메뉴 건너뛰기




Volumn 36, Issue 8, 2010, Pages 917-925

Preparation and evaluation of solid dispersions of piroxicam and Eudragit S100 by spherical crystallization technique

Author keywords

Aerosil; Enteric microparticles; Eudragit S100; Piroxicam; Spherical crystallization

Indexed keywords

AEROSIL; EUDRAGIT; PIROXICAM; EXCIPIENT; METHYLMETHACRYLATE-METHACRYLIC ACID COPOLYMER; MICROSPHERE; NONSTEROID ANTIINFLAMMATORY AGENT; POLYMETHACRYLIC ACID DERIVATIVE; SILICON DIOXIDE; SUSPENSION;

EID: 77954203501     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.3109/03639040903585127     Document Type: Article
Times cited : (30)

References (44)
  • 1
    • 0020071251 scopus 로고
    • Pharmacology, clinical efficacy, and adverse effects of piroxicam, a new nonsteroidal anti-inflammatory agent
    • Dahl SL, Ward JR. (1982). Pharmacology, clinical efficacy, and adverse effects of piroxicam, a new nonsteroidal anti-inflammatory agent. Pharmacotherapy, 2:80-89
    • (1982) Pharmacotherapy , vol.2 , pp. 80-89
    • Dahl, S.L.1    Ward, J.R.2
  • 2
    • 0000225791 scopus 로고
    • Pharmacology and therapeutics of non-steroidal anti-inflammatory drugs in the dog and cat: 2 Individual agents
    • Mckellar QA, May SA, Lees P. (1991). Pharmacology and therapeutics of non-steroidal anti-inflammatory drugs in the dog and cat: 2 Individual agents. J Small Anim Pract, 32:225-235
    • (1991) J Small Anim Pract , vol.32 , pp. 225-235
    • McKellar, Q.A.1    May, S.A.2    Lees, P.3
  • 3
    • 0025819464 scopus 로고
    • Pharmacokinetics and pharmacodynamics of piroxicam in dogs
    • Galbraith EA, Mckellar QA. (1991). Pharmacokinetics and pharmacodynamics of piroxicam in dogs. Vet Rec, 128:561-565
    • (1991) Vet Rec , vol.128 , pp. 561-565
    • Galbraith, E.A.1    McKellar, Q.A.2
  • 4
    • 33748430023 scopus 로고    scopus 로고
    • Drug delivery to the upper small intestine window using gastroretentive technologies
    • Streubel A, Siepmann J, Bodmeier R. (2006). Drug delivery to the upper small intestine window using gastroretentive technologies. Curr Opin Pharmacol, 6:501-508
    • (2006) Curr Opin Pharmacol , vol.6 , pp. 501-508
    • Streubel, A.1    Siepmann, J.2    Bodmeier, R.3
  • 5
    • 33645758286 scopus 로고    scopus 로고
    • Development of novel sustained-release system, disintegration-controlled matrix tablet (DCMT) with solid dispersion granules of nilvadipine (II): In vivo evaluation
    • Tanaka N, Imai K, Okimoto K, Ueda S, Tokunaga Y, Ibuki R, et al. (2006). Development of novel sustained-release system, disintegration-controlled matrix tablet (DCMT) with solid dispersion granules of nilvadipine (II): In vivo evaluation. J Control Release, 112:51-56
    • (2006) J Control Release , vol.112 , pp. 51-56
    • Tanaka, N.1    Imai, K.2    Okimoto, K.3    Ueda, S.4    Tokunaga, Y.5    Ibuki, R.6
  • 6
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • Leuner C, Dressman J. (2000). Improving drug solubility for oral delivery using solid dispersions. Eur J Pharm Biopharm, 50:47-60.
