Synthesis, antibacterial and antifungal activity of some novel 3-[5-(4-substituted phenyl) 1,3,4-thiadiazole-2-yl]-2-styryl quinazoline-4(3H)-ones

Medicinal Chemistry Research

Volumn 17, Issue 2-7, 2008, Pages 169-181

  Jatav, Varsha ^a   Kashaw, Sushil ^a   Mishra, Pradeep ^a  

^a DR H S GOUR UNIVERSITY   (India)

Author keywords

[No Author keywords available]

Indexed keywords

2 METHYL 3 (1,3,4 THIADIAZOLE 2' YL) 4(3H)QUINAZOLINONE; 2 STYRYL QUINAZOLINE 4(3H)ONE; 3 (1,3,4 THIADIAZOLYL) 2 STYRYLQUINAZOLIN 4(3H)ONE; 4(3H) QUINAZOLINONE DERIVATIVE; NORFLOXACIN; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ASPERGILLUS NIGER; BACILLUS SUBTILIS; BACTERIAL STRAIN; CANDIDA ALBICANS; CONFERENCE PAPER; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; FUSARIUM OXYSPORUM; MINIMUM INHIBITORY CONCENTRATION; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS;

EID: 52949131576     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00044-007-9047-2     Document Type: Conference Paper

References (15)

1. WL Armarego 1963 Quinazolines. Adv Heterocycl Chem 11 253 309
2. MT Bogert HA Seil 1905 The synthesis of 2-methyl-5-nitro-4- ketodihydroquinazolines from 6-nitroacetanthranil and primary amines. J Am Chem Soc 27 1305 1310
3. SL Cao YP Feng YY Jiang SY Liu GY RT Ding Li 2005 Synthesis and in vitro antitumor activity of 4(3H)-quinazolinone derivatives with dithiocarbamate side chains. Bioorg Med Chem Lett 15 1915 1917
4. th ed. Chandighar, India (Medium No-137), p138
5. Dhananjaya U, Reddy GBS (1998) Chem Pharm Bull 46:1254
6. L Fisnerova J Grimova Z Roubal E Maturova B Brunova 1986 Esters of 3-(2-hydroxyethyl)-4(3H)-quinazolinone with an analgesic effect. Cesk Farm 3 447 450
7. Ghai CL (1999) A Textbook of Practical Physiology, Jaypee brothers, Medical, 5th ed. New Delhi, India. p 34
8. D Gravier G Hou F Casadebaig JP Dupin H Bernard M Boisseau 1992 Thieno[2,3-d]pyrimidin-4(3H)-one derivatives and 1,2-dihydrogenated homologues: synthesis, enhanced in vitro antiaggregant activity for reduced compounds. Pharmazie 47 754 757
9. th ed. London
10. SK Jain P Mishra 2000 Synthesis of some 2-Amino-5-Aryl-1,3,4- Thiadiazoles. Asian Journal of Chemistry 12 1341 1343
11. V Murugan CC Thomas GVS Rama Sharma EP Kumar B Suresh 2003 Synthesis of 2-substituted quinayolin-4(3H)-ones as a new class of anticancer agents. J Ind Pharm Sci 65 386 389
12. D Raffa G Daidone B Maggio S Cascioferro F Plescia D Schillaci 2004 Synthesis and antileukemic activity of new 3-(5-methylisoxazol-3-yl) and 3-(pyrimidin-2-yl)-2-styrylquinazolin-4(3H)-ones. Farmaco 59 451 455
13. AR Saundane K Rudresh ND Satyanarayan SP Hiremath 1998 Pharmacological screening of 6H, 11H-indolo {3, 2-c} isoquinolin-5-ones and their derivatives. J Ind Pharm Sci 60 379 383
14. thed. New Delhi, India. Vol-II, A-112
15. rd ed., p 243