Structural characteristics of thiosemicarbazones as inhibitors of melanogenesis

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 22, 2010, Pages 6794-6796

  Lee, Ki Cheul ^a   Thanigaimalai, Pillaiyar ^a   Sharma, Vinay K ^a   Kim, Min Seok ^a   Roh, Eunmiri ^b   Hwang, Bang Yeon ^b   Kim, Youngsoo ^b   Jung, Sang Hun ^a  

^a Chungnam National University   (South Korea)

^b Chungbuk National University   (South Korea)

Author keywords

Hydrophobicity; Melanogenesis inhibitor; Thiosemicarbazones

Indexed keywords

HORMONE RECEPTOR BLOCKING AGENT; THIOSEMICARBAZONE DERIVATIVE;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; HORMONE INHIBITION; HYDROPHOBICITY; IC 50; MELANOGENESIS; STRUCTURE ACTIVITY RELATION;

ANIMALS; MELANINS; MELANOMA, EXPERIMENTAL; MICE; STRUCTURE-ACTIVITY RELATIONSHIP; THIOSEMICARBAZONES;

EID: 77958064836     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.08.114     Document Type: Article

References (31)

1. A. Sánchez-Ferrer, J.N. Rodríguez-López, F. García-Cánovas, and F. García-Carmona Biochim. Biophys. Acta 1247 1995 1
2. M.R. Chase, K. Raina, J. Bruno, and M. Sugumaran Insect Biochem. Mol. 30 2000 953
3. V.J. Hearing, and M. Jimenez Int. J. Biochem. 19 1987 1141
4. R. Halaban, R.S. Patton, E. Cheng, S. Svedine, E.S. Trombetta, M.L. Wahl, S. Ariyan, and D.N. Hebert J. Biol. Chem. 277 2002 14821
5. Y. Xu, A.H. Stokes, R.J. Roskosi, and K.E. Vrana J. Neurosci. Res. 54 1998 691
6. M. Asanuma, I. Miyazaki, and N. Ogawa Neurotoxicol. Res. 5 2003 165
7. W.S. Oetting Pigment Cell Res. 13 2000 320
8. M. Ashida, and P. Brey Proc. Natl. Acad. Sci. U.S.A. 92 1995 10698
9. T.B. Fitzpatrick, A.Z. Eisen, K. Wolff, I.M. Freedberg, and K.F. Austen Dermatology in General Medicine 1983 McGraw-Hill, Inc. New York, NY
10. K. Maeda, and M. Fukuda J. Soc. Cosmet. Chem. 42 1991 361
11. S. Kojima, H. Yamaguchi, K. Morita, and Y. Ueno Biol. Pharm. Bull. 18 1995 1076
12. V.M. Verallo-Rowell, V. Verallo, K. Graupe, L. Lopez-Villafuerte, and M. Garcia-Lopez Acta Derm. Venereol. 143 1989 58
13. H. Takiwake, S. Shirai, H. Kohono, H. Soh, and S. Arase J. Invest. Dermatol. 103 1994 642
14. C.K. Kimbrough-Green Arch. Dermatol. 130 1994 727
15. K.P. DuBois, and W.F. Erway J. Biol. Chem. 165 1946 711
16. M. Criton, and V. Le Mallay-Harmon Bioorg. Med. Chem. Lett. 18 2008 3607
17. C. Gerdemann, C. Eicken, and B. Krebs Acc. Chem. Res. 35 2002 183
18. T. Klabunde, C. Eicken, J.C. Sacchettini, and B. Krebs Nat. Struct. Biol. 5 1998 1084
19. P.C. Lv, C.F. Zhou, J. Chen, P.G. Liu, K.R. Wang, W.J. Mao, H.Q. Li, Y. Yang, J. Xiong, and H.L. Zhu Bioorg. Med. Chem. 18 2010 314
20. P. Thanigaimalai, T.A. Le Hoang, K.C. Lee, S.C. Bang, V.K. Sharma, C.Y. Yun, E. Roh, B.Y. Hwang, Y. Kim, and S.H. Jung Bioorg. Med. Chem. Lett. 20 2010 2991
21. J. Varsha, M. Pradeep, K. Sushil, and J.P. Stables Eur. J. Med. Chem. 43 2008 135
22. X.Y. Xie, L. Jiang, C.B. Xue, and W.C. Luo Huaxue Shiji 29 2007 34
23. V. Jatav, S. Kashaw, and P. Mishra Med. Chem. Res. 17 2008 169
24. H. Wuyts, L. Berman, and A. Lacourt Bull. Soc. Chimiques Belg. 40 1931 665
25. S.S. Karki, S. Thota, S.Y. Darj, J. Balzarini, and E. De Clercq Bioorg. Med. Chem. 15 2007 6632
26. M.S. Bakkar, M. Yamin, and M.S. Monshi Synth. React. Inorg. Met.-Org. Chem. 33 2003 1157
27. W. Yi, R.H. Cao, Z.Y. Chen, L. Yu, L. Ma, and H.C. Song Chem. Pharm. Bull. 57 2009 1273
28. G. Brahmeshwari, V.R. Rao, T.S. Kumari, and T.V.P. Rao Phosphorus, Sulfur Silicon Relat. Elem. 92 1994 51
29. M. Li, L. Yao, Z. Wang, and J. Wang Huaxue Yanjiu 17 2006 44
30. P. Thanigaimalai, K.C. Lee, S.C. Bang, J.H. Lee, C.Y. Yun, E. Roh, B.Y. Hwang, Y. Kim, and S.H. Jung Bioorg. Med. Chem. 18 2010 1135
31. C.B. Xue, L. Zhang, W.C. Luo, X.Y. Xie, L. Jiang, and T. Xiao Bioorg. Med. Chem. 15 2007 2006