Inhibition of recombinant L-type voltage-gated calcium channels by positive allosteric modulators of GABA A receptors

Journal of Pharmacology and Experimental Therapeutics

Volumn 337, Issue 1, 2011, Pages 301-311

  Earl, Damien E ^a   Tietz, Elizabeth I ^a  

^a MEDICAL COLLEGE OF OHIO   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3ALPHA HYDROXY 5ALPHA PREGNAN 20 ONE; 4 AMINOBUTYRIC ACID A RECEPTOR; ALCOHOL; AMINO ACID; BARIUM ION; CALCIUM CHANNEL BLOCKING AGENT; CALCIUM CHANNEL L TYPE; DEALKYLFLURAZEPAM; DIAZEPAM; DIHYDROPYRIDINE; FLURAZEPAM; GABAERGIC RECEPTOR AFFECTING AGENT; PENTOBARBITAL; RECOMBINANT PROTEIN; VOLTAGE GATED CALCIUM CHANNEL;

ALLOSTERISM; ANIMAL CELL; ARTICLE; BINDING AFFINITY; CALCIUM CURRENT; CELL STRAIN HEK293; CHEMICAL STRUCTURE; CONCENTRATION RESPONSE; CONTROLLED STUDY; HUMAN; HUMAN CELL; IC 50; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN EXPRESSION; RAT; STRUCTURAL HOMOLOGY; UPREGULATION;

ALLOSTERIC REGULATION; ANIMALS; BRAIN; CALCIUM CHANNEL BLOCKERS; CALCIUM CHANNELS, L-TYPE; GABA MODULATORS; HEK293 CELLS; HUMANS; RATS; RECEPTORS, GABA-A; RECOMBINANT PROTEINS;

EID: 79953017457     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.110.178244     Document Type: Article

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