SCOPUS 정보 검색 플랫폼

Volumn 5, Issue 7, 2010, Pages 1102-1109

Synthesis and evaluation of bis-thiazolium salts as potential antimalarial drugs

(7) Caldarelli, Sergio A a Duckert, Jean Frédéric a Wein, Sharon a Calas, Michèle a Périgaud, Christian a Vial, Henri a Peyrottes, Suzanne a

a UNIV MONTPELLIER (France)

Author keywords

Bioorganic chemistry; Choline analogues; Malaria; Microwave chemistry; Structure activity relationships

Indexed keywords

3,3' [4,4' (1,4 PHENYLENE)BIS(BUTANE 4,1 DIYL)]BIS[5 (2 METHOXYETHYL) 4 METHYLTHIAZOL 3 IUM]; 5 (2 HYDROXYETHYL) 3 [4 [4 [4 [5 (2 HYDROXYETHYL)THIAZ OL 3 IUM 3 YL]BUTYL]PHENYL]BUTYL] 4 METHYLTHIAZOL 3 IUM; ANTIMALARIAL AGENT; AROMATIC COMPOUND; POLYCYCLIC AROMATIC HYDROCARBON DERIVATIVE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG; 3,3'-(4,4'-(1,4-PHENYLENE)BIS(BUTANE-4,1-DIYL))BIS(5-(2-METHOXYETHYL)-4-METHYLTHIAZOL-3-IUM); 5-(2-HYDROXYETHYL)-3-(4-(4-(4-(5-(2-HYDROXYETHYL)THIAZ-OL-3-IUM-3-YL)BUTYL)PHENYL)BUTYL)-4-METHYLTHIAZOL-3-IUM;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMALARIAL ACTIVITY; ARTICLE; CHEMICAL BOND; CONCENTRATION RESPONSE; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; MALARIA; MOUSE; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; ANIMAL; CHEMISTRY; DRUG EFFECTS; SYNTHESIS;

ANIMALS; ANTIMALARIALS; MICE; PLASMODIUM FALCIPARUM; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 77954114198 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000097 Document Type: Article

Times cited : (8)

References (21)

1
- 57649122948
- World Health Organization, Geneva (Switzerland) (accessed May 12, 2010)
- World Malaria Report 2008, World Health Organization, Geneva (Switzerland) 2008, http://www.who.int/malaria/wmr2008/ (accessed May 12, 2010).
- (2008) World Malaria Report 2008

2
- 41849125318
- B. M. Greenwood, D. A. Fidock, D. E. Kyle, S. H. I. Kappe, P. L. Alonso, F. H. Collins, P. E. Duffy, J. Clin. Invest. 2008, 118, 1266-1276.
- (2008) J. Clin. Invest. , vol.118 , pp. 1266-1276
- Greenwood, B.M.¹ Fidock, D.A.² Kyle, D.E.³ Kappe, S.H.I.⁴ Alonso, P.L.⁵ Collins, F.H.⁶ Duffy, P.E.⁷

3
- 48749090404
- Geneva (Switzerland) (accessed May 12, 2010)
- Roll Back Malaria, The Global Malaria Action Plan for a Malaria-Free World, Geneva (Switzerland) 2008, http://www.rollbackmalaria.org/gmap/index.html (accessed May 12, 2010).
- (2008) Roll Back Malaria, The Global Malaria Action Plan for a Malaria-Free World

4
- 68049123592
- A. M. Dondorp, F. Nosten, P. Yi, D. Das, A. P. Phyo, J. Tarning, K. M. Lwin, F. Ariey, W. Hanpithakpong, S. J. Lee, P. Ringwald, K. Silamut, M. Imwong, K. Chotivanich, P. Lim, T. Herdman, S. S. An, S. Yeung, P. Singhasivanon, N. P. J. Day, N. Lindegardh, D. Socheat, N. J. White, New Engl. J. Med. 2009, 361, 455-467.
- (2009) New Engl. J. Med. , vol.361 , pp. 455-467
- Dondorp, A.M.¹ Nosten, F.² Yi, P.³ Das, D.⁴ Phyo, A.P.⁵ Tarning, J.⁶ Lwin, K.M.⁷ Ariey, F.⁸ Hanpithakpong, W.⁹ Lee, S.J.¹⁰ Ringwald, P.¹¹ Silamut, K.¹² Imwong, M.¹³ Chotivanich, K.¹⁴ Lim, P.¹⁵ Herdman, T.¹⁶ An, S.S.¹⁷ Yeung, S.¹⁸ Singhasivanon, P.¹⁹ Day, N.P.J.²⁰ more..

