메뉴 건너뛰기




Volumn 40, Issue 2, 2010, Pages 83-92

High concentrations of commonly used drugs can inhibit the in vitro glucuronidation of bisphenol A and nonylphenol in rats

Author keywords

Bisphenol A; Drugs; Hepatocytes; Interactions; Metabolism; Microsomes; P nonylphenol; Rat

Indexed keywords

4,4' ISOPROPYLIDENEDIPHENOL; AMOXICILLIN; CARBAMAZEPINE; CIMETIDINE; DICLOFENAC; ERYTHROMYCIN; GLICLAZIDE; IBUPROFEN; MEFENAMIC ACID; NAPROXEN; NONYLPHENOL; PARACETAMOL; RANITIDINE; SALAZOSULFAPYRIDINE; SALICYLIC ACID; VALPROIC ACID;

EID: 75649110847     PISSN: 00498254     EISSN: 13665928     Source Type: Journal    
DOI: 10.3109/00498250903383334     Document Type: Article
Times cited : (20)

References (45)
  • 1
    • 0021267790 scopus 로고
    • Comparative pharmacokinetics of sulphasalazine and sulphapyridine after rectal and oral administration to patients with ulcerative colitis
    • Allgayer H, Kruis W, Eisenburg J, Paumgartner G. (1984). Comparative pharmacokinetics of sulphasalazine and sulphapyridine after rectal and oral administration to patients with ulcerative colitis. Eur J Clin Pharmacol 26(2):275-277
    • (1984) Eur J Clin Pharmacol , vol.26 , Issue.2 , pp. 275-277
    • Allgayer, H.1    Kruis, W.2    Eisenburg, J.3    Paumgartner, G.4
  • 2
    • 33747881994 scopus 로고    scopus 로고
    • Estrogen-like response to p-nonylphenol in human first trimester placenta and BeWo choriocarcinoma cells
    • Bechi N, Ietta F, Romagnoli R, Focardi S, Corsi I, Buffi C, Paulesu L. (2006). Estrogen-like response to p-nonylphenol in human first trimester placenta and BeWo choriocarcinoma cells. Toxicol Sci 93(1):75-81.
    • (2006) Toxicol Sci , vol.93 , Issue.1 , pp. 75-81
    • Bechi, N.1    Ietta, F.2    Romagnoli, R.3    Focardi, S.4    Corsi, I.5    Buffi, C.6    Paulesu, L.7
  • 3
    • 0015325312 scopus 로고
    • Amoxicillin: In vitro and pharmacological studies
    • Bodey GP, Nance J. (1972). Amoxicillin: in vitro and pharmacological studies. Antimicrob Agents Chemother 1(4):358-362
    • (1972) Antimicrob Agents Chemother , vol.1 , Issue.4 , pp. 358-362
    • Bodey, G.P.1    Nance, J.2
  • 4
    • 0019996083 scopus 로고
    • Bioavailability of acetylsalicylic acid and salicylic acid from rapid- and slow-release formulations, and in combination with dipyridamol
    • Brantmark B, Wahlin-Boll E, Melander A. (1982). Bioavailability of acetylsalicylic acid and salicylic acid from rapid- and slow-release formulations, and in combination with dipyridamol. Eur J Clin Pharmacol 22(4):309-314
    • (1982) Eur J Clin Pharmacol , vol.22 , Issue.4 , pp. 309-314
    • Brantmark, B.1    Wahlin-Boll, E.2    Melander, A.3
  • 7
    • 0041525234 scopus 로고    scopus 로고
    • Glucuronidation and excretion of nonylphenol in perfused rat liver
    • Daidoji T, Inoue H, Kato S, Yokota H. (2003). Glucuronidation and excretion of nonylphenol in perfused rat liver. Drug Metab Dispos 31(8):993-998
    • (2003) Drug Metab Dispos , vol.31 , Issue.8 , pp. 993-998
    • Daidoji, T.1    Inoue, H.2    Kato, S.3    Yokota, H.4
  • 8
    • 0034020162 scopus 로고    scopus 로고
    • Pharmacokinetics and pharmacodynamics of gliclazide in Caucasians and Australian Aborigines with type 2 diabetes
