메뉴 건너뛰기




Volumn 100, Issue 5, 2011, Pages 1805-1818

Tadalafil inclusion in microporous silica as effective dissolution enhancer: Optimization of loading procedure and molecular state characterization

Author keywords

Amorphous; Dissolution; Inclusions; Mathematical model; Solid state

Indexed keywords

SILICON DIOXIDE; TADALAFIL;

EID: 79952234982     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.22420     Document Type: Article
Times cited : (39)

References (52)
  • 1
    • 0036783940 scopus 로고    scopus 로고
    • Efficacy and safety of tadalafil for the treatment of erectile dysfunction: Results of integrated analysis
    • Brock GB, McMahon CG, Chen KK. 2002. Efficacy and safety of tadalafil for the treatment of erectile dysfunction: Results of integrated analysis. J Urol 168:1332-1336.
    • (2002) J Urol , vol.168 , pp. 1332-1336
    • Brock, G.1    Mcmahon, C.2    Chen, K.3
  • 2
    • 0036189959 scopus 로고    scopus 로고
    • Human PDE5A gene encodes three PDE5 isoforms from two alternate promoters
    • Lin CS, Chow S, Lau AR. 2002. Human PDE5A gene encodes three PDE5 isoforms from two alternate promoters. Int J Impot Res 14:15-24.
    • (2002) Int J Impot Res , vol.14 , pp. 15-24
    • Lin, C.1    Chow, S.2    Lau, A.3
  • 3
    • 61549092523 scopus 로고    scopus 로고
    • Tadalafil in the treatment of erectile dysfunction
    • Coward RM, Carson CC. 2008. Tadalafil in the treatment of erectile dysfunction. Ther Clin Risk Manag 4:315-329.
    • (2008) Ther Clin Risk Manag , vol.4 , pp. 315-329
    • Coward, R.1    Carson, C.2
  • 4
    • 78349304097 scopus 로고    scopus 로고
    • Biopharmaceutics classification system
    • Chavda HV, Patel CN, Anand IS. 2010. Biopharmaceutics classification system. Syst Rev Pharm 1:62-69.
    • (2010) Syst Rev Pharm , vol.1 , pp. 62-69
    • Chavda, H.1    Patel, C.2    Anand, I.3
  • 5
    • 35648976611 scopus 로고    scopus 로고
    • Phosphodiesterase type 5 inhibitors: State of the therapeutic class
    • Carson CC. 2007. Phosphodiesterase type 5 inhibitors: State of the therapeutic class. Urol Clin North Am 34:507-515.
    • (2007) Urol Clin North Am , vol.34 , pp. 507-515
    • Carson, C.1
  • 8
    • 78349312679 scopus 로고    scopus 로고
    • In sight into tadalafil-block copolymer binary solid dispersion: Mechanistic investigation of dissolution enhancement
    • Mehanna MM, Motawaa AM, Samaha MW, 2010. In sight into tadalafil-block copolymer binary solid dispersion: Mechanistic investigation of dissolution enhancement. Int J Pharm 402:78-88.
    • (2010) Int J Pharm , vol.402 , pp. 78-88
    • Mehanna, M.1    Motawaa, A.2    Samaha, M.3
  • 9
    • 27144527867 scopus 로고    scopus 로고
    • Functionalized SAB-15 material as carrier for controlled drug delivery: Influence of surface properties on matrix-drug interactions
    • Song S-W, Hidajat K, Kawi S. 2005. Functionalized SAB-15 material as carrier for controlled drug delivery: Influence of surface properties on matrix-drug interactions. Langmuir 21:9568-9575.
    • (2005) Langmuir , vol.21 , pp. 9568-9575
    • Song, S.-W.1    Hidajat, K.2    Kawi, S.3
  • 10
    • 3242720476 scopus 로고    scopus 로고
    • Fabrication of porous hollow silica nanoparticles and their applications in drug release control
    • Li Z, Wen L, Shao L, Chen J. 2004. Fabrication of porous hollow silica nanoparticles and their applications in drug release control. J Control Release 98:244-254.
