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Volumn 18, Issue 15, 2010, Pages 5489-5497

Synthesis and in vivo evaluation of [11C]tariquidar, a positron emission tomography radiotracer based on a third-generation P-glycoprotein inhibitor

(12) Bauer, Florian b,c Kuntner, Claudia a Bankstahl, Jens P d Wanek, Thomas a Bankstahl, Marion d Stanek, Johann a,c Mairinger, Severin a,b,c Dörner, Bernd b Löscher, Wolfgang d Müller, Markus c Erker, Thomas b Langer, Oliver a,c

a AIT AUSTRIAN INSTITUTE OF TECHNOLOGY (Austria)

b UNIVERSITY OF VIENNA (Austria)

c MEDICAL UNIVERSITY OF VIENNA (Austria)

d UNIVERSITY OF VETERINARY MEDICINE HANNOVER (Germany)

Author keywords

11C tariquidar; Blood brain barrier; Breast cancer resistance protein; P glycoprotein; PET

Indexed keywords

ANTINEOPLASTIC AGENT; BREAST CANCER RESISTANCE PROTEIN; BREAST CANCER RESISTANCE PROTEIN 1; CARBON 11; ELACRIDAR; GLYCOPROTEIN P; GLYCOPROTEIN P INHIBITOR; MEMBRANE PROTEIN; METHYLTRIFLATE C 11; MULTIDRUG RESISTANCE PROTEIN 1; MULTIDRUG RESISTANCE PROTEIN 1A; MULTIDRUG RESISTANCE PROTEIN 1B; O DESMETHYL TARIQUIDAR; SULFONIC ACID DERIVATIVE; TARIQUIDAR; TARIQUIDAR C 11; TRACER; UNCLASSIFIED DRUG; ABC TRANSPORTER; ABCG2 PROTEIN, MOUSE; CARBON; MULTIDRUG RESISTANCE PROTEIN; QUINOLINE DERIVATIVE; RADIOPHARMACEUTICAL AGENT;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BLOOD BRAIN BARRIER; BRAIN; CHEMICAL REACTION; CONTROLLED STUDY; DRUG BINDING; DRUG BLOOD LEVEL; DRUG BRAIN LEVEL; DRUG DISTRIBUTION; DRUG SYNTHESIS; DRUG TRANSPORT; ELECTROENCEPHALOGRAM; FEMALE; IN VITRO STUDY; IN VIVO STUDY; INCUBATION TIME; INJECTION; ISOTOPE LABELING; MOUSE; NEUROIMAGING; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RAT; WILD TYPE; ANIMAL; ANTAGONISTS AND INHIBITORS; CHEMISTRY; DIAGNOSTIC USE; KNOCKOUT MOUSE; METABOLISM; SPRAGUE DAWLEY RAT; SYNTHESIS;

ANIMALS; ATP-BINDING CASSETTE TRANSPORTERS; AUTORADIOGRAPHY; BLOOD-BRAIN BARRIER; CARBON RADIOISOTOPES; FEMALE; MICE; MICE, KNOCKOUT; P-GLYCOPROTEIN; POSITRON-EMISSION TOMOGRAPHY; QUINOLINES; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY;

ANIMALIA; MUS; RATTUS;

EID: 77955419945 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2010.06.057 Document Type: Article

Times cited : (66)

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