    • Davis TM, Daly F, Walsh JP, Ilett KF, Beilby JP, Dusci LJ, Barrett PH. (2000). Pharmacokinetics and pharmacodynamics of gliclazide in Caucasians and Australian Aborigines with type 2 diabetes. Br J Clin Pharmacol 49(3):223-230
    • (2000) Br J Clin Pharmacol , vol.49 , Issue.3 , pp. 223-230
    • Davis, T.M.1    Daly, F.2    Walsh, J.P.3    Ilett, K.F.4    Beilby, J.P.5    Dusci, L.J.6    Barrett, P.H.7
  • 9
    • 0034605688 scopus 로고    scopus 로고
    • Bioavailability of ibuprofen from matrix mini-tablets based on a mixture of starch and microcrystalline wax
    • De Brabander C, Vervaet C, Gortz JP, Remon JP, Berlo JA. (2000). Bioavailability of ibuprofen from matrix mini-tablets based on a mixture of starch and microcrystalline wax. Int J Pharm 208(1-2):81-86
    • (2000) Int J Pharm , vol.208 , Issue.1-2 , pp. 81-86
    • De Brabander, C.1    Vervaet, C.2    Gortz, J.P.3    Remon, J.P.4    Berlo, J.A.5
  • 10
    • 0035087551 scopus 로고    scopus 로고
    • Comparison of the modulatory effects of human and rat liver microsomal metabolism on the estrogenicity of bisphenol A: Implications for extrapolation to humans
    • Elsby R, Maggs JL, Ashby J, Park BK. (2001). Comparison of the modulatory effects of human and rat liver microsomal metabolism on the estrogenicity of bisphenol A: implications for extrapolation to humans. J Pharmacol Exp Ther 297(1):103-113
    • (2001) J Pharmacol Exp Ther , vol.297 , Issue.1 , pp. 103-113
    • Elsby, R.1    Maggs, J.L.2    Ashby, J.3    Park, B.K.4
  • 11
    • 0038741909 scopus 로고    scopus 로고
    • The effect of valproic acid on drug and steroid glucuronidation by expressed human UDP-glucuronosyltransferases
    • Ethell BT, Anderson GD, Burchell B. (2003). The effect of valproic acid on drug and steroid glucuronidation by expressed human UDP- glucuronosyltransferases. Biochem Pharmacol 65(9): 1441-1449
    • (2003) Biochem Pharmacol , vol.65 , Issue.9 , pp. 1441-1449
    • Ethell, B.T.1    Anderson, G.D.2    Burchell, B.3
  • 15
    • 55649123233 scopus 로고    scopus 로고
    • Human UDPglucuronosyltransferase isoforms involved in bisphenol A glucuronidation
    • Hanioka N, Naito T, Narimatsu S. (2008). Human UDPglucuronosyltransferase isoforms involved in bisphenol A glucuronidation. Chemosphere 74(1):33-36
    • (2008) Chemosphere , vol.74 , Issue.1 , pp. 33-36
    • Hanioka, N.1    Naito, T.2    Narimatsu, S.3
  • 16
    • 0021998435 scopus 로고
    • Acetaminophen decreases adenosine 3″-phosphate 5″- phosphosulfate and uridine diphosphoglucuronic acid in rat liver
    • Hjelle JJ, Hazelton GA, Klaassen CD. (1985). Acetaminophen decreases adenosine 3″-phosphate 5″-phosphosulfate and uridine diphosphoglucuronic acid in rat liver. Drug Metab Dispos 13(1):35-41.
    • (1985) Drug Metab Dispos , vol.13 , Issue.1 , pp. 35-41
    • Hjelle, J.J.1    Hazelton, G.A.2    Klaassen, C.D.3
  • 17
    • 0022459940 scopus 로고
    • Depletion of hepatic UDP-glucuronic acid by drugs that are glucuronidated
    • Howell SR, Hazelton GA, Klaassen CD. (1986). Depletion of hepatic UDP-glucuronic acid by drugs that are glucuronidated. J Pharmacol Exp Ther 236(3):610-614
    • (1986) J Pharmacol Exp Ther , vol.236 , Issue.3 , pp. 610-614
    • Howell, S.R.1    Hazelton, G.A.2    Klaassen, C.D.3
  • 18
    • 0028340580 scopus 로고
