Y.⁵ Joy, K.C.⁶ Wilson, S.J.⁷ Galindo, J.E.⁸ Glass, C.A.⁹ Luo, L.¹⁰ Jackson, M.R.¹¹ Lovenberg, T.W.¹² Erlander, M.G.¹³

13
- 27844502487
- K. L. Price, S. C. Lummis, J. Neurosci. Methods 2005, 149, 172-177;
- (2005) J. Neurosci. Methods , vol.149 , pp. 172-177
- Price, K.L.¹ Lummis, S.C.²

14
- 34247598903
- K. Krzywkowski, A. A. Jensen, C. N. Connolly, H. Brauner-Osborne, Pharmacogenet. Genomics 2007, 17, 255-266.
- (2007) Pharmacogenet. Genomics , vol.17 , pp. 255-266
- Krzywkowski, K.¹ Jensen, A.A.² Connolly, C.N.³ Brauner-Osborne, H.⁴

15
- 34648836438
- A. A. Jensen, D. P. Zlotos, T. Liljefors, J. Med. Chem. 2007, 50, 4616-4629.
- (2007) J. Med. Chem. , vol.50 , pp. 4616-4629
- Jensen, A.A.¹ Zlotos, D.P.² Liljefors, T.³

16
- 0025921597
- N. A. Sharif, E. H. Wong, D. N. Loury, E. Stefanich, A. D. Michel, R. M. Eglen, R. L. Whiting, Br. J. Pharmacol. 1991, 102, 919-925.
- (1991) Br. J. Pharmacol. , vol.102 , pp. 919-925
- Sharif, N.A.¹ Wong, E.H.² Loury, D.N.³ Stefanich, E.⁴ Michel, A.D.⁵ Eglen, R.M.⁶ Whiting, R.L.⁷

17
- 0035847383
- J. E. Macor, D. Gurley, T. Lanthorn, J. Loch, R. A. Mack, G. Mullen, O. Tran, N. Wright, J. C. Gordon, Bioorg. Med. Chem. Lett. 2001, 11, 319-321;
- (2001) Bioorg. Med. Chem. Lett. , vol.11 , pp. 319-321
- Macor, J.E.¹ Gurley, D.² Lanthorn, T.³ Loch, J.⁴ Mack, R.A.⁵ Mullen, G.⁶ Tran, O.⁷ Wright, N.⁸ Gordon, J.C.⁹

18
- 34247184782
- F. G. Boess, J. DeVry, C. Erb, T. Flessner, M. Hendrix, J. Luithle, C. Methfessel, B. Riedl, K. Schnizler, F. J. van der Staay, M. vanKampen, W. B. Wiese, G. Koenig, J. Pharmacol. Exp. Ther. 2007, 321, 716-725;
- (2007) J. Pharmacol. Exp. Ther. , vol.321 , pp. 716-725
- Boess, F.G.¹ DeVry, J.² Erb, C.³ Flessner, T.⁴ Hendrix, M.⁵ Luithle, J.⁶ Methfessel, C.⁷ Riedl, B.⁸ Schnizler, K.⁹ van der Staay, F.J.¹⁰ vanKampen, M.¹¹ Wiese, W.B.¹² Koenig, G.¹³

19
- 0032524624
- D. A. Gurley, T. H. Lanthorn, Neurosci. Lett. 1998, 247, 107-110;
- (1998) Neurosci. Lett. , vol.247 , pp. 107-110
- Gurley, D.A.¹ Lanthorn, T.H.²

20
- 0037020529
- L. M. Broad, C. Felthouse, R. Zwart, G. I. McPhie, K. H. Pearson, P. J. Craig, L. Wallace, R. J. Broadmore, J. R. Boot, M. Keenan, S. R. Baker, E. Sher, Eur. J. Pharmacol. 2002, 452, 137-144.
- (2002) Eur. J. Pharmacol. , vol.452 , pp. 137-144
- Broad, L.M.¹ Felthouse, C.² Zwart, R.³ McPhie, G.I.⁴ Pearson, K.H.⁵ Craig, P.J.⁶ Wallace, L.⁷ Broadmore, R.J.⁸ Boot, J.R.⁹ Keenan, M.¹⁰ Baker, S.R.¹¹ Sher, E.¹²