    • (2000) Eur J Pharm Biopharm , vol.50 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 7
    • 33845484838 scopus 로고    scopus 로고
    • Bioavailability enhancement of an active substance by supercritical antisolvent precipitation
    • Majerik V, Charbit G, Badens E, Horvath G, Szokonya L, Bosc N, et al. (2007). Bioavailability enhancement of an active substance by supercritical antisolvent precipitation. J Supercrit Fluids, 40:101-110
    • (2007) J Supercrit Fluids , vol.40 , pp. 101-110
    • Majerik, V.1    Charbit, G.2    Badens, E.3    Horvath, G.4    Szokonya, L.5    Bosc, N.6
  • 8
    • 23944483499 scopus 로고    scopus 로고
    • Novel lipid-based formulations enhancing the in vitro dissolution and permeability characteristics of a poorly water-soluble model drug, piroxicam
    • Prabhu S, Ortega M, Ma Ch. (2005). Novel lipid-based formulations enhancing the in vitro dissolution and permeability characteristics of a poorly water-soluble model drug, piroxicam. Int J Pharm, 301:209-216
    • (2005) Int J Pharm , vol.301 , pp. 209-216
    • Prabhu, S.1    Ortega, M.2    Ma, Ch.3
  • 9
    • 21444460249 scopus 로고    scopus 로고
    • Tolerance and clinical evaluation of piroxicam in dogs
    • Sumano H, Devizcaya A. (1996). Tolerance and clinical evaluation of piroxicam in dogs. Canine Pract, 21:16-19
    • (1996) Canine Pract , vol.21 , pp. 16-19
    • Sumano, H.1    Devizcaya, A.2
  • 10
    • 0029758444 scopus 로고    scopus 로고
    • Nonsteroidal anti-inflammatory drug-induced gastrointestinal injury
    • Bjorkman DJ. (1996). Nonsteroidal anti-inflammatory drug-induced gastrointestinal injury. Am J Med, 101:S25-S32.
    • (1996) Am J Med , vol.101
    • Bjorkman, D.J.1
  • 11
    • 0014815890 scopus 로고
    • Oral absorption of griseofulvin in dogs: Increased absorption via solid dispersion in polyethylene glycol 6000
    • Chiou WL, Riegelman S. (1970). Oral absorption of griseofulvin in dogs: Increased absorption via solid dispersion in polyethylene glycol 6000. J Pharm Sci, 59:937-942
    • (1970) J Pharm Sci , vol.59 , pp. 937-942
    • Chiou, W.L.1    Riegelman, S.2
  • 12
    • 85008071016 scopus 로고
    • Studies on absorption of eutectic mixture. I. A comparison of the behavior of eutectic mixture of sulfathiazole and that of ordinary sulfathiazole in man
    • Sekiguchi K, Obi N. (1961). Studies on absorption of eutectic mixture. I. A comparison of the behavior of eutectic mixture of sulfathiazole and that of ordinary sulfathiazole in man. Chem Pharm Bull, 9:866-872
    • (1961) Chem Pharm Bull , vol.9 , pp. 866-872
    • Sekiguchi, K.1    Obi, N.2
  • 13
    • 0013795160 scopus 로고
    • Increasing dissolution rates and gastrointestinal absorption of drugs via solid solutions and eutectic mixtures.I. Theoretical considerations and discussion of the literature
    • Goldberg AH, Gibaldi M, Kamig JL. (1965). Increasing dissolution rates and gastrointestinal absorption of drugs via solid solutions and eutectic mixtures. I. Theoretical considerations and discussion of the literature. J Pharm Sci, 54:1145-1148
    • (1965) J Pharm Sci , vol.54 , pp. 1145-1148
    • Goldberg, A.H.1    Gibaldi, M.2    Kamig, J.L.3
  • 14
    • 0015124656 scopus 로고
    • Pharmaceutical applications of solid dispersion systems
    • Chiou WL, Reigelman S. (1971). Pharmaceutical applications of solid dispersion systems. J Pharm Sci, 60:1281-1302
    • (1971) J Pharm Sci , vol.60 , pp. 1281-1302
    • Chiou, W.L.1    Reigelman, S.2
  • 15
    • 0022650603 scopus 로고
    • The current status of solid dispersions
    • Ford JL. (1986). The current status of solid dispersions. Pharm Acta Helv, 61:69-88.
