메뉴 건너뛰기




Volumn 399, Issue 1-2, 2010, Pages 109-115

A thermal analysis method to predict the complete phase diagram of drug-polymer solid dispersions

Author keywords

Felodipine PAA system; Phase diagram; Phase separation; Solid dispersion; The Flory Huggins theory

Indexed keywords

FELODIPINE; POLYACRYLIC ACID;

EID: 77956885126     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2010.08.013     Document Type: Article
Times cited : (104)

References (30)
  • 1
    • 0023305850 scopus 로고
    • Amorphous thermoreversible gels of atactic polystyrene
    • Arnauts J., Berghmans H. Amorphous thermoreversible gels of atactic polystyrene. Polym. Commun. 1987, 28:66-68.
    • (1987) Polym. Commun. , vol.28 , pp. 66-68
    • Arnauts, J.1    Berghmans, H.2
  • 3
    • 0015124656 scopus 로고
    • Pharmaceutical applications of solid dispersion systems
    • Chiou W.L., Riegelman S. Pharmaceutical applications of solid dispersion systems. J. Pharm. Sci. 1971, 60:1281-1302.
    • (1971) J. Pharm. Sci. , vol.60 , pp. 1281-1302
    • Chiou, W.L.1    Riegelman, S.2
  • 6
    • 70349649718 scopus 로고    scopus 로고
    • Differences in the interaction between aryl propionic acid derivatives and poly(vinylpyrrolidone) K30: a multi-methodological approach
    • Gashi Z., Censi R., Malaj L., Gobetto R., Mozzicafreddo M., Angeletti M., Masic A., Martino P.D. Differences in the interaction between aryl propionic acid derivatives and poly(vinylpyrrolidone) K30: a multi-methodological approach. J. Pharm. Sci. 2009, 98:4216-4228.
    • (2009) J. Pharm. Sci. , vol.98 , pp. 4216-4228
    • Gashi, Z.1    Censi, R.2    Malaj, L.3    Gobetto, R.4    Mozzicafreddo, M.5    Angeletti, M.6    Masic, A.7    Martino, P.D.8
  • 7
    • 0024104931 scopus 로고
    • Temperature, composition and molecular-weight dependence of the binary interaction parameter of polystyrene/poly(vinyl methyl ether) blends
    • Han C.C., Bauer B.J., Clark J.C., Muroga Y., Matsushita Y., Okada M., Tran-cong Q., Chang T., Sanchez I.C. Temperature, composition and molecular-weight dependence of the binary interaction parameter of polystyrene/poly(vinyl methyl ether) blends. Polymer 1988, 29:2002-2014.
    • (1988) Polymer , vol.29 , pp. 2002-2014
    • Han, C.C.1    Bauer, B.J.2    Clark, J.C.3    Muroga, Y.4    Matsushita, Y.5    Okada, M.6    Tran-cong, Q.7    Chang, T.8    Sanchez, I.C.9
  • 8
    • 75749094421 scopus 로고    scopus 로고
    • Review: physical chemistry of solid dispersions
    • Janssens S., Van den Mooter G. Review: physical chemistry of solid dispersions. J. Pharm. Pharmacol. 2009, 61:1571-1586.
    • (2009) J. Pharm. Pharmacol. , vol.61 , pp. 1571-1586
    • Janssens, S.1    Van den Mooter, G.2
  • 9
    • 24644474682 scopus 로고    scopus 로고
    • Miscibility behavior and formation mechanism of stabilized felodipine-polyvinylpyrrolidone amorphous solid dispersions
    • Karavas E., Ktistis G., Xenakis A., Georgarakis E. Miscibility behavior and formation mechanism of stabilized felodipine-polyvinylpyrrolidone amorphous solid dispersions. Drug Dev. Ind. Pharm. 2005, 31:473-489.
    • (2005) Drug Dev. Ind. Pharm. , vol.31 , pp. 473-489
    • Karavas, E.1    Ktistis, G.2    Xenakis, A.3    Georgarakis, E.4
  • 11
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • Leuner C., Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur. J. Pharm. Biopharm. 2000, 50:47-60.
    • (2000) Eur. J. Pharm. Biopharm. , vol.50 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 12
    • 33749442356 scopus 로고    scopus 로고
    • Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility
    • Marsac P.J., Shamblin S.L., Taylor L.S. Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility. Pharm. Res. 2006, 23:2417-2426.
    • (2006) Pharm. Res. , vol.23 , pp. 2417-2426
    • Marsac, P.J.1    Shamblin, S.L.2    Taylor, L.S.3