    • (2004) J Control Release , vol.98 , pp. 244-254
    • Li, Z.1    Wen, L.2    Shao, L.3    Chen, J.4
  • 11
    • 0037769850 scopus 로고    scopus 로고
    • Multiple unit gastroretentive drug delivery systems: A new method for low density microparticles
    • Streubel A, Sipemann J, Bodmeier R. 2003. Multiple unit gastroretentive drug delivery systems: A new method for low density microparticles. J Microencapsul 20:329-347.
    • (2003) J Microencapsul , vol.20 , pp. 329-347
    • Streubel, A.1    Sipemann, J.2    Bodmeier, R.3
  • 12
    • 0343967746 scopus 로고
    • Controlled drug release by the use of porous calcium silicate
    • Murakami T, Yata N. 1995. Controlled drug release by the use of porous calcium silicate. Drug Del Syst 10:159-166.
    • (1995) Drug Del Syst , vol.10 , pp. 159-166
    • Murakami, T.1    Yata, N.2
  • 13
    • 11844283277 scopus 로고    scopus 로고
    • Effect of adsorbents on the absorption of lansoprazole with surfactant
    • Ito Y, Arai H, Uchino K, Iwasaki K, Shibata N, Takada K. 2005. Effect of adsorbents on the absorption of lansoprazole with surfactant. Int J Pharm 289:69-77.
    • (2005) Int J Pharm , vol.289 , pp. 69-77
    • Ito, Y.1    Arai, H.2    Uchino, K.3    Iwasaki, K.4    Shibata, N.5    Takada, K.6
  • 14
    • 0037057346 scopus 로고    scopus 로고
    • Use of commercial porous ceramic particles for sustained drug delivery
    • Byrne RS, Deasy PB. 2002. Use of commercial porous ceramic particles for sustained drug delivery. Int J Pharm. 246:61-73.
    • (2002) Int J Pharm. , vol.246 , pp. 61-73
    • Byrne, R.1    Deasy, P.2
  • 15
    • 30744434648 scopus 로고    scopus 로고
    • 3 microparticles and encapsulation by polyelectrolyte multilayer films for sustained drug delivery
    • 3 microparticles and encapsulation by polyelectrolyte multilayer films for sustained drug delivery. Int J Pharm 308:160-167.
    • (2006) Int J Pharm , vol.308 , pp. 160-167
    • Wang, C.1    He, C.2    Tong, Z.3    Liu, X.4    Ren, B.5
  • 16
    • 0004117882 scopus 로고    scopus 로고
    • Pharmaceutical experimental design
    • New York: Marcel Dekker Inc.
    • Lewis GA, Mathieu D, Phan-Tan-Luu R, Pharmaceutical experimental design. 1999, New York: Marcel Dekker Inc.
    • (1999)
    • Lewis, G.1    Mathieu, D.2    Phan-Tan-Luu, R.3
  • 17
    • 67049114625 scopus 로고    scopus 로고
    • Ciprofloxacin liposomes as vesicular reservoirs for ocular delivery: formulation, optimization, and in vitro characterization
    • Mehanna MM, Elmaradny HA, Samaha MS. 2009. Ciprofloxacin liposomes as vesicular reservoirs for ocular delivery: formulation, optimization, and in vitro characterization. Drug Dev Ind Pharm 35:583-593.
    • (2009) Drug Dev Ind Pharm , vol.35 , pp. 583-593
    • Mehanna, M.1    Elmaradny, H.2    Samaha, M.3
  • 20
    • 85031273713 scopus 로고    scopus 로고
    • Overview of modern design of experiments methods for computational simulations (AIAA 2003-0649)by American Institute of Aeronautics and Astronautics, Sandia National Laboratories. Albuquerque, New Mexico.
    • Giunta AA, Wojtkiewicz SF, Eldred MS. 2003. Overview of modern design of experiments methods for computational simulations (AIAA 2003-0649)by American Institute of Aeronautics and Astronautics, Sandia National Laboratories. Albuquerque, New Mexico.
    • (2003)
    • Giunta, A.1    Wojtkiewicz, S.2    Eldred, M.3
  • 21
    • 0037043107 scopus 로고    scopus 로고
    • In vitro evaluation of nimodipine permeation through human epidermis using response surface methodology
    • Giannakou SA, Dallas PP, Rekkas DM, Choulis NH. 2002. In vitro evaluation of nimodipine permeation through human epidermis using response surface methodology. Int J Pharm 241:27-34.
