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Volumn 6, Issue 5, 2009, Pages 1492-1505

Phase behavior of poly(vinylpyrrolidone) containing amorphous solid dispersions in the presence of moisture

Author keywords

Amorphous; Crystallization; Miscibility; Moisture; Solid dispersion

Indexed keywords

DROPERIDOL; FELODIPINE; INDOMETACIN; KETOPROFEN; NIFEDIPINE; PIMOZIDE; POVIDONE;

EID: 70350057599     PISSN: 15438384     EISSN: 15438392     Source Type: Journal    
DOI: 10.1021/mp900050c     Document Type: Conference Paper
Times cited : (194)

References (45)
  • 1
    • 0015124656 scopus 로고
    • Pharmaceutical Applications of Solid Dispersion Systems
    • Chiou, W. L.; Riegelman, S. Pharmaceutical Applications Of Solid Dispersion Systems. J. Pharm. Sci. 1971, 60 (9), 1281-1302.
    • (1971) J. Pharm. Sci. , vol.60 , Issue.9 , pp. 1281-1302
    • Chiou, W.L.1    Riegelman, S.2
  • 2
    • 0030638567 scopus 로고    scopus 로고
    • Characteristics and Significance of the Amorphous State in Pharmaceutical Systems
    • Review
    • Hancock, B. C.; Zografi, G. Characteristics and Significance of the Amorphous State in Pharmaceutical Systems [Review]. J. Pharm. Sci. 1997, 86 (1), 1-12.
    • (1997) J. Pharm. Sci. , vol.86 , Issue.1 , pp. 1-12
    • Hancock, B.C.1    Zografi, G.2
  • 3
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • DOI 10.1016/S0939-6411(00)00076-X, PII S093964110000076X
    • Leuner, C.; Dressman, J. Improving drug solubility for oral delivery using solid dispersions. Eur. J. Pharm. Biopharm. 2000, 50 (1), 47-60. (Pubitemid 30326688)
    • (2000) European Journal of Pharmaceutics and Biopharmaceutics , vol.50 , Issue.1 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 4
    • 0035897584 scopus 로고    scopus 로고
    • Amorphous pharmaceutical solids: Preparation, characterization and stabilization
    • Yu, L. Amorphous pharmaceutical solids: preparation, characterization and stabilization. Adv. Drug Delivery Rev. 2001, 48 (1), 27-42.
    • (2001) Adv. Drug Delivery Rev. , vol.48 , Issue.1 , pp. 27-42
    • Yu, L.1
  • 5
    • 0018379090 scopus 로고
    • Cefoxitin Sodium - Solution and Solid-State Chemical-Stability Studies
    • Oberholtzer, E. R.; Brenner, G. S. Cefoxitin Sodium - Solution and Solid-State Chemical-Stability Studies. J. Pharm. Sci. 1979, 68 (7), 863-866.
    • (1979) J. Pharm. Sci. , vol.68 , Issue.7 , pp. 863-866
    • Oberholtzer, E.R.1    Brenner, G.S.2
  • 6
    • 0017857869 scopus 로고
    • Quantitative crystallinity determinations for β-lactam antibiotics by solution calorimetry: Correlations with stability
    • Pikal, M. J.; Lukes, A. L.; Lang, J. E.; Gaines, K. Quantitative Crystallinity Determinations for Beta-Lactam Antibiotics by Solution Calorimetry - Correlations with Stability. J. Pharm. Sci. 1978, 67 (6), 767-772. (Pubitemid 8355230)
    • (1978) Journal of Pharmaceutical Sciences , vol.67 , Issue.6 , pp. 767-773
    • Pikal, M.J.1    Lukes, A.L.2    Lang, J.E.3    Gaines, K.4
  • 7
    • 0033707107 scopus 로고    scopus 로고
    • Crystal nucleation and growth of indomethacin polymorphs from the amorphous state
    • DOI 10.1016/S0022-3093(00)00107-1
    • Andronis, V.; Zografi, G. Crystal nucleation and growth of indomethacin polymorphs from the amorphous state. J. Non -Cryst. Solids 2000, 271 (3), 236-248. (Pubitemid 30876406)
    • (2000) Journal of Non-Crystalline Solids , vol.271 , Issue.3 , pp. 236-248
    • Andronis, V.1    Zografi, G.2
  • 8
    • 0027275797 scopus 로고