  • 13
    • 57749206650 scopus 로고    scopus 로고
    • Estimation of drug-polymer miscibility and solubility in amorphous solid dispersions using experimentally determined interaction parameters
    • Marsac P.J., Li T.L., Taylor L.S. Estimation of drug-polymer miscibility and solubility in amorphous solid dispersions using experimentally determined interaction parameters. Pharm. Res. 2009, 26:139-151.
    • (2009) Pharm. Res. , vol.26 , pp. 139-151
    • Marsac, P.J.1    Li, T.L.2    Taylor, L.S.3
  • 14
    • 73949151261 scopus 로고    scopus 로고
    • Effect of temperature and moisture on the miscibility of amorphous dispersions of felodipine and poly(vinyl pyrrolidone)
    • Marsac P.J., Rumondor A.C.F., Nivens D.E., Kestur U.S., Stanciu L., Taylor L.S. Effect of temperature and moisture on the miscibility of amorphous dispersions of felodipine and poly(vinyl pyrrolidone). J. Pharm. Sci. 2010, 99:169-185.
    • (2010) J. Pharm. Sci. , vol.99 , pp. 169-185
    • Marsac, P.J.1    Rumondor, A.C.F.2    Nivens, D.E.3    Kestur, U.S.4    Stanciu, L.5    Taylor, L.S.6
  • 15
    • 0037130753 scopus 로고    scopus 로고
    • Solubility measurement using differential scanning calorimetry
    • Mohan R., Lorenz H., Myerson A.S. Solubility measurement using differential scanning calorimetry. Ind. Eng. Chem. Res. 2002, 41:4854-4862.
    • (2002) Ind. Eng. Chem. Res. , vol.41 , pp. 4854-4862
    • Mohan, R.1    Lorenz, H.2    Myerson, A.S.3
  • 16
    • 77953296607 scopus 로고    scopus 로고
    • Drug-polymer solubility and miscibility: stability consideration and practical challenge in amorphous solid dispersion development
    • Qian F., Huang J., Hussain M.A. Drug-polymer solubility and miscibility: stability consideration and practical challenge in amorphous solid dispersion development. J. Pharm. Sci. 2010, 99:2941-2947.
    • (2010) J. Pharm. Sci. , vol.99 , pp. 2941-2947
    • Qian, F.1    Huang, J.2    Hussain, M.A.3
  • 18
    • 70350057599 scopus 로고    scopus 로고
    • Phase behavior of poly(vinylpyrrolidone) containing amorphous solid dispersions in the presence of moisture
    • Rumondor A.C.F., Marsac P.J., Stanford L.A., Taylor L.S. Phase behavior of poly(vinylpyrrolidone) containing amorphous solid dispersions in the presence of moisture. Mol. Pharm. 2009, 6:1492-1505.
    • (2009) Mol. Pharm. , vol.6 , pp. 1492-1505
    • Rumondor, A.C.F.1    Marsac, P.J.2    Stanford, L.A.3    Taylor, L.S.4
  • 19
    • 70350220585 scopus 로고    scopus 로고
    • Evaluation of drug-polymer miscibility in amorphous solid dispersion systems
    • Rumondor A.C.F., Ivanisevic I., Bates S., Alonzo D.E., Taylor L.S. Evaluation of drug-polymer miscibility in amorphous solid dispersion systems. Pharm. Res. 2009, 26:2523-2534.
    • (2009) Pharm. Res. , vol.26 , pp. 2523-2534
    • Rumondor, A.C.F.1    Ivanisevic, I.2    Bates, S.3    Alonzo, D.E.4    Taylor, L.S.5
  • 20
    • 70449107051 scopus 로고    scopus 로고
    • Effects of polymer type and storage relative humidity on the kinetics of felodipine crystallization from amorphous solid dispersions
    • Rumondor A.C.F., Stanford L.A., Taylor L.S. Effects of polymer type and storage relative humidity on the kinetics of felodipine crystallization from amorphous solid dispersions. Pharm. Res. 2009, 26:2599-2606.
    • (2009) Pharm. Res. , vol.26 , pp. 2599-2606
    • Rumondor, A.C.F.1    Stanford, L.A.2    Taylor, L.S.3
  • 21
    • 0032885450 scopus 로고    scopus 로고
    • Solid dispersion of poorly water-soluble drugs: early promises, subsequent problems, and recent breakthroughs
    • Serajuddin A.T.M. Solid dispersion of poorly water-soluble drugs: early promises, subsequent problems, and recent breakthroughs. J. Pharm. Sci. 1999, 88:1058-1066.
    • (1999) J. Pharm. Sci. , vol.88 , pp. 1058-1066
    • Serajuddin, A.T.M.1
