메뉴 건너뛰기




Volumn 68, Issue 11, 2010, Pages 1195-1206

Pd0-mediated rapid C-[11C]methylations and C-[ 18F]fluoromethylations: Revolutionary new methodologies for the synthesis of short-lived PET molecular probes

Author keywords

[No Author keywords available]

Indexed keywords

CARBON FRAMEWORK; CROSS COUPLING REACTIONS; IN-VIVO; MOLECULAR PROBES; MOLECULAR SCIENCE; ORGANOBORON COMPOUND; RAPID REACTIONS;

EID: 79551513244     PISSN: 00379980     EISSN: None     Source Type: Journal    
DOI: 10.5059/yukigoseikyokaishi.68.1195     Document Type: Article
Times cited : (10)

References (81)
  • 5
    • 79551568075 scopus 로고    scopus 로고
    • The European Medicines Agency, Evaluation of Medicines for Human Use, Position paper on non-clinical safety studies to support clinical trials with a single microdose, CPMP/SWP/2599/02/Rev1, June 23, 2004
    • The European Medicines Agency, Evaluation of Medicines for Human Use, Position paper on non-clinical safety studies to support clinical trials with a single microdose, CPMP/SWP/2599/02/Rev1, June 23, 2004;
  • 6
    • 79551560984 scopus 로고    scopus 로고
    • U. S. Department of Health and Human Services, Food and Drug Administration, Center for Drug Evaluation and Research, Guidance for Industry, Investigators, and Reviewers, Exploratory IND Studies, January 2006
    • U. S. Department of Health and Human Services, Food and Drug Administration, Center for Drug Evaluation and Research, Guidance for Industry, Investigators, and Reviewers, Exploratory IND Studies, January 2006;
  • 7
    • 79551505489 scopus 로고    scopus 로고
    • Japan's response to microdosing study, Notification No. 0603001, June 3
    • e) Japan's response to microdosing study, Notification No. 0603001, June 3,2008, Guidance for the Conduct of Microdosing Clinical Trials, Evaluation and Licensing Division, Pharmaceutical and Food Safety Bureau, Ministry of Health, Labour and Welfare, Japan.
    • (2008)
  • 31
    • 84985570392 scopus 로고
    • For reviews of the Stille reaction, see
    • (a) Stille, J. K., Angew. Chem., Int. Ed Engl. 1986, 25, 508. For reviews of the Stille reaction, see:
    • (1986) Angew. Chem., Int. Ed Engl. , vol.25 , pp. 508
    • Stille, J.K.1
  • 41
    • 0000808892 scopus 로고
    • also see references cited therein
    • (b) Falck, J. R.; Bhatt, R. K.; Ye, J., J. Am. Chem. Soc. 1995, 117, 5973, also see references cited therein.
    • (1995) J. Am. Chem. Soc. , vol.117 , pp. 5973
    • Falck, J.R.1    Bhatt, R.K.2    Ye, J.3
  • 45
    • 79551559185 scopus 로고    scopus 로고
    • 2 in a cyclotron
    • 2 in a cyclotron.
  • 50
    • 79551549730 scopus 로고    scopus 로고
    • 11C-8 was 37-100 GBq/|μmol. The total synthesis time was 35-40 min
    • 11C]-8 was 37-100 GBq/|μmol. The total synthesis time was 35-40 min.
  • 51
    • 79551530319 scopus 로고    scopus 로고
    • 11C-labeled compound by mechanical synthesis under PET radiolabeling conditions
    • 11C-labeled compound by mechanical synthesis under PET radiolabeling conditions.
  • 67
    • 79551523366 scopus 로고    scopus 로고
    • 11C]-14 will be reported in due course
    • 11C]-14 will be reported in due course.
  • 70
    • 2042507954 scopus 로고
    • For reviews of the Suzuki-Miyaura reaction, see: a) Miyaura, N.; Suzuki, A., Chem. Rev. 1995, 95, 2457.
    • (1995) Chem. Rev. , vol.95 , pp. 2457
    • Miyaura, N.1    Suzuki, A.2
  • 72
    • 17144421373 scopus 로고    scopus 로고
    • Astruc, D., Ed.; Wiley- VCH
    • Suzuki, A. In Modern Arene Chemistry, Astruc, D., Ed.; Wiley-VCH, 2002, 53-106.
    • (2002) Modern Arene Chemistry , pp. 53-106
    • Suzuki, A.1
  • 74
    • 11844294723 scopus 로고    scopus 로고
    • Ser. B 80, For the cross-coupling reactions between alkyl iodide and boron compounds by the Suzuki-Miyaura reaction
    • e) Suzuki, A., Proc. Jpn. Acad. 2004, Ser. B 80, 359. For the cross-coupling reactions between alkyl iodide and boron compounds by the Suzuki-Miyaura reaction,
    • (2004) Proc. Jpn. Acad. , pp. 359
    • Suzuki, A.1
  • 81
    • 79551507962 scopus 로고    scopus 로고
    • 11C] methylation of Flurbiprofen methyl ester
    • 11C] methylation of Flurbiprofen methyl ester.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.