5
- 0032519825
- M. L. Ancelin, M. Calas, J. Bompart, G. Cordina, D. Martin, M. Ben Bari, T. Jei, P. Druilhe, H. J. Vial, Blood 1998, 91, 1426-1437.
- (1998) Blood , vol.91 , pp. 1426-1437
- Ancelin, M.L.¹ Calas, M.² Bompart, J.³ Cordina, G.⁴ Martin, D.⁵ Ben Bari, M.⁶ Jei, T.⁷ Druilhe, P.⁸ Vial, H.J.⁹

6
- 0034628578
- M. Calas, M. L. Ancelin, G. Cordina, P. Portefaix, G. Piquet, V. Vidal-Sailhan, H. Vial, J. Med. Chem. 2000, 43, 505-516.
- (2000) J. Med. Chem. , vol.43 , pp. 505-516
- Calas, M.¹ Ancelin, M.L.² Cordina, G.³ Portefaix, P.⁴ Piquet, G.⁵ Vidal-Sailhan, V.⁶ Vial, H.⁷

7
- 20844453564
- A. Hamze, E. Rubi, P. Arnal, M. Boisbrun, C. Carcel, X. Salom-Roig, M. Maynadier, S. Wein, H. Vial, M. Calas, J. Med. Chem. 2005, 48, 3639-3643.
- (2005) J. Med. Chem. , vol.48 , pp. 3639-3643
- Hamze, A.¹ Rubi, E.² Arnal, P.³ Boisbrun, M.⁴ Carcel, C.⁵ Salom-Roig, X.⁶ Maynadier, M.⁷ Wein, S.⁸ Vial, H.⁹ Calas, M.¹⁰

8
- 0017691206
- G. G. Holz, Bull. World Health Organ. 1977, 55, 237-248.
- (1977) Bull. World Health Organ. , vol.55 , pp. 237-248
- Holz, G.G.¹

9
- 33646074865
- (Ed.: I. W. Sherman), ASM Press, Washington DC
- H. Vial, C. Mamoun in Molecular Approaches to Malaria (Ed.: I. W. Sherman), ASM Press, Washington DC, 2005, pp. 327-352.
- (2005) Molecular Approaches to Malaria , pp. 327-352
- Vial, H.¹ Mamoun, C.²

10
- 0037325017
- H. J. Vial, P. Eldin, A. G. M. Tielens, J. J. Van Hellemond, Mol. Biochem. Parasitol. 2003, 126, 143-154.
- (2003) Mol. Biochem. Parasitol. , vol.126 , pp. 143-154
- Vial, H.J.¹ Eldin, P.² Tielens, A.G.M.³ Van Hellemond, J.J.⁴

11
- 0003766888
- (Ed. P. J. Rosenthal), Humana Press, Totowa, NJ
- H. J. Vial, M. Calas in Antimalarial Chemotherapy: Mechanisms of Action, Resistance, and New Directions in Drug Discovery (Ed. P. J. Rosenthal), Humana Press, Totowa, NJ, 2001, pp. 347-365.
- (2001) Antimalarial Chemotherapy: Mechanisms of Action, Resistance, and New Directions in Drug Discovery , pp. 347-365
- Vial, H.J.¹ Calas, M.²

12
- 0030725087
- M. Calas, G. Cordina, J. Bompart, M. Ben Bari, T. Jei, M. L. Ancelin, H. Vial, J. Med. Chem. 1997, 40, 3557-3566.
- (1997) J. Med. Chem. , vol.40 , pp. 3557-3566
- Calas, M.¹ Cordina, G.² Bompart, J.³ Ben Bari, M.⁴ Jei, T.⁵ Ancelin, M.L.⁶ Vial, H.⁷