    • (2002) Int J Pharm , vol.241 , pp. 27-34
    • Giannakou, S.1    Dallas, P.2    Rekkas, D.3    Choulis, N.4
  • 22
    • 0004117882 scopus 로고    scopus 로고
    • Pharmaceutical experimental design
    • In, Swarbrick, J. Ed. New York: Marcel Dekker Inc.
    • Lewis GA, Mathieu D, Phan-Tan-Luu R. 1999. Response surface methodology. In Pharmaceutical experimental design., Swarbrick, J. Ed. New York: Marcel Dekker Inc., pp 185-246.
    • (1999) Response surface methodology , pp. 185-246
    • Lewis, G.1    Mathieu, D.2    Phan-Tan-Luu, R.3
  • 23
    • 0017857869 scopus 로고
    • Quantitative crystallinity determinations for beta-lactam antibiotics by solution calorimetry: Correlation with stability
    • Pikal MJ, Lukes AL, Lang JE, Gaines K. 1978. Quantitative crystallinity determinations for beta-lactam antibiotics by solution calorimetry: Correlation with stability. J Pharm Sci 67:767-773.
    • (1978) J Pharm Sci , vol.67 , pp. 767-773
    • Pikal, M.1    Lukes, A.2    Lang, J.3    Gaines, K.4
  • 24
    • 12444272525 scopus 로고
    • Adsorption of gases in multimolecular layers
    • Brunauer S, Emmet PH, Teller E. 1938. Adsorption of gases in multimolecular layers. J Am Chem Soc 60:309-319.
    • (1938) J Am Chem Soc , vol.60 , pp. 309-319
    • Brunauer, S.1    Emmet, P.2    Teller, E.3
  • 25
    • 0037104111 scopus 로고    scopus 로고
    • Critical appraisal of classical methods for determination of mesopore size distributions of MCM-41 materials
    • Choma J, Jaroniec M., Burakiewicz-Mortka W, Kloske M. 2002. Critical appraisal of classical methods for determination of mesopore size distributions of MCM-41 materials. Appl Surf Sci 196:216-223.
    • (2002) Appl Surf Sci , vol.196 , pp. 216-223
    • Choma, J.1    Jaroniec, M.2    Burakiewicz-Mortka, W.3    Kloske, M.4
  • 26
    • 0032668615 scopus 로고    scopus 로고
    • Standard nitrogen adsorption data for characterization of nanoporous silica
    • Jaroniec M, Kruk M, Olivier JP. 1999. Standard nitrogen adsorption data for characterization of nanoporous silica. Langmuir 15:5410-5413.
    • (1999) Langmuir , vol.15 , pp. 5410-5413
    • Jaroniec, M.1    Kruk, M.2    Olivier, J.3
  • 27
    • 85031239426 scopus 로고    scopus 로고
    • Guidance for industry Q1A stability testing of new drug substances and products, at U.S. Department of Health and Human Services Food and Drug administration.
    • Guidance for industry Q1A stability testing of new drug substances and products, at 2010, U.S. Department of Health and Human Services Food and Drug administration.
    • (2010)
  • 28
    • 77955308221 scopus 로고    scopus 로고
    • Template occluded SBA-15: An effective dissolution enhancer for poorly water-soluble drug
    • Tingming F, Liwei G, Kang L, Tianyao W, Jin L. 2010. Template occluded SBA-15: An effective dissolution enhancer for poorly water-soluble drug. Appl Surf Sci 256:6963-6968.
    • (2010) Appl Surf Sci , vol.256 , pp. 6963-6968
    • Tingming, F.1    Liwei, G.2    Kang, L.3    Tianyao, W.4    Jin, L.5
  • 29
    • 0034988419 scopus 로고    scopus 로고
    • Comparative studies of the enhancing effects of cyclodextrins on the solubility and oral bioavailability of tacrolimus in rats
    • Arima H, Yunomae K, Miyake K, Irie T, Hirayama F, Uekama K, 2001. Comparative studies of the enhancing effects of cyclodextrins on the solubility and oral bioavailability of tacrolimus in rats. J Pharm Sci 90:690-701.
