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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 16, 2010, Pages 4836-4839

Improvement of both plasmepsin inhibitory activity and antimalarial activity by 2-aminoethylamino substitution

(10) Miura, Takuya a Hidaka, Koushi a Uemura, Tsuyoshi a Kashimoto, Keisuke a Hori, Yuto a Kawasaki, Yuko b Ruben, Adam J b Freire, Ernesto b Kimura, Tooru a Kiso, Yoshiaki a

a KYOTO PHARMACEUTICAL UNIVERSITY (Japan)

b JOHNS HOPKINS UNIVERSITY (United States)

Author keywords

Allophenylnorstatine; Antimalarial drug; Aspartic protease; Hydoxymethylcarbonyl; Peptidomimetics; Plasmepsin inhibitor

Indexed keywords

ALLOPHENYLNORSTATINE; ANTIMALARIAL AGENT; ASPARTIC PROTEINASE; CARBONYL DERIVATIVE; CHLOROQUINE; HYDROXYMETHYLCARBONYL; KNI 10006; KNI 10538; KNI 10737; KNI 10740; KNI 10742; KNI 10743; PEPTIDOMIMETIC AGENT; PLASMEPSIN I; PLASMEPSIN II; PLASMEPSIN INHIBITOR; UNCLASSIFIED DRUG; 3-AMINO-2-HYDROXY-4-PHENYLBUTANOIC ACID; ARYLBUTYRIC ACID DERIVATIVE; ETHYLENEDIAMINE DERIVATIVE; PROTEINASE INHIBITOR; PROTOZOAL PROTEIN; THIAZOLE DERIVATIVE;

ANTIMALARIAL ACTIVITY; ARTICLE; DRUG POTENCY; DRUG STRUCTURE; FLUORESCENCE ANALYSIS; MALARIA; MALARIA FALCIPARUM; NONHUMAN; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION; ANTAGONISTS AND INHIBITORS; BINDING SITE; CHEMISTRY; COMPUTER SIMULATION; METABOLISM; SYNTHESIS;

ANTIMALARIALS; ASPARTIC ACID ENDOPEPTIDASES; BINDING SITES; COMPUTER SIMULATION; ETHYLENEDIAMINES; PHENYLBUTYRATES; PROTEASE INHIBITORS; PROTOZOAN PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 77955424007 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.06.099 Document Type: Article

Times cited : (17)

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