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Volumn 40, Issue 22, 1997, Pages 3557-3566

Antimalarial activity of molecules interfering with Plasmodium falciparum phospholipid metabolism. Structure-activity relationship analysis

Author keywords

[No Author keywords available]

Indexed keywords

ANTIMALARIAL AGENT; CHOLINE DERIVATIVE; ETHANOLAMINE DERIVATIVE; QUATERNARY AMMONIUM DERIVATIVE; TERTIARY AMINE;

EID: 0030725087     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm9701886     Document Type: Article
Times cited : (103)

References (18)
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    • Regulation of phosphatidylcholine biosynthesis in Plasmodium-infected erythrocytes
    • Ancelin M. L.; Vial, H. J. Regulation of phosphatidylcholine biosynthesis in Plasmodium-infected erythrocytes Biochim. Biophys. Acta 1989, 1001, 82-89.
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    • Ancelin, M.L.1    Vial, H.J.2
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    • Quaternary ammonium compounds efficiently inhibit Plasmodium falciparum growth in vitro by impairment of choline transport
    • Ancelin, M. L.; Vial, H. J. Quaternary ammonium compounds efficiently inhibit Plasmodium falciparum growth in vitro by impairment of choline transport. Antimicrob. Agents Chemother. 1986, 29, 814-820.
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  • 6
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    • Vial, H. J.; Thuet, M. J.; Ancelin, M. L.; Philippot, J. R.; Chavis, C. Phosphohpid metabolism as a new target for malaria chemotherapy. Mechanism of action of D-2-amino-1-butanol Bio. chem. Pharmacol. 1984, 33, 2761-2770.
    • (1984) Bio. Chem. Pharmacol. , vol.33 , pp. 2761-2770
    • Vial, H.J.1    Thuet, M.J.2    Ancelin, M.L.3    Philippot, J.R.4    Chavis, C.5
  • 12
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    • Inhibitors of choline transport into Plasmodium-infected erythrocytes are effective antiplasmodial compounds in vitro
    • Ancelin, M. L.; Vial, H. J.; Philippot, J. R. Inhibitors of choline transport into Plasmodium-infected erythrocytes are effective antiplasmodial compounds in vitro. Biochem. Pharmacol 1985 34, 4068-4071.
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    • Correlation of the efficiency of fatty derivatives in suppressing Plasmodium falciparum growth in culture with their inhibitory effect on acyl-CoA synthetase activity
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    • Beaumelle, B.D.1    Vial, H.J.2
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    • Structure-activity studies on inhibition of choline uptake by a mouse brain synaptosomal preparation: Basic data
    • Tamaru, M.; Roberts, E. Structure-activity studies on inhibition of choline uptake by a mouse brain synaptosomal preparation: basic data. Brain Res. 1988, 473, 205-226.
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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.