    • The use of solution theories for predicting water vapor absorption by amorphous pharmaceutical solids: A test of the Flory-Huggins and Vrentas models
    • DOI 10.1023/A:1018901325842
    • Hancock, B. C.; Zografi, G. The use of solution theories for predicting water vapor absorption by amorphous pharmaceutical solids: A test of the Flory-Huggins and Vrentas models. Pharm. Res. 1993, 10 (9), 1262-1267. (Pubitemid 23261823)
    • (1993) Pharmaceutical Research , vol.10 , Issue.9 , pp. 1262-1267
    • Hancock, B.C.1    Zografi, G.2
  • 9
    • 0031056536 scopus 로고    scopus 로고
    • Effects of sorbed water on the crystallization of indomethacin from the amorphous state
    • DOI 10.1021/js9602711
    • Andronis, V.; Yoshioka, M.; Zografi, G. Effects of sorbed water on the crystallization of indomethacin from the amorphous state. J. Pharm. Sci. 1997, 86 (3), 346-351. (Pubitemid 27113770)
    • (1997) Journal of Pharmaceutical Sciences , vol.86 , Issue.3 , pp. 346-357
    • Andronis, V.1    Yoshioka, M.2    Zografi, G.3
  • 10
    • 0032784693 scopus 로고    scopus 로고
    • The effects of absorbed water on the properties of amorphous mixtures containing sucrose
    • DOI 10.1023/A:1018960405504
    • Shamblin, S. L.; Zografi, G. The effects of absorbed water on the properties of amorphous mixtures containing sucrose. Pharm. Res. 1999, 16 (7), 1119-1124. (Pubitemid 29368163)
    • (1999) Pharmaceutical Research , vol.16 , Issue.7 , pp. 1119-1124
    • Shamblin, S.L.1    Zografi, G.2
  • 11
    • 0022650603 scopus 로고
    • The Current Status of Solid Dispersions
    • Ford, J. L. The Current Status of Solid Dispersions. Pharm. Acta HelV. 1986, 61, 69-88.
    • (1986) Pharm. Acta HelV. , vol.61 , pp. 69-88
    • Ford, J.L.1
  • 12
    • 0028147099 scopus 로고
    • Nonisothermal and Isothermal Crystallization of Sucrose from the Amorphous State
    • Saleki-Gerhardt, A.; Zografi, G. Nonisothermal And Isothermal Crystallization Of Sucrose From The Amorphous State. Pharm. Res. 1994, 11 (8), 1166-1173.
    • (1994) Pharm. Res. , vol.11 , Issue.8 , pp. 1166-1173
    • Saleki-Gerhardt, A.1    Zografi, G.2
  • 13
    • 0034943639 scopus 로고    scopus 로고
    • Fourier transform Raman spectroscopic study of the interaction of water vapor with amorphous polymers
    • DOI 10.1002/jps.1041
    • Taylor, L. S.; Langkilde, F. W.; Zografi, G. Fourier transform Raman spectroscopic study of the interaction of water vapor with amorphous polymers. J. Pharm. Sci. 2001, 90 (7), 888-901. (Pubitemid 32645946)
    • (2001) Journal of Pharmaceutical Sciences , vol.90 , Issue.7 , pp. 888-901
    • Taylor, L.S.1    Langkilde, F.W.2    Zografi, G.3
  • 14
    • 0036599307 scopus 로고    scopus 로고
    • 13C-NMR relaxation time
    • DOI 10.1248/cpb.50.822
    • Aso, Y.; Yoshioka, S.; Zhang, J.; Zografi, G. Effect of water on the molecular mobility of sucrose and poly(vinylpyrrolidone) in a colyophilized formulation as measured by C-13-NMR relaxation time. Chem. Pharm. Bull. 2002, 50 (6), 822-826. (Pubitemid 41694902)
    • (2002) Chemical and Pharmaceutical Bulletin , vol.50 , Issue.6 , pp. 822-826
    • Aso, Y.1    Yoshioka, S.2    Zhang, J.3    Zografi, G.4
  • 15
    • 40549086641 scopus 로고    scopus 로고
    • Recrystallization of nifedipine and felodipine from amorphous molecular level solid dispersions containing poly(vinylpyrrolidone) and sorbed water
    • Marsac, P. J.; Konno, H.; Rumondor, A. C. F.; Taylor, L. S. Recrystallization of nifedipine and felodipine from amorphous molecular level solid dispersions containing poly(vinylpyrrolidone) and sorbed water. Pharm. Res. 2008, 25 (3), 647-656.
