Simple and rapid determination of the enzyme kinetics of HIV-1 reverse transcriptase and anti-HIV-1 agents by a fluorescence based method

Journal of Virological Methods

Volumn 171, Issue 2, 2011, Pages 381-387

  Silprasit, Kun ^a   Thammaporn, Ratsupa ^a   Tecchasakul, Supanna ^a   Hannongbua, Supa ^a   Choowongkomon, Kiattawee ^a  

^a KASETSART UNIVERSITY   (Thailand)

Author keywords

Anti HIV agents; Fluorometric method; High throughput screening; HIV 1 reverse transcriptase; PicoGreen

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; DIPYRIDODIAZEPINONE DERIVATIVE; FLUORESCENT DYE; NEVIRAPINE; NONNUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITOR; PICOGREEN DYE; PLANT EXTRACT; RNA DIRECTED DNA POLYMERASE; UNCLASSIFIED DRUG;

ANALYTIC METHOD; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG POTENCY; DRUG SCREENING; ENZYME INHIBITION; ENZYME KINETICS; ENZYME SUBSTRATE COMPLEX; FLUOROMETRY; HIGH THROUGHPUT SCREENING; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50; MEDICINAL PLANT; NONHUMAN; PRIORITY JOURNAL; QUANTITATIVE ASSAY; SOLVENT EXTRACTION; SOXHLET EXTRACTION;

ANTI-HIV AGENTS; DRUG EVALUATION, PRECLINICAL; FLUORESCENCE; HIV REVERSE TRANSCRIPTASE; HUMANS; ORGANIC CHEMICALS;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 78651231649     PISSN: 01660934     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jviromet.2010.12.001     Document Type: Article

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