    • (1986) Pharm Acta Helv , vol.61 , pp. 69-88
    • Ford, J.L.1
  • 16
    • 0001000807 scopus 로고
    • Spherical crystallization: Direct spherical agglomeration of salicylic acid crystals during crystallization
    • Kawashima Y, Okumura M, Takenaka H. (1982). Spherical crystallization: Direct spherical agglomeration of salicylic acid crystals during crystallization. Science, 216:1127-1128
    • (1982) Science , vol.216 , pp. 1127-1128
    • Kawashima, Y.1    Okumura, M.2    Takenaka, H.3
  • 17
    • 0037453819 scopus 로고    scopus 로고
    • Improved flowability and compactibility of spherically agglomerated crystals of ascorbic acid for direct tableting designed by spherical crystallization process
    • Kawashima Y, Imai M, Takeuchi H, Yamamoto H, Kamiya K, Hino T. (2003). Improved flowability and compactibility of spherically agglomerated crystals of ascorbic acid for direct tableting designed by spherical crystallization process. Powder Technol, 130:283-289
    • (2003) Powder Technol , vol.130 , pp. 283-289
    • Kawashima, Y.1    Imai, M.2    Takeuchi, H.3    Yamamoto, H.4    Kamiya, K.5    Hino, T.6
  • 18
    • 36749088151 scopus 로고    scopus 로고
    • Improved compaction and packing properties of naproxen agglomerated crystals obtained by spherical crystallization technique
    • Maghsoodi M, Hassan-zadeh D, Barzegar-jalali M, Nokhodchi A, Martin G. (2007). Improved compaction and packing properties of naproxen agglomerated crystals obtained by spherical crystallization technique. Drug Dev Ind Pharm, 33:1216-1224
    • (2007) Drug Dev Ind Pharm , vol.33 , pp. 1216-1224
    • Maghsoodi, M.1    Hassan-Zadeh, D.2    Barzegar-Jalali, M.3    Nokhodchi, A.4    Martin, G.5
  • 19
    • 0029965779 scopus 로고    scopus 로고
    • Preparation of controlled releasing acrylic polymer microspheres of acebutolol hydrochloride and those powder coated microspheres with sodium alginate in a polymeric spherical crystallization system
    • Cui FD, Kawashima Y, Takeuchi H, Niwa T, Hino T. (1996). Preparation of controlled releasing acrylic polymer microparti-cles of acebutolol hydrochloride and microparticles with sodium alginate in a polymeric spherical crystallization system. Chem Pharm Bull, 44:837-842 (Pubitemid 26149886)
    • (1996) Chemical and Pharmaceutical Bulletin , vol.44 , Issue.4 , pp. 837-842
    • Cui, F.1    Kawashima, Y.2    Takeuchi, H.3    Niwa, T.4    Hino, T.5
  • 20
    • 70350647611 scopus 로고    scopus 로고
    • Preparation of microparticles of naproxen with Eudragit RS and Talc by spherical crystallization technique
    • Maghsoodi M, Esfahani M. (2009). Preparation of microparticles of naproxen with Eudragit RS and Talc by spherical crystallization technique. Pharm Dev Technol, 14(4):442-450
    • (2009) Pharm Dev Technol , vol.14 , Issue.4 , pp. 442-450
    • Maghsoodi, M.1    Esfahani, M.2
  • 21
    • 0028207193 scopus 로고
    • Preparation of agglomerated crystals for direct tablet-ting and microencapsulation by the spherical crystallization technique with a continuous system
    • Niwa T, Takeuchi H, Hino T, Itoh A, Kawashima Y, Kiuchi K. (1994). Preparation of agglomerated crystals for direct tablet-ting and microencapsulation by the spherical crystallization technique with a continuous system. Pharm Res, 11:478-484
    • (1994) Pharm Res , vol.11 , pp. 478-484
    • Niwa, T.1    Takeuchi, H.2    Hino, T.3    Itoh, A.4    Kawashima, Y.5    Kiuchi, K.6
  • 22
    • 0025799715 scopus 로고
    • Preparation of multiple unit hollow microparticles (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vitro)
    • Kawashima Y, Niwa T, Kakeuchi H, Hino T, Itoh Y. (1991). Preparation of multiple unit hollow microparticles (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vitro). J Control Release, 16:279-290
    • (1991) J Control Release , vol.16 , pp. 279-290
    • Kawashima, Y.1    Niwa, T.2    Kakeuchi, H.3    Hino, T.4    Itoh, Y.5
  • 23
    • 0027155794 scopus 로고
    • Preparation of biodegradable nanospheres of water-soluble and insoluble drugs with DL-lactide/glycolide copolymer by a novel spontaneous emulsification solvent diffusion method and the drug release behavior
    • Niwa T, Takeuchi H, Hino T, Kunou N, Kawashima Y. (1993). Preparation of biodegradable nanospheres of water-soluble and insoluble drugs with DL-lactide/glycolide copolymer by a novel spontaneous emulsification solvent diffusion method and the drug release behavior. J Control Release, 25:89-98.