13
- 0043095590
- M. L. Ancelin, M. Calas, V. Vidal-Sailhan, S. Herbute, P. Ringwald, H. J. Vial, Antimicrob. Agents Chemother. 2003, 47, 2590-2597.
- (2003) Antimicrob. Agents Chemother. , vol.47 , pp. 2590-2597
- Ancelin, M.L.¹ Calas, M.² Vidal-Sailhan, V.³ Herbute, S.⁴ Ringwald, P.⁵ Vial, H.J.⁶

14
- 0042594674
- M. L. Ancelin, M. Calas, A. Bonhoure, S. Herbute, H. J. Vial, Antimicrob. Agents Chemother. 2003, 47, 2598-2605.
- (2003) Antimicrob. Agents Chemother. , vol.47 , pp. 2598-2605
- Ancelin, M.L.¹ Calas, M.² Bonhoure, A.³ Herbute, S.⁴ Vial, H.J.⁵

15
- 0037083529
- K. Wengelnik, V. Vidal, M. L. Ancelin, A. M. Cathiard, J. L. Morgat, C. H. Kocken, M. Calas, S. Herrera, A. W. Thomas, H. J. Vial, Science 2002, 295, 1311-1314.
- (2002) Science , vol.295 , pp. 1311-1314
- Wengelnik, K.¹ Vidal, V.² Ancelin, M.L.³ Cathiard, A.M.⁴ Morgat, J.L.⁵ Kocken, C.H.⁶ Calas, M.⁷ Herrera, S.⁸ Thomas, A.W.⁹ Vial, H.J.¹⁰

16
- 7444260721
- H. J. Vial, S. Wein, C. Farenc, C. Kocken, O. Nicolas, M. L. Ancelin, F. Bressolle, A. Thomas, M. Calas, Proc. Natl. Acad. Sci. USA 2004, 101, 15458-15463.
- (2004) Proc. Natl. Acad. Sci. USA , vol.101 , pp. 15458-15463
- Vial, H.J.¹ Wein, S.² Farenc, C.³ Kocken, C.⁴ Nicolas, O.⁵ Ancelin, M.L.⁶ Bressolle, F.⁷ Thomas, A.⁸ Calas, M.⁹

17
- 24144440791
- O. Nicolas, D. Margout, N. Taudon, S. Wein, M. Calas, H. J. Vial, F. M. M. Bressolle, Antimicrob. Agents Chemother. 2005, 49, 3631-3639.
- (2005) Antimicrob. Agents Chemother. , vol.49 , pp. 3631-3639
- Nicolas, O.¹ Margout, D.² Taudon, N.³ Wein, S.⁴ Calas, M.⁵ Vial, H.J.⁶ Bressolle, F.M.M.⁷

18
- 0035289779
- C. A. Lipinski, F. Lombardo, B. W. Dominy, P. J. Feeney, Adv. Drug Delivery Rev. 2001, 46, 3-26.
- (2001) Adv. Drug Delivery Rev. , vol.46 , pp. 3-26
- Lipinski, C.A.¹ Lombardo, F.² Dominy, B.W.³ Feeney, P.J.⁴

19
- 0001334658
- M. A. Navia, P. R. Chaturvedi, Drug Discovery Today 1996, 1, 179-189.
- (1996) Drug Discovery Today , vol.1 , pp. 179-189
- Navia, M.A.¹ Chaturvedi, P.R.²

20
- 0037030653
- D. F. Veber, S. R. Johnson, H. Y. Cheng, B. R. Smith, K. W. Ward, K. D. Kopple, J. Med. Chem. 2002, 45, 2615-2623.
- (2002) J. Med. Chem. , vol.45 , pp. 2615-2623
- Veber, D.F.¹ Johnson, S.R.² Cheng, H.Y.³ Smith, B.R.⁴ Ward, K.W.⁵ Kopple, K.D.⁶

21
- 3242656139
- J. S. Choi, C. W. Kang, K. Jung, J. W. Yang, Y. G. Kim, H. Y. Han, J. Am. Chem. Soc. 2004, 126, 8606-8607.
- (2004) J. Am. Chem. Soc. , vol.126 , pp. 8606-8607
- Choi, J.S.¹ Kang, C.W.² Jung, K.³ Yang, J.W.⁴ Kim, Y.G.⁵ Han, H.Y.⁶

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