    • Pharmacokinetics of valproate after multiple-dose oral and intravenous infusion administration: Gastrointestinal-related diurnal variation
    • Hussein Z, Mukherjee D, Lamm J, Cavanaugh JH, Granneman GR. (1994). Pharmacokinetics of valproate after multiple-dose oral and intravenous infusion administration: gastrointestinal-related diurnal variation. J Clin Pharmacol 34(7):754-759
    • (1994) J Clin Pharmacol , vol.34 , Issue.7 , pp. 754-759
    • Hussein, Z.1    Mukherjee, D.2    Lamm, J.3    Cavanaugh, J.H.4    Granneman, G.R.5
  • 19
    • 0036851180 scopus 로고    scopus 로고
    • Determination of bisphenol A concentrations in human biological fluids reveals significant early prenatal exposure
    • Ikezuki Y, Tsutsumi O, Takai Y, Kamei Y, Taketani Y. (2002). Determination of bisphenol A concentrations in human biological fluids reveals significant early prenatal exposure. Hum Reprod 17(11):2839-2841
    • (2002) Hum Reprod , vol.17 , Issue.11 , pp. 2839-2841
    • Ikezuki, Y.1    Tsutsumi, O.2    Takai, Y.3    Kamei, Y.4    Taketani, Y.5
  • 20
    • 0037671242 scopus 로고    scopus 로고
    • Bisphenol A glucuronidation and absorption in rat intestine
    • Inoue H, Yuki G, Yokota H, Kato S. (2003). Bisphenol A glucuronidation and absorption in rat intestine. Drug Metab Dispos 31(1):140-144
    • (2003) Drug Metab Dispos , vol.31 , Issue.1 , pp. 140-144
    • Inoue, H.1    Yuki, G.2    Yokota, H.3    Kato, S.4
  • 21
    • 0035116968 scopus 로고    scopus 로고
    • Migration of 4-nonylphenol from polyvinyl chloride food packaging films into food simulants and foods
    • Inoue K, Kondo S, Yoshie Y, Kato K, Yoshimura Y, Horie M, Nakazawa H. (2001). Migration of 4-nonylphenol from polyvinyl chloride food packaging films into food simulants and foods. Food Addit Contam 18(2):157-164
    • (2001) Food Addit Contam , vol.18 , Issue.2 , pp. 157-164
    • Inoue, K.1    Kondo, S.2    Yoshie, Y.3    Kato, K.4    Yoshimura, Y.5    Horie, M.6    Nakazawa, H.7
  • 23
    • 15244342411 scopus 로고    scopus 로고
    • UDP-glucuronosyltransferases and clinical drug-drug interactions
    • Kiang TK, Ensom MH, Chang TK. (2005). UDP-glucuronosyltransferases and clinical drug-drug interactions. Pharmacol Ther 106(1):97-132.
    • (2005) Pharmacol Ther , vol.106 , Issue.1 , pp. 97-132
    • Kiang, T.K.1    Ensom, M.H.2    Chang, T.K.3
  • 24
    • 0035038561 scopus 로고    scopus 로고
    • Characterization of rat and human UDP-glucuronosyltransferases responsible for the in vitro glucuronidation of diclofenac
    • King C, Tang W, Ngui J, Tephly T, Braun M. (2001). Characterization of rat and human UDP-glucuronosyltransferases responsible for the in vitro glucuronidation of diclofenac. Toxicol Sci 61(1):49-53.
    • (2001) Toxicol Sci , vol.61 , Issue.1 , pp. 49-53
    • King, C.1    Tang, W.2    Ngui, J.3    Tephly, T.4    Braun, M.5
  • 25
    • 0346784817 scopus 로고    scopus 로고
    • Pharmacokinetics of diclofenac and inhibition of cyclooxygenases 1 and 2: No relationship to the CYP2C9 genetic polymorphism in humans
    • Kirchheiner J, Meineke I, Steinbach N, Meisel C, Roots I, Brockmoller J. (2003). Pharmacokinetics of diclofenac and inhibition of cyclooxygenases 1 and 2: no relationship to the CYP2C9 genetic