    • (2008) Pharm. Res. , vol.25 , Issue.3 , pp. 647-656
    • Marsac, P.J.1    Konno, H.2    Rumondor, A.C.F.3    Taylor, L.S.4
  • 16
    • 43349097105 scopus 로고    scopus 로고
    • Ability of different polymers to inhibit the crystallization of amorphous felodipine in the presence of moisture
    • Konno, H.; Taylor, L. S. Ability of different polymers to inhibit the crystallization of amorphous felodipine in the presence of moisture. Pharm. Res. 2008, 25 (4), 969-978.
    • (2008) Pharm. Res. , vol.25 , Issue.4 , pp. 969-978
    • Konno, H.1    Taylor, L.S.2
  • 18
    • 17644395269 scopus 로고    scopus 로고
    • Phase behavior of amorphous molecular dispersions - II: Role of hydrogen bonding in solid solubility and phase separation kinetics
    • Vasanthavada, M.; Tong, W. Q.; Joshi, Y.; Kislalioglu, M. S. Phase behavior of amorphous molecular dispersions - II: Role of hydrogen bonding in solid solubility and phase separation kinetics. Pharm. Res. 2005, 22 (3), 440-448.
    • (2005) Pharm. Res. , vol.22 , Issue.3 , pp. 440-448
    • Vasanthavada, M.1    Tong, W.Q.2    Joshi, Y.3    Kislalioglu, M.S.4
  • 19
    • 0031423468 scopus 로고    scopus 로고
    • Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions
    • DOI 10.1023/A:1012167410376
    • Taylor, L. S.; Zografi, G. Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions. Pharm. Res. 1997, 14 (12), 1691-1698. (Pubitemid 28062912)
    • (1997) Pharmaceutical Research , vol.14 , Issue.12 , pp. 1691-1698
    • Taylor, L.S.1    Zografi, G.2
  • 20
    • 26444493103 scopus 로고    scopus 로고
    • Preparation and evaluation of solid dispersion for nitrendipine-Carbopol and nitrendipine-HPMCP systems using a twin screw extruder
    • Wang, L. A.; Cui, F. D.; Hayase, T.; Sunada, H. Preparation and evaluation of solid dispersion for nitrendipine-Carbopol and nitrendipine-HPMCP systems using a twin screw extruder. Chem. Pharm. Bull. 2005, 53 (10), 1240-1245.
    • (2005) Chem. Pharm. Bull. , vol.53 , Issue.10 , pp. 1240-1245
    • Wang, L.A.1    Cui, F.D.2    Hayase, T.3    Sunada, H.4
  • 21
    • 33749447574 scopus 로고    scopus 로고
    • A comparison of the physical stability of amorphous felodipine and nifedipine systems
    • Marsac, P. J.; Konno, H.; Taylor, L. S. A comparison of the physical stability of amorphous felodipine and nifedipine systems. Pharm. Res. 2006, 23 (10), 2306-2316.
    • (2006) Pharm. Res. , vol.23 , Issue.10 , pp. 2306-2316
    • Marsac, P.J.1    Konno, H.2    Taylor, L.S.3
  • 22
    • 0031664813 scopus 로고    scopus 로고
    • Phase behavior of binary and ternary amorphous mixtures containing indomethacin, citric acid, and PVP
    • DOI 10.1023/A:1011983606606
    • Lu, Q.; Zografi, G. Phase behavior of binary and ternary amorphous mixtures containing indomethacin, citric acid, and PVP. Pharm. Res. 1998, 15 (8), 1202-1206. (Pubitemid 28401710)
    • (1998) Pharmaceutical Research , vol.15 , Issue.8 , pp. 1202-1206
    • Lu, Q.1    Zografi, G.2
  • 23
    • 0037258305 scopus 로고    scopus 로고
    • Identification of phase separation in solid dispersions of itraconazole and Eudragit (R) E100 using microthermal analysis
    • Six, K.; Murphy, J.; Weuts, I.; Craig, D. Q. M.; Verreck, G.; Peeters, J.; Brewster, M.; Van den Mooter, G. Identification of phase separation in solid dispersions of itraconazole and Eudragit (R) E100 using microthermal analysis. Pharm. Res. 2003, 20 (1), 135-138.
