Identification and inhibitory properties of a novel Ca2+/ calmodulin antagonist

Biochemistry

Volumn 49, Issue 19, 2010, Pages 4244-4254

  Colomer, Josep ^a   Schmitt, Allison A ^a   Toone, Eric J ^a   Means, Anthony R ^a  

^a DUKE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CHEMICAL INHIBITORS; HIGH-THROUGHPUT; IN-VITRO; ISOTHERMAL TITRATION CALORIMETRY; LIVING CELL; MITOGENS; TRIFLUOPERAZINE;

ASSAYS; BINDING ENERGY; BINDING SITES; BIOCHEMISTRY; CALCIUM; CALMODULIN; CALORIMETRY; LIBRARIES; STOICHIOMETRY; TITRATION;

CAMS;

125 C9; CALCIUM ION; CALMODULIN INHIBITOR; N (4 AMINOBUTYL) 5 CHLORO 2 NAPSYLAMIDE; PROTON; TRIFLUOPERAZINE; UNCLASSIFIED DRUG;

ACIDITY; ARTICLE; BINDING SITE; CELL PROLIFERATION; CELL STRAIN HEK293; CONTROLLED STUDY; HIGH THROUGHPUT SCREENING; HUMAN; HUMAN CELL; HYPOTHESIS; IN VITRO STUDY; ISOTHERMAL TITRATION CALORIMETRY; MOLECULE; NONHUMAN; PRIORITY JOURNAL; STOICHIOMETRY; YEAST;

BINDING SITES; CALMODULIN; HYDROGEN-ION CONCENTRATION; SUBSTRATE SPECIFICITY; SULFONAMIDES; TRIFLUOPERAZINE;

EID: 77952356292     PISSN: 00062960     EISSN: 15204995     Source Type: Journal    
DOI: 10.1021/bi1001213     Document Type: Article

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