    • (2001) J Pharm Sci , vol.90 , pp. 690-701
    • Arima, H.1    Yunomae, K.2    Miyake, K.3    Irie, T.4    Hirayama, F.5    Uekama, K.6
  • 31
    • 1942434694 scopus 로고    scopus 로고
    • Self association of cyclodextrin and cyclodextrin complexes
    • Loftsson T, Masson M, Brewster ME. 2004. Self association of cyclodextrin and cyclodextrin complexes. J Pharm Sci 93:1091-1099.
    • (2004) J Pharm Sci , vol.93 , pp. 1091-1099
    • Loftsson, T.1    Masson, M.2    Brewster, M.3
  • 32
    • 59349089796 scopus 로고    scopus 로고
    • The influence of natural organic matter and cations on the rejection of endocrine disrupting and pharmaceutically active compounds by nanofiltration
    • Comerton AM, Andrews RC, Bagley DM. 2009. The influence of natural organic matter and cations on the rejection of endocrine disrupting and pharmaceutically active compounds by nanofiltration. Water Res 43:613-622.
    • (2009) Water Res , vol.43 , pp. 613-622
    • Comerton, A.1    Andrews, R.2    Bagley, D.3
  • 33
    • 3543017331 scopus 로고    scopus 로고
    • Investigating the molecular interactions of oxytetracycline in clay and organic matter: Insights on factors affecting its mobility in soil
    • Kulshrestha P, Giese RF, Aga DS. 2004. Investigating the molecular interactions of oxytetracycline in clay and organic matter: Insights on factors affecting its mobility in soil. Environ Sci Technol 38:4097-4105.
    • (2004) Environ Sci Technol , vol.38 , pp. 4097-4105
    • Kulshrestha, P.1    Giese, R.2    Aga, D.3
  • 34
    • 33947359836 scopus 로고    scopus 로고
    • Sorption of tetracycline and chlortetracycline on K- and Ca-saturated soil clays, humic substances, and clay-humic complexes
    • Pils JRV, Laird DA. 2007. Sorption of tetracycline and chlortetracycline on K- and Ca-saturated soil clays, humic substances, and clay-humic complexes. Environ Sci Technol 41:1928-1933.
    • (2007) Environ Sci Technol , vol.41 , pp. 1928-1933
    • Pils, J.1    Laird, D.2
  • 35
    • 72849146646 scopus 로고    scopus 로고
    • pH-dependent sorption of acidic organic chemicals to soil organic matter
    • Tulp HC, Fenner K, Schwarzenbach RP, Goss K-U. 2009. pH-dependent sorption of acidic organic chemicals to soil organic matter. Environ Sci Technol 43:9189-9195.
    • (2009) Environ Sci Technol , vol.43 , pp. 9189-9195
    • Tulp, H.1    Fenner, K.2    Schwarzenbach, R.3    Goss, K.-U.4
  • 36
    • 0030638567 scopus 로고    scopus 로고
    • Characteristics and significance of the amorphous state in pharmaceutical systems
    • Hancock BC, Zografi G. 1997. Characteristics and significance of the amorphous state in pharmaceutical systems. J Pharm Sci 86:1-12.
    • (1997) J Pharm Sci , vol.86 , pp. 1-12
    • Hancock, B.1    Zografi, G.2
  • 37
    • 79952221329 scopus 로고    scopus 로고
    • Adsorption on silica surfaces
    • In; Papirer, E, Ed., New York: Marcel Dekker Inc.
    • Van Damme H 2000Nanoscale and mesoscale morphology of silica surfaces. In Adsorption on silica surfaces; Papirer, E, Ed., New York: Marcel Dekker Inc., pp 119-165.
    • (2000) Nanoscale and mesoscale morphology of silica surfaces , pp. 119-165
    • Van Damme, H.1
  • 38
    • 31544439894 scopus 로고    scopus 로고
    • Well-ordered mesoporous bioactive glasses (MBG): A promising bioactive drug delivery system
    • Xia W, Chang J, 2006. Well-ordered mesoporous bioactive glasses (MBG): A promising bioactive drug delivery system. J Control Release 110:522-530.
    • (2006) J Control Release , vol.110 , pp. 522-530
    • Xia, W.1    Chang, J.2
  • 39
    • 77957255299 scopus 로고    scopus 로고
    • Enhancement of dissolution rate and oral absorption of a poorly water-soluble drug, K-832, by adsorption onto porous silica using supercritical carbon dioxide
    • Miura H, Kanebako M, Shirai H, Nakao H, Inagi T, Terada K. 2010. Enhancement of dissolution rate and oral absorption of a poorly water-soluble drug, K-832, by adsorption onto porous silica using supercritical carbon dioxide. Eur J Pharm Biopharm 76:215-221.