21
- 0037072311
- D. L. Beene, G. S. Brandt, W. Zhong, N. Zacharias, H. A. Lester, D. A. Dougherty, Biochemistry 2002, 41, 10262-10269;
- (2002) Biochemistry , vol.41 , pp. 10262-10269
- Beene, D.L.¹ Brandt, G.S.² Zhong, W.³ Zacharias, N.⁴ Lester, H.A.⁵ Dougherty, D.A.⁶

22
- 1842475289
- P. H. Celie, S. E. vanRossum-Fikkert, W. J. vanDijk, K. Brejc, A. B. Smit, T. K. Sixma, Neuron 2004, 41, 907-917;
- (2004) Neuron , vol.41 , pp. 907-917
- Celie, P.H.¹ vanRossum-Fikkert, S.E.² vanDijk, W.J.³ Brejc, K.⁴ Smit, A.B.⁵ Sixma, T.K.⁶

23
- 34547520128
- C. D. Dellisanti, Y. Yao, J. C. Stroud, Z. Z. Wang, L. Chen, Nat. Neurosci. 2007, 10, 953-962.
- (2007) Nat. Neurosci. , vol.10 , pp. 953-962
- Dellisanti, C.D.¹ Yao, Y.² Stroud, J.C.³ Wang, Z.Z.⁴ Chen, L.⁵

24
- 49949093837
- C. Rojas, M. Stathis, A. G. Thomas, E. B. Massuda, J. Alt, J. Zhang, E. Rubenstein, S. Sebastiani, S. Cantoreggi, S. H. Snyder, B. Slusher, Anesth. Analg. 2008, 107, 469-478.
- (2008) Anesth. Analg. , vol.107 , pp. 469-478
- Rojas, C.¹ Stathis, M.² Thomas, A.G.³ Massuda, E.B.⁴ Alt, J.⁵ Zhang, J.⁶ Rubenstein, E.⁷ Sebastiani, S.⁸ Cantoreggi, S.⁹ Snyder, S.H.¹⁰ Slusher, B.¹¹

25
- 9744261622
- M. S. Karadsheh, M. S. Shah, X. Tang, R. L. Macdonald, J. A. Stitzel, J. Neurochem. 2004, 91, 1138-1150;
- (2004) J. Neurochem. , vol.91 , pp. 1138-1150
- Karadsheh, M.S.¹ Shah, M.S.² Tang, X.³ Macdonald, R.L.⁴ Stitzel, J.A.⁵

26
- 0031595642
- Y. Xiao, E. L. Meyer, J. M. Thompson, A. Surin, J. Wroblewski, K. J. Kellar, Mol. Pharmacol. 1998, 54, 322-333;
- (1998) Mol. Pharmacol. , vol.54 , pp. 322-333
- Xiao, Y.¹ Meyer, E.L.² Thompson, J.M.³ Surin, A.⁴ Wroblewski, J.⁵ Kellar, K.J.⁶

27
- 13444291352
- D. Feuerbach, K. Lingenhohl, P. Dobbins, J. Mosbacher, N. Corbett, J. Nozulak, D. Hoyer, Neuropharmacology 2005, 48, 215-227.
- (2005) Neuropharmacology , vol.48 , pp. 215-227
- Feuerbach, D.¹ Lingenhohl, K.² Dobbins, P.³ Mosbacher, J.⁴ Corbett, N.⁵ Nozulak, J.⁶ Hoyer, D.⁷

28
- 77951236537
- A. A. Jensen, M. L. Bergmann, T. Sander, T. Balle, J. Biol. Chem. 2010, 285, 10141-10153.
- (2010) J. Biol. Chem. , vol.285 , pp. 10141-10153
- Jensen, A.A.¹ Bergmann, M.L.² Sander, T.³ Balle, T.⁴

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