    • (2003) Pharm. Res. , vol.20 , Issue.1 , pp. 135-138
    • Six, K.1    Murphy, J.2    Weuts, I.3    Craig, D.Q.M.4    Verreck, G.5    Peeters, J.6    Brewster, M.7    Van Den Mooter, G.8
  • 25
    • 2442648607 scopus 로고    scopus 로고
    • Polymorphism and devitrification of nifedipine under controlled humidity: A combined FT-Raman, IR and Raman microscopic investigation
    • Chan, K. L. A.; Fleming, O. S.; Kazarian, S. G.; Vassou, D.; Chryssikos, G. D.; Gionis, V. Polymorphism and devitrification of nifedipine under controlled humidity: a combined FT-Raman, IR and Raman microscopic investigation. J. Raman Spectrosc. 2004, 35 (5), 353-359.
    • (2004) J. Raman Spectrosc. , vol.35 , Issue.5 , pp. 353-359
    • Chan, K.L.A.1    Fleming, O.S.2    Kazarian, S.G.3    Vassou, D.4    Chryssikos, G.D.5    Gionis, V.6
  • 26
    • 0035092508 scopus 로고    scopus 로고
    • Conformational color polymorphism and control of crystallization of 5-methyl-2-[(4-methy1-2-nitrophenyl)amino]-3-thiophenecarbonitrile
    • He, X. R.; Griesser, U. J.; Stowell, J. G.; Borchardt, T. B.; Byrn, S. R. Conformational color polymorphism and control of crystallization of 5-methyl-2-[(4-methy1-2-nitrophenyl)amino]-3-thiophenecarbonitrile. J. Pharm. Sci. 2001, 90 (3), 371-388.
    • (2001) J. Pharm. Sci. , vol.90 , Issue.3 , pp. 371-388
    • He, X.R.1    Griesser, U.J.2    Stowell, J.G.3    Borchardt, T.B.4    Byrn, S.R.5
  • 29
    • 0036786457 scopus 로고    scopus 로고
    • Water vapor absorption into amorphous hydrophobic drug/ poly(vinylpyrrolidone) dispersions
    • DOI 10.1002/jps.10205
    • Crowley, K. J.; Zografi, G. Water vapor absorption into amorphous hydrophobic drug/poly(vinylpyrrolidone) dispersions. J. Pharm. Sci. 2002, 91 (10), 2150-2165. (Pubitemid 35050700)
    • (2002) Journal of Pharmaceutical Sciences , vol.91 , Issue.10 , pp. 2150-2165
    • Crowley, K.J.1    Zografi, G.2
  • 32
    • 36849125484 scopus 로고
    • Thermodynamic Driving Force in Nucleation and Growth Processes
    • Hoffman, J. D. Thermodynamic Driving Force In Nucleation And Growth Processes. J. Chem. Phys. 1958, 29 (5), 1192-1193.
    • (1958) J. Chem. Phys. , vol.29 , Issue.5 , pp. 1192-1193
    • Hoffman, J.D.1
  • 33
    • 57749206650 scopus 로고    scopus 로고
    • Estimation of Drug-Polymer Miscibility and Solubility in Amorphous Solid Dispersions Using Experimentally Determined Interaction Parameters
    • Marsac, P. J.; Li, T.; Taylor, L. S. Estimation of Drug-Polymer Miscibility and Solubility in Amorphous Solid Dispersions Using Experimentally Determined Interaction Parameters. Pharm. Res. 2009, 26 (1), 139-151.
    • (2009) Pharm. Res. , vol.26 , Issue.1 , pp. 139-151
    • Marsac, P.J.1    Li, T.2    Taylor, L.S.3
  • 34
    • 1842510723 scopus 로고    scopus 로고
    • Mixing of the organic aerosol fractions: Liquids as the thermodynamically stable phases
    • Marcolli, C.; Luo, B. P.; Peter, T. Mixing of the organic aerosol fractions: Liquids as the thermodynamically stable phases. J. Phys. Chem. A 2004, 108 (12), 2216-2224.
