Synthesis and antimicrobial activity of novel 2-(aryl)-3-[5-(2-oxo-2H-3- chromenyl)-1,3-oxazol-2-yl]-1,3-thiazolan-4-ones

Journal of Heterocyclic Chemistry

Volumn 48, Issue 1, 2011, Pages 176-182

  Reddy, Ch Sanjeeva ^a   Devi, M Vani ^a   Kumar, G Rajesh ^a   Rao, L Sanjeeva ^a   Nagaraj, A ^b  

^a KAKATIYA UNIVERSITY   (India)

^b TELANGANA UNIVERSITY   (India)

Author keywords

[No Author keywords available]

Indexed keywords

2 (1,3 BENZODIOXOL 5 YL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (2 FURYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (2,6 DIFLUOROPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (3 NITROPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (4 CHLOROPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (4 HYDROXY 3 METHOXYPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (4 HYDROXYPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (4 METHYLPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 (4 NITROPHENYL) 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; 2 [4 (DIMETHYLAMINO)PHENYL] 3 [5 (2 OXO 2H 3 CHROMENYL) 1,3 OXAZOL 2 YL] 1,3 THIAZOLAN 4 ONE; AMPHOTERICIN B; ANTIINFECTIVE AGENT; OXAZOLE DERIVATIVE; STREPTOMYCIN; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS; BACILLUS SUBTILIS; CANDIDA ALBICANS; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; ESCHERICHIA COLI; MICROCOCCUS LUTEUS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PROTEUS VULGARIS; SALMONELLA TYPHIMURIUM; STANDARD; STAPHYLOCOCCUS AUREUS; TRICHOPHYTON MENTAGROPHYTES; TRICHOPHYTON RUBRUM;

EID: 79251590274     PISSN: 0022152X     EISSN: 19435193     Source Type: Journal    
DOI: 10.1002/jhet.505     Document Type: Article

References (38)

