Characterization of non-lipid autotaxin inhibitors

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 2, 2010, Pages 769-776

  Hoeglund, Adrienne B ^a,b   Howard, Angela L ^a,b   Wanjala, Irene W ^a,b   Pham, Truc Chi T ^a   Parrill, Abby L ^a,b   Baker, Daniel L ^a  

^a University of Memphis   (United States)

^b UNIVERSITY OF MEMPHIS   (United States)

Author keywords

ATX; Autotaxin; FS 3; Nucleotide pyrophosphatase phosphodiesterase; para Nitrophenyl thymidine 5 monophosphate

Indexed keywords

4 NITROPHENYL THYMIDINE 5' MONOPHOSPHATE; AUTOTAXIN; CYTOKINE RECEPTOR ANTAGONIST; FS 3; H2L 5210574; H2L 5564949; H2L 5761473; H2L 7839888; H2L 7905958; H2L 7921385; LYSOPHOSPHATIDYLCHOLINE; LYSOPHOSPHOLIPASE; LYSOPHOSPHOLIPASE D; LYSOPHOSPHOLIPID; NUCLEOTIDE DERIVATIVE; NUCLEOTIDE PYROPHOSPHATASE; PHOSPHODIESTERASE; UNCLASSIFIED DRUG;

ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; EMBRYO; FLUORESCENCE; HUMAN; HUMAN CELL; HYDROLYSIS; IC 50;

DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; HUMANS; KINETICS; MOLECULAR WEIGHT; MULTIENZYME COMPLEXES; PHOSPHODIESTERASE I; PYROPHOSPHATASES; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; STEREOISOMERISM;

EID: 76449086955     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2009.11.056     Document Type: Article

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