    • (1993) J Control Release , vol.25 , pp. 89-98
    • Niwa, T.1    Takeuchi, H.2    Hino, T.3    Kunou, N.4    Kawashima, Y.5
  • 24
    • 0042735320 scopus 로고
    • Spherical crystallization as a novel particle design technique for oral drug delivery system
    • Kawashima Y. (1989). Spherical crystallization as a novel particle design technique for oral drug delivery system. Chin Pharm J, 41:163-172
    • (1989) Chin Pharm J , vol.41 , pp. 163-172
    • Kawashima, Y.1
  • 26
    • 0007591301 scopus 로고
    • The flow properties of magnesia
    • Pilpel N. (1964). The flow properties of magnesia. J Pharm Pharmacol, 16:705-716
    • (1964) J Pharm Pharmacol , vol.16 , pp. 705-716
    • Pilpel, N.1
  • 27
    • 0000496231 scopus 로고
    • Evaluation flow properties of solids
    • Carr RL. (1965). Evaluation flow properties of solids. Chem Eng, 72:163-168
    • (1965) Chem Eng , vol.72 , pp. 163-168
    • Carr, R.L.1
  • 28
    • 0000496232 scopus 로고
    • Classify flow properties of solids
    • Carr RL. (1965). Classify flow properties of solids. Chem Eng, 72:69-72.
    • (1965) Chem Eng , vol.72 , pp. 69-72
    • Carr, R.L.1
  • 29
    • 0033082386 scopus 로고    scopus 로고
    • Preparation of microparticles of Keto-profen with acrylic polymers by a quasi-emulsion solvent diffusion method
    • Re MI, Biscans B. (1999). Preparation of microparticles of Keto-profen with acrylic polymers by a quasi-emulsion solvent diffusion method. Powder Technol, 101:120-133
    • (1999) Powder Technol , vol.101 , pp. 120-133
    • Re, M.I.1    Biscans, B.2
  • 30
    • 0033998382 scopus 로고    scopus 로고
    • Spherical crystal agglomeration of ibuprofen by the solvent-change technique in presence of methacrylic polymers
    • Kachrimanis K, Nikolakakis I, Malamataris S. (2000). Spherical crystal agglomeration of ibuprofen by the solvent-change technique in presence of methacrylic polymers. J Pharm Sci, 89(2):250-258
    • (2000) J Pharm Sci , vol.89 , Issue.2 , pp. 250-258
    • Kachrimanis, K.1    Nikolakakis, I.2    Malamataris, S.3
  • 31
    • 0029080004 scopus 로고
    • Production and characterization of enteric beads
    • Zaniboni HC, Fell JT, Collett JH. (1995). Production and characterization of enteric beads. Int J Pharm, 125:151-155
    • (1995) Int J Pharm , vol.125 , pp. 151-155
    • Zaniboni, H.C.1    Fell, J.T.2    Collett, J.H.3
  • 33
    • 0037685276 scopus 로고    scopus 로고
    • Preparation of sustained-release nitrendipine microparticles with eudragit RS and aerosil using quasi-emulsion solvent diffusion method
    • Yang MS, Cui F, You B, Fan Y, Wang L, Yue P, et al. (2003). Preparation of sustained-release nitrendipine microparticles with Eudragit RS and Aerosil using quasi-emulsion solvent diffusion method. Int J Pharm, 259:103-113
    • (2003) Int J Pharm , vol.259 , pp. 103-113
    • Yang, M.S.1    Cui, F.2    You, B.3    Fan, Y.4    Wang, L.5    Yue, P.6
  • 34
    • 0026585145 scopus 로고
    • Hollow microparticles for use as a floating controlled drug delivery system in the stomach
    • Kawashima Y, Niwa T, Takeuchi H, Hino T, Itoh Y. (1992). Hollow microparticles for use as a floating controlled drug delivery system in the stomach. J Pharm Sci, 81(2):135-140
    • (1992) J Pharm Sci , vol.81 , Issue.2 , pp. 135-140
    • Kawashima, Y.1    Niwa, T.2    Takeuchi, H.3    Hino, T.4    Itoh, Y.5
  • 36
    • 0032940583 scopus 로고    scopus 로고
    • Properties of solid dispersions of piroxicam in polyvi-nylpyrrolidone
    • Tantishaiyakul V, Kaewnopparat N, Ingkatawornwong S. (1999). Properties of solid dispersions of piroxicam in polyvi-nylpyrrolidone. Int J Pharm, 181:143-151
    • (1999) Int J Pharm , vol.181 , pp. 143-151
    • Tantishaiyakul, V.1    Kaewnopparat, N.2    Ingkatawornwong, S.3
  • 37
    • 77956907571 scopus 로고
    • Piroxicam
    • Florey, K, ed London: Academic Press
    • Mihalic M. (1986). Piroxicam. In: Florey, K, ed. Analytical profiles of drug substances, vol.15. London: Academic Press, 509-531
    • (1986) Analytical Profiles of Drug Substances , vol.15 , pp. 509-531
    • Mihalic, M.1
  • 38
    • 0037473468 scopus 로고    scopus 로고
    • Characterization of piroxicam crystal modifications
    • Vrecer F, Vrbinc M, Meden A. (2003). Characterization of piroxicam crystal modifications. Int J Pharm, 256:3-15.