1. Billeret, D.,;, Blondeau, D.,;, Sliwa, H., J Heterocycl Chem 1993, 30, 671.
2. Vallet, F. M., J Ger Offen 1978, 2, 751.
3. Suzmann, M. M., In Abstr. IV World Congress of Cardiology, Mexico City, 1962, p 344.
4. Doucet, C.,;, Pochet, L.,;, Thierry, N.,;, Pirotte, B.,;, Delarge, J.,;, Reboud-Ravaux, M., J Med Chem 1999, 42, 4161.
5. Pochet, L.,;, Doucet, C.,;, Schynts, M.,;, Therry, N.,;, Boggetto, N.,;, Pirotte, B.,;, Jiang, K. Y.,;, Masereel. B.,;, de Tullio, P.,;, Delarge, J.,;, Reboud-Ravaux, M., J Med Chem 1996, 39, 2579.
6. Spiro, V.,;, Madonia, P., Atti Acad Sci Lett Antipalermo 1959, A95920187.
7. (a), Mitra, A. K.,;, De, A.,;, Karchaudhuri, N.,;, Misra, S. K.,;, Mukhopadhyay, A. K., J Indian Chem Soc 1998, 75, 666
8. (b), Cravotto, G.,;, Nano, G. M.,;, Palmisano, G.,;, Tagliapietra, S., Tetrahedron: Asymmetry 2001, 12, 707.
9. Wang, C. J.,;, Hsieh, Y. J.,;, Chu, C. Y.,;, Lin, Y. L.,;, Tseng, T. H., Cancer Lett 2002, 183, 163.
10. Kirkiacharian, S.,;, Thuy, D. T.,;, Sicsis, S.,;, Bakhchinian, R.,;, Kurkjian, R.,;, Tonnaire, T., Il Farmaco 2002, 57, 703.
11. Kayser, O.,;, Kolodziej, H., Planta Med 1997, 63, 508.
12. Olayinka, O. A.,;, Obinna, C. N., J Heterocycl Chem 2010, 47, 179.
13. Vigorita, M. G.,;, Ottana, R.,;, Monforte, F.,;, Maccari, R.,;, Trovato, A.,;, Monforte, M. T.,;, Taviano, M. F., Bioorg Med Chem Lett 2001, 11, 2791.
14. Chande, M. S.,;, Suryanarayan, V., J Chem Res 2005, 345.
15. Kavitha, C. V.,;, Basappa, S.,;, Swamy, N.,;, Mantelingu, K.,;, Doreswamy, S.,;, Sridhar, M. A.,;, Prasad, S.,;, Rangappa, K. S., Bioorg Med Chem 2006, 14, 2290.
16. Ergene, N.,;, Capan, G., Il Farmaco 1994, 49, 449.
17. Diurno, M. V.,;, Mazzoni, O.,;, Izzo, A. A.,;, Bolognese, A., Il Farmaco 1997, 52, 237.
18. Tanabe, Y.,;, Komuro, Y.,;, Imanishi, N.,;, Morooka, S.,;, Enomoto, M.,;, Kojima, A.,;, Sanemitsu, Y.,;, Mizutani, M., Tetrahedron Lett 1991, 32, 379.
19. Koike, H.,;, Imanashi, N.,;, Natsume, Y.,;, Morooka, S., Eur J Pharmacol 1994, 269, 299.
20. Tanabe, Y.,;, Yamamoto, H.,;, Murakami, M.,;, Yanagi, K.,;, Kubota, Y.,;, Okumura, H.,;, Sanemitsu, Y.,;, Suzukamo, G., J Chem Soc Perkin Trans I 1995, 7, 935.
21. Diurno, M. V.,;, Mazzoni, O.,;, Correale, G.,;, Monterry, I. G., Il Farmaco 1999, 54, 579.
22. Previtera, T.,;, Vigorita, M. G.,;, Bisila, M.,;, Orshini, F.,;, Benetolla, F.,;, Bombieri, G., Eur J Med Chem 1994, 29, 317.
23. Sharma, R. C.,;, Kumar, D., J Indian Chem Soc 2000, 77, 492.
24. Piscapo, E.,;, Diurno, M. V.,;, Gagliardi, R.,;, Mazzoni, O., Boll Soc Ital Biol Sper 1989, 65, 853.
25. Ueno, H.,;, Oe, T.,;, Snehiro, I.,;, Nakamura, S., US Pat. 5,594,116 (1997); Chem Abstr 1977, 126, 157507.
26. Ottana, R.,;, Mazzon, E.,;, Dugo, L.,;, Monforte, F.,;, Maccari, R.,;, Sautebin, L.,;, De Luca, G.,;, Vigorita, M. G.,;, Alcaro, S.,;, Ortuso, F., Eur J Pharmacol 2002, 448, 71.
27. Kato, T.,;, Ozaki, T.,;, Tamura, K., J Med Chem 1999, 42, 3134.
28. Tanabe, Y.,;, Suzukamo, G.,;, Komuro, Y.,;, Imanishi, N.,;, Morooka, S.,;, Enomoto, M.,;, Kojima, A.,;, Sanemitsu, Y.,;, Mizutani, M., Tetrahedron Lett 1991, 32, 379.
29. Kato, T.,;, Ozaki, T.,;, Ohi, N., Tetrahedron: Asymmetry 1999, 10, 3963.
30. Adachi, Y.,;, Suzuki, Y.,;, Homma, N.,;, Fukazawa, M.,;, Tamura, K.,;, Nishie, I.,;, Kuromaru, O., Eur J Pharmacol 1999, 367, 267.
31. Ebeid, M. Y.,;, Fathallah, O. A.,;, El-Zaber, M. I.,;, Kamel, M. M.,;, Abdon, W. A.,;, Anwar, M. M., Bull Fac Pharmacol 1996, 34, 125.
32. Voss, M. E.,;, Carter, P. H.,;, Tebben, A. J.,;, Scherle, P. A.,;, Brown, G. D.,;, Thompson, L. A.,;, Xu, M.,;, Lo, Y. C.,;, Yang Liu, R. R.-Q., Bioorg Med Chem Lett 2006, 16, 1907.
33. Manrao, M. R.,;, Monika, J.,;, Kaul, V. K., Pl Dis Res 1997, 12, 70.
34. Sanjeeva Reddy, Ch.,;, Nagaraj, A.,;, Srinivas, A., Chem Pharm Bull 2009, 57, 685.
35. Sanjeeva Reddy, Ch.,;, Raghu, M.,;, Nagaraj, A., J Heterocycl Chem 2009, 46, 261.
36. Sanjeeva Reddy, Ch.,;, Raghu, M.,;, Nagaraj, A., J Heterocycl Chem 2008, 45, 1121.
37. Sahu, S. K.,;, Mishra, A.,;, Behera, R. K., Indian J Heterocycl Chem 1996, 6, 91.
38. National Committee for Clinical Laboratory Standards (NCCLS). Standard methods for dilution antimicrobial susceptibility tests for bacteria, which grows aerobically. Nat Comm Lab Stands Villanova, 1982, p 242.