Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure-activity relationships

European Journal of Medicinal Chemistry

Volumn 46, Issue 3, 2011, Pages 819-824

  Pan, Bin ^a   Huang, Renzheng ^b   Zheng, Likang ^a   Chen, Chen ^a   Han, Shiqing ^a   Qu, Di ^b   Zhu, Mingli ^a   Wei, Ping ^a  

^a NANJING TECH UNIVERSITY   (China)

^b FUDAN UNIVERSITY   (China)

Author keywords

Antibiofilm activity; Inhibitors; Staphylococcus epidermidis; Thiazolidione

Indexed keywords

3 [5 [(6 (ETHOXYCARBONYL) 5 (BENZO[1,3]DIOXOL 5 YL) 3 OXO 7 PHENYL THIAZOLO[3,2 A]PYRIMIDIN 2(5H)YLIDENE)METHYL]FURAN 2 YL]BENZOIC ACID; 4 [5 [(4 OXO 3 (2 METHYLPHENYL) 2 (2 METHYLPHENYLIMINO)THIAZOLIDIN 5 YLIDENE)METHYL]FURAN 2 YL]BENZOIC ACID; ANTIINFECTIVE AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL GROWTH; BIOFILM; BIOLOGICAL ACTIVITY; DRUG DESIGN; DRUG SYNTHESIS; HUMAN; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; STAPHYLOCOCCUS EPIDERMIDIS; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; BIOFILMS; HUMANS; MICROBIAL SENSITIVITY TESTS; STAPHYLOCOCCAL INFECTIONS; STAPHYLOCOCCUS EPIDERMIDIS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLIDINES;

EID: 79951671509     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2010.12.014     Document Type: Article

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