    • (2003) Int J Pharm , vol.256 , pp. 3-15
    • Vrecer, F.1    Vrbinc, M.2    Meden, A.3
  • 39
    • 33745585586 scopus 로고    scopus 로고
    • Preparation of roxithromycin-polymeric microparticles by the emulsion solvent diffusion method for taste masking
    • Gao Y, Cui F, Guan Y, Yang L, Wang Y, Zhang L. (2006). Preparation of roxithromycin-polymeric microparticles by the emulsion solvent diffusion method for taste masking. Int J Pharm, 318:62-69
    • (2006) Int J Pharm , vol.318 , pp. 62-69
    • Gao, Y.1    Cui, F.2    Guan, Y.3    Yang, L.4    Wang, Y.5    Zhang, L.6
  • 40
    • 0030601850 scopus 로고    scopus 로고
    • Properties of solid dispersions of piroxicam in polyvi-nylpyrrolidone K-30
    • Tantishaiyakul V, Kaewnopparat N, Ingkatawornwong S. (1996). Properties of solid dispersions of piroxicam in polyvi-nylpyrrolidone K-30. Int J Pharm, 143:59-66.
    • (1996) Int J Pharm , vol.143 , pp. 59-66
    • Tantishaiyakul, V.1    Kaewnopparat, N.2    Ingkatawornwong, S.3
  • 41
    • 0035800245 scopus 로고    scopus 로고
    • A comparison of alternative polymer excipients and processing methods for making solid dispersions of a poorly water-soluble drug
    • Broman E, Khoo C, Taylor LS. (2001). A comparison of alternative polymer excipients and processing methods for making solid dispersions of a poorly water-soluble drug. Int J Pharm, 222:139-151
    • (2001) Int J Pharm , vol.222 , pp. 139-151
    • Broman, E.1    Khoo, C.2    Taylor, L.S.3
  • 42
    • 0025864425 scopus 로고
    • Preformula-tion studies on solid dispersions containing triamterene or temazepam in polyethylene glycols or Gelucire 44/14 for liquid filling of hard gelatin capsules
    • Dordunoo SK, Ford JL, Rubinstein MH. (1991). Preformula-tion studies on solid dispersions containing triamterene or temazepam in polyethylene glycols or Gelucire 44/14 for liquid filling of hard gelatin capsules. Drug Dev Ind Pharm, 17:1685-1713
    • (1991) Drug Dev Ind Pharm , vol.17 , pp. 1685-1713
    • Dordunoo, S.K.1    Ford, J.L.2    Rubinstein, M.H.3
  • 43
    • 0036281847 scopus 로고    scopus 로고
    • Characterization of carmazepinegelucire 50/13 microparticles prepared by a spray-congealing process using ultrasounds
    • Passerini N, Perissutti B, Moneghini M, Voinovich D, Albertini B, Cavallari C, et al. (2002). Characterization of carmazepinegelucire 50/13 microparticles prepared by a spray-congealing process using ultrasounds. J Pharm Sci, 91:699-707.
    • (2002) J Pharm Sci , vol.91 , pp. 699-707
    • Passerini, N.1    Perissutti, B.2    Moneghini, M.3    Voinovich, D.4    Albertini, B.5    Cavallari, C.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.