  • 22
    • 0037258305 scopus 로고    scopus 로고
    • Identification of phase separation in solid dispersions of itraconazole and Eudragit E100 using microthermal analysis
    • Six K., Murphy J., Weuts I., Craig D.Q.M., Verreck G., Peeters J., Brewster M., Van den Mooter G. Identification of phase separation in solid dispersions of itraconazole and Eudragit E100 using microthermal analysis. Pharm. Res. 2003, 20:135-138.
    • (2003) Pharm. Res. , vol.20 , pp. 135-138
    • Six, K.1    Murphy, J.2    Weuts, I.3    Craig, D.Q.M.4    Verreck, G.5    Peeters, J.6    Brewster, M.7    Van den Mooter, G.8
  • 24
    • 77956381209 scopus 로고    scopus 로고
    • Solubilities of crystalline drugs in polymers: an improved analytical method and comparison of solubilities of indomethacin and nifedipine in PVP, PVP/VA, and PVAc
    • Sun Y., Tao J., Zhang G.G.Z., Yu L. Solubilities of crystalline drugs in polymers: an improved analytical method and comparison of solubilities of indomethacin and nifedipine in PVP, PVP/VA, and PVAc. J. Pharm. Sci. 2010, 99:4023-4031.
    • (2010) J. Pharm. Sci. , vol.99 , pp. 4023-4031
    • Sun, Y.1    Tao, J.2    Zhang, G.G.Z.3    Yu, L.4
  • 25
    • 61449135800 scopus 로고    scopus 로고
    • Solubility of small-molecule crystals in polymers: d-mannitol in PVP, indomethacin in PVP/VA, and nifedipine in PVP/VA
    • Tao J., Sun Y., Zhang G.G.Z., Yu L. Solubility of small-molecule crystals in polymers: d-mannitol in PVP, indomethacin in PVP/VA, and nifedipine in PVP/VA. Pharm. Res. 2009, 26:855-864.
    • (2009) Pharm. Res. , vol.26 , pp. 855-864
    • Tao, J.1    Sun, Y.2    Zhang, G.G.Z.3    Yu, L.4
  • 26
    • 17644395269 scopus 로고    scopus 로고
    • Phase behavior of amorphous molecular dispersions II: role of hydrogen bonding in solid solubility and phase separation kinetics
    • Vasanthavada M., Tong W.Q., Joshi Y., Kislalioglu M.S. Phase behavior of amorphous molecular dispersions II: role of hydrogen bonding in solid solubility and phase separation kinetics. Pharm. Res. 2005, 22:440-448.
    • (2005) Pharm. Res. , vol.22 , pp. 440-448
    • Vasanthavada, M.1    Tong, W.Q.2    Joshi, Y.3    Kislalioglu, M.S.4
  • 27
    • 36549042006 scopus 로고    scopus 로고
    • Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs
    • Vasconcelos T., Sarmento B., Costa P. Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs. Drug Discov. Today 2007, 12:1068-1075.
    • (2007) Drug Discov. Today , vol.12 , pp. 1068-1075
    • Vasconcelos, T.1    Sarmento, B.2    Costa, P.3
  • 28
    • 55749113671 scopus 로고    scopus 로고
    • Miscibility and interactions between 17β-estradiol and Eudragit RS in solid dispersion
    • Wiranidchapong C., Tucker I.G., Rades T., Kulvanich P. Miscibility and interactions between 17β-estradiol and Eudragit RS in solid dispersion. J. Pharm. Sci. 2008, 97:4879-4887.
    • (2008) J. Pharm. Sci. , vol.97 , pp. 4879-4887
    • Wiranidchapong, C.1    Tucker, I.G.2    Rades, T.3    Kulvanich, P.4
  • 29
    • 33645162736 scopus 로고    scopus 로고
    • Characteristics of konjac glucomannan and poly(acrylic acid) blend films for controlled drug release
    • Yu H.Q., Huang A.B., Xiao C.B. Characteristics of konjac glucomannan and poly(acrylic acid) blend films for controlled drug release. J. Appl. Polym. Sci. 2006, 100:1561-1570.
    • (2006) J. Appl. Polym. Sci. , vol.100 , pp. 1561-1570
    • Yu, H.Q.1    Huang, A.B.2    Xiao, C.B.3
  • 30
    • 0035897584 scopus 로고    scopus 로고
    • Amorphous pharmaceutical solids: preparation, characterization and stabilization
    • Yu L. Amorphous pharmaceutical solids: preparation, characterization and stabilization. Adv. Drug Deliv. Rev. 2001, 48:27-42.
    • (2001) Adv. Drug Deliv. Rev. , vol.48 , pp. 27-42
    • Yu, L.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.