    • (2004) J. Phys. Chem. A , vol.108 , Issue.12 , pp. 2216-2224
    • Marcolli, C.1    Luo, B.P.2    Peter, T.3
  • 36
    • 0034820643 scopus 로고    scopus 로고
    • Water vapor absorption into amorphous sucrose-poly(vinyl pyrrolidone) and trehalose-poly(vinyl pyrrolidone) mixtures
    • DOI 10.1002/jps.1090
    • Zhang, J.; Zografi, G. Water vapor absorption into amorphous sucrose-poly(vinyl pyrrolidone) and trehalose-poly(vinyl pyrrolidone) mixtures. J. Pharm. Sci. 2001, 90 (9), 1375-1385. (Pubitemid 32867986)
    • (2001) Journal of Pharmaceutical Sciences , vol.90 , Issue.9 , pp. 1375-1385
    • Zhang, J.1    Zografi, G.2
  • 37
    • 34548049521 scopus 로고    scopus 로고
    • Impact of water on the miscibility of DAB-dendr-(NH2)(64) and benzene
    • Gregorowicz, J.; Luszczyk, M. Impact of water on the miscibility of DAB-dendr-(NH2)(64) and benzene. Macromolecules 2007, 40 (16), 5966-5972.
    • (2007) Macromolecules , vol.40 , Issue.16 , pp. 5966-5972
    • Gregorowicz, J.1    Luszczyk, M.2
  • 38
    • 0033811783 scopus 로고    scopus 로고
    • The relationship between "BET"- and "Free volume"-derived parameters for water vapor absorption into amorphous solids
    • Zhang, J.; Zografi, G. The relationship between "BET"- and "Free volume"-derived parameters for water vapor absorption into amorphous solids. J. Pharm. Sci. 2000, 89 (8), 1063-1072.
    • (2000) J. Pharm. Sci. , vol.89 , Issue.8 , pp. 1063-1072
    • Zhang, J.1    Zografi, G.2
  • 39
    • 0037369754 scopus 로고    scopus 로고
    • Formation of physically stable amorphous drugs by milling with Neusilin
    • Gupta, M. K.; Vanwert, A.; Bogner, R. H. Formation of physically stable amorphous drugs by milling with Neusilin. J. Pharm. Sci. 2003, 92 (3), 536-551.
    • (2003) J. Pharm. Sci. , vol.92 , Issue.3 , pp. 536-551
    • Gupta, M.K.1    Vanwert, A.2    Bogner, R.H.3
  • 42
    • 0035209946 scopus 로고    scopus 로고
    • A study of amorphous molecular dispersions of indomethacin and its sodium salt
    • DOI 10.1002/jps.1150
    • Tong, P.; Zografi, G. A study of amorphous molecular dispersions of indomethacin and its sodium salt. J. Pharm. Sci. 2001, 90 (12), 1991-2004. (Pubitemid 33144445)
    • (2001) Journal of Pharmaceutical Sciences , vol.90 , Issue.12 , pp. 1991-2004
    • Tong, P.1    Zografi, G.2
  • 43
    • 39149103092 scopus 로고    scopus 로고
    • The crystal and molecular structure of a polymorph and a pseudo-polymorph of droperidol
    • Actins, A.; Arajs, R.; Belakovs, S.; Orola, L.; Veidis, M. V. The crystal and molecular structure of a polymorph and a pseudo-polymorph of droperidol. J. Chem. Crystallogr. 2008, 38 (3), 169-174.
    • (2008) J. Chem. Crystallogr. , vol.38 , Issue.3 , pp. 169-174
    • Actins, A.1    Arajs, R.2    Belakovs, S.3    Orola, L.4    Veidis, M.V.5
  • 44
    • 0031742175 scopus 로고    scopus 로고
    • A crystallographic and molecular modeling study of butyrophenones
    • DOI 10.1021/js980253e
    • Liang, L.; Zhu, N. J.; White, J.; Brown, C.; Klein-Stevens, C. L. A crystallographic and molecular modeling study of butyrophenones. J. Pharm. Sci. 1998, 87 (12), 1496-1501. (Pubitemid 28559630)
    • (1998) Journal of Pharmaceutical Sciences , vol.87 , Issue.12 , pp. 1496-1501
    • Liang, L.1


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