Three-component reaction: Synthesis, characterization, and biological study of some fused bridgehead nitrogen heterocyclic systems containing 4-methylthiophenyl moiety

Phosphorus, Sulfur and Silicon and the Related Elements

Volumn 186, Issue 3, 2011, Pages 526-532

  Manjunatha, K ^a   Poojary, Boja ^a   Lobo, Prajwal L ^a   Kumari, N Suchetha ^b   Anoop, C ^c  

^a MANGALORE UNIVERSITY   (India)

^b NITTE DEEMED TO BE UNIVERSITY   (India)

^c Biocon Limited   (India)

Author keywords

1,2,4 triazole 5 thiol; 4 methylthiobenzyl; Anti inflammatory activity; antimicrobial activity; three component reaction

Indexed keywords

EID: 79952660803     PISSN: 10426507     EISSN: 15635325     Source Type: Journal    
DOI: 10.1080/10426507.2010.506454     Document Type: Article

References (29)

1. Beck, B.; Hess, S.; Domling, A. Bioorg. Med. Chem. Lett. 2000, 10, 1701-1705.
2. Lee, D.; Sello, J. K.; Schreiber, S. L. Org. Lett. 2000, 2, 709-712.
3. Lednicer, D.; Mitscher, L. A.; George, G. I. Organic Chemistry of Drug Synthesis, Vol. 4;Wiley, New York, 1990; pp. 95-97.
4. Rehman, M. Z.; Anwar, C. J.; Ahmad, S. Bull. Kor. Chem. Soc. 2005, 26, 1771-1775.
5. Knadlar, M. P.; Bergstrom, R. F.; Callaghan, J. T.; Rubin, A. Drug Metab. Dispos. 1986, 14, 175-182.
6. Vijaya Raj, K. K.; Narayana, B.; Ashalatha, B. V.; Kumari, N. S.; Sarojini, B.K. Eur. J. Med. Chem. 2007, 42, 425-429.
7. Holla, B. S.; Malini, K. V.; Rao, B. S.; Sarojini, B. K.; Kumari, N.S. Eur. J. Med. Chem. 2003, 38, 313-318.
8. Jiang, B. X.; Gu, H. Bioorg. Med. Chem. Lett. 2000, 8, 363-371.
9. Medime, E.; Capan, G. Il Farmaco, 1994, 49, 449-451.
10. Bordi, F.; Catellani, P. L.; Morinha, G.; Plazzi, P. V.; Silva, C.; Barocelli, E.; Chiavarini, M. Il Farmaco, 1989, 44, 795-805.
11. Lesyk, R.; Vladzimirska, O.; Holota, S.; Zaprutko, L.; Gzella, A. Eur. J. Med. Chem. 2007, 42, 641-648.
12. Karthikeyan, M. S. Eur. J. Med. Chem. 2009, 44, 827-833.
13. Tozkoparan, B.; Gokhan, N.; Aktay, G.; Yesilada, E.; Ertan. M. Eur. J. Med. Chem. 2000, 35, 743-750.
14. Ashok, M.; Holla, B. S.; Kumari, N.S. Eur. J. Med. Chem. 2007, 42, 380-385.
15. Walczak, K.; Gondela, A.; Suwinski, J. Eur. J. Med. Chem. 2004, 39, 849-853.
16. Kawashima, Y.; Ishikawa, H.; Kida, S.; Tanaka, T.; Masuda, T.; Japan Kokai, 1986, 61, 260085;
17. Chem. Abstr. 1987, 106, 138475.
18. Nagar, S.; Singh, H. H.; Sinha, J. N.; Parmar, S. S. J. Med. Chem. 1973, 16(2) , 178-180.
19. Prasad, D. J.; Ashok, M.; Karegoudar, P.; Poojary, B.; Holla, B. S.; Kumari, N. S. Eur.J. Med. Chem. 2009, 44, 551-557.
20. Karabasanagouda, T.; Adhikari, A. V.; Girisha, M. Indian J. Chem. 2009, 48B, 430-437.
21. Ashok, M.; Holla, B. S. Phosphorus, Sulfur Silicon Relat. Elem. 2007, 182, 1599-1608.
22. Karabasanagouda, T.; Adhikari, A. V.; Shetty, N. S. Phosphorus, Sulfur Silicon Relat. Elem. 2007, 182, 2925-2941.
23. Karthikeyan, M. S.; Holla, B. S. Monatsh. Chem. 2008, 139, 691-696.
24. Holla, B. S.; Malini, K. V.; Sarojini, B. K.; Poojary, B. Synth. Commun. 2005, 35, 333-340.
25. Winter, C. A.; Risley, E. A.; Nuss, G. W. Proc. Soc. Exp. Biol. Med. 1962, 111, 544.
26. Barry, A. L. In Antibiotics in Laboratory Medicine (V. L. Corian, Ed.) ; Williams and Wilkins: Baltimore, MD, 1991; p. 1.
27. MacLowry, J. D.; Jaqua, M. J.; Selepak, S. T. Appl. Microbiol. 1970, 20, 46-53.
28. Arthington-Skaggs, B. A.; Motley, M.;Warnock, D.W.;Morrison, C. J. J. Clin.Microbiol. 2000, 8, 2254-2260.
29. Verma, R. S.; Khan, Z. K.; Singh, A. P. (Eds.) . Antifungal Agent: Past, Present and Future Prospects; National Academy of Chemistry and Biology: Lucknow, India, 1986; p. 55.