Helix 11 dynamics is critical for constitutive androstane receptor activity

Structure

Volumn 19, Issue 1, 2011, Pages 37-44

  Wright, Edward ^a   Busby, Scott A ^b   Wisecarver, Sarah ^a   Vincent, Jeremy ^a   Griffin, Patrick R ^b   Fernandez, Elias J ^a  

^a UNIVERSITY OF TENNESSEE   (United States)

^b SCRIPPS RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1,4 BIS(3,5 DICHLORO 2 PYRIDYLOXY)BENZENE; CONSTITUTIVE ANDROSTANE RECEPTOR; DEUTERIUM; HYDROGEN; MECLOZINE; RETINOID X RECEPTOR;

ARTICLE; BINDING SITE; COMPLEX FORMATION; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN STRUCTURE;

ALLOSTERIC SITE; ANIMALS; BINDING SITES; HUMANS; MECLIZINE; MICE; MODELS, MOLECULAR; NUCLEAR RECEPTOR COACTIVATOR 1; PROTEIN BINDING; PROTEIN MULTIMERIZATION; PROTEIN STABILITY; PROTEIN STRUCTURE, SECONDARY; PROTEIN STRUCTURE, TERTIARY; PYRIDINES; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECOMBINANT FUSION PROTEINS; RETINOID X RECEPTORS; THERMODYNAMICS; TRANSCRIPTIONAL ACTIVATION;

EID: 78651256360     PISSN: 09692126     EISSN: 18784186     Source Type: Journal    
DOI: 10.1016/j.str.2010.11.008     Document Type: Article

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