HIV protease-mediated activation of sterically capped proteasome inhibitors and substrates

Journal of the American Chemical Society

Volumn 133, Issue 4, 2011, Pages 698-700

  Buckley, Dennis L ^a   Corson, Timothy W ^a,c   Aberle, Nicholas ^a   Crews, Craig M ^a,b  

^a YALE UNIVERSITY   (United States)

^b YALE UNIVERSITY SCHOOL OF MEDICINE   (United States)

^c INDIANA UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIRETROVIRAL DRUGS; CHEMICAL BIOLOGY; CYTOTOXIC; HIV-1 PROTEASE; HIV-PROTEASE; INFECTED CELLS; POLYLYSINE DENDRIMERS; PROOF OF CONCEPT; PROTEASOME INHIBITORS; PROTEASOMES; SMALL MOLECULES; TROJAN HORSE;

DENDRIMERS;

HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE; PROTEASOME INHIBITOR;

ARTICLE; ENZYME INHIBITION; ENZYME INHIBITOR COMPLEX; ENZYME INHIBITOR INTERACTION; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; NONHUMAN;

ANIMALS; CATTLE; HIV PROTEASE; HIV-1; PROTEASE INHIBITORS; PROTEASOME ENDOPEPTIDASE COMPLEX;

EID: 79851474437     PISSN: 00027863     EISSN: 15205126     Source Type: Journal    
DOI: 10.1021/ja109377p     Document Type: Article

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