BFPP, a phloroglucinol derivative, induces cell apoptosis in human chondrosarcoma cells through endoplasmic reticulum stress

Biochemical Pharmacology

Volumn 79, Issue 10, 2010, Pages 1410-1417

  Liu, Ju Fang ^a   Yang, Wei Hung ^a,b   Fong, Yi Chin ^a,c   Kuo, Sheng Chu ^a   Chang, Chih Shiang ^a   Tang, Chih Hsin ^a  

^a CHINA MEDICAL UNIVERSITY   (Taiwan)

^b CHINA MEDICAL UNIVERSITY BEIGANG HOSPITAL   (Taiwan)

^c CHINA MEDICAL UNIVERSITY HOSPITAL   (Taiwan)

Author keywords

BFPP; Calpain; Chondrosarcoma; ER; GRP78

Indexed keywords

1 NAPHTHYL; 2 CHLOROPHENYL; 2 FLUOROPHENYL; 2,4 BIS(2 FLUOROPHENYLACETYL)PHLOROGLUCINOL; 3 CHLOROPHENYL; 3 FLUOROPHENYL; 3,4 DICHLOROPHENYL; 3,4 DIMETHOXYPHENYL; 3,4 METHYLENEDIOXY; 4 CHLOROPHENYL; 4 FLUOROPHENYL; 4 METHOXYPHENYL; 4 METHYLPHENYL; 4 NOTIROPHENYL; ANTINEOPLASTIC AGENT; CALCIUM; CALPAIN; GLUCOSE REGULATED PROTEIN 78; PHENYL; PHLOROGLUCINOL DERIVATIVE; SMALL INTERFERING RNA; THIOPHENYL; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTINEOPLASTIC ACTIVITY; APOPTOSIS; ARTICLE; CANCER SIZE; CARTILAGE CELL; CHONDROSARCOMA; CONTROLLED STUDY; CYTOSOL; DRUG EFFECT; DRUG MECHANISM; ENDOPLASMIC RETICULUM STRESS; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; SARCOMA CELL;

ANIMALS; ANTINEOPLASTIC AGENTS; APOPTOSIS; BLOTTING, WESTERN; BONE NEOPLASMS; CALPAIN; CASPASES; CELL LINE; CELL LINE, TUMOR; CHONDROCYTES; CHONDROSARCOMA; ENDOPLASMIC RETICULUM; FLOW CYTOMETRY; GENE EXPRESSION REGULATION, NEOPLASTIC; HEAT-SHOCK PROTEINS; HUMANS; MALE; MEMBRANE GLYCOPROTEINS; MICE; MICE, INBRED BALB C; PHLOROGLUCINOL; POLYMERASE CHAIN REACTION;

EID: 77649185144     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2010.01.002     Document Type: Article

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