    • (2010) Eur J Pharm Biopharm , vol.76 , pp. 215-221
    • Miura, H.1    Kanebako, M.2    Shirai, H.3    Nakao, H.4    Inagi, T.5    Terada, K.6
  • 40
    • 47049131872 scopus 로고    scopus 로고
    • Dissolution-rate enhancement of fenofibrate by adsorption onto silica using supercritical carbon dioxide
    • Sanganwar GP, Gupta RB. 2008. Dissolution-rate enhancement of fenofibrate by adsorption onto silica using supercritical carbon dioxide. Int J Pharm 360:213-218.
    • (2008) Int J Pharm , vol.360 , pp. 213-218
    • Sanganwar, G.1    Gupta, R.2
  • 41
    • 0032215146 scopus 로고    scopus 로고
    • Characterization of a inclusion complex of cholesterol and hydroxypropyl-b-cyclodextrin
    • Williams RO, Mahaguna V, Sriwongjanya M. 1998. Characterization of a inclusion complex of cholesterol and hydroxypropyl-b-cyclodextrin. Eur J Pharm Biopharm 46:355-360.
    • (1998) Eur J Pharm Biopharm , vol.46 , pp. 355-360
    • Williams, R.1    Mahaguna, V.2    Sriwongjanya, M.3
  • 45
    • 0031917155 scopus 로고    scopus 로고
    • Effect of pore size on the gaseous adsorption on ethenzamide on porous crystalline cellulose and the physicochemical stability of ethenzamide after storage
    • Matsumoto K, Nakai Y, Yonemochi E, Oguchi T, Yamamoto K. 1998. Effect of pore size on the gaseous adsorption on ethenzamide on porous crystalline cellulose and the physicochemical stability of ethenzamide after storage. Chem Pharm Bull 46:314-318.
    • (1998) Chem Pharm Bull , vol.46 , pp. 314-318
    • Matsumoto, K.1    Nakai, Y.2    Yonemochi, E.3    Oguchi, T.4    Yamamoto, K.5
  • 47
    • 0037677557 scopus 로고    scopus 로고
    • Adsorption and entrapment of salicylamide molecules into the mesoporous structure of folded sheets mesoporous material (FSM-16)
    • Tozuka Y, Oguchi T, Yamamoto K. 2003. Adsorption and entrapment of salicylamide molecules into the mesoporous structure of folded sheets mesoporous material (FSM-16). Pharm Res 20:926-930.
    • (2003) Pharm Res , vol.20 , pp. 926-930
    • Tozuka, Y.1    Oguchi, T.2    Yamamoto, K.3
  • 49
    • 27744566574 scopus 로고    scopus 로고
    • Mesoporous silicon microparticles for oral drug delivery: Loading and release of five model drugs
    • Salonen J, Laitinen L, Kaukonen AM. 2005. Mesoporous silicon microparticles for oral drug delivery: Loading and release of five model drugs. J Control Release 108:362-374.
    • (2005) J Control Release , vol.108 , pp. 362-374
    • Salonen, J.1    Laitinen, L.2    Kaukonen, A.3
  • 50
    • 0035095847 scopus 로고    scopus 로고
    • Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with amorphous polymers
    • Froster A, Hempenstall J, Rades T. 2001. Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with amorphous polymers. J Pharm Pharmacol 53:303-315.
    • (2001) J Pharm Pharmacol , vol.53 , pp. 303-315
    • Froster, A.1    Hempenstall, J.2    Rades, T.3
  • 51
    • 5144219871 scopus 로고    scopus 로고
    • Amorphous drug delivery systems: Molecular aspects, design, and performance
    • Kaushal AM, Gupta P, Bansal AK. 2004. Amorphous drug delivery systems: Molecular aspects, design, and performance. Crit Rev Ther Drug Carrier Syst 21:133-193.
    • (2004) Crit Rev Ther Drug Carrier Syst , vol.21 , pp. 133-193
    • Kaushal, A.1    Gupta, P.2    Bansal, A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.