QSAR study of substituted 1,3,4-oxadiazole naphthyridines as HIV-1 integrase inhibitors

European Journal of Medicinal Chemistry

Volumn 45, Issue 7, 2010, Pages 2791-2797

  Ravichandran, Veerasamy ^a   Shalini, Sivadasan ^a   Sundram, Karupiah ^a   Sokkalingam, Arumugam Dhanaraj ^a  

^a AIMST UNIVERSITY   (Malaysia)

Author keywords

1,3,4 Oxadiazole substituted naphthyridine derivatives; Human immunodeficiency virus; Inhibition; Integrase; Quantitative Structure Activity Relationship

Indexed keywords

1,3,4 OXADIAZOLE NAPHTHYRIDINE; INTEGRASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DATA BASE; DRUG CONFORMATION; DRUG INHIBITION; MULTIPLE LINEAR REGRESSION ANALYSIS; PREDICTIVE VALIDITY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STATISTICAL SIGNIFICANCE;

HIV INTEGRASE; HIV INTEGRASE INHIBITORS; MODELS, MOLECULAR; NAPHTHYRIDINES; OXADIAZOLES; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; REGRESSION ANALYSIS; SOFTWARE;

EID: 77954349380     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2010.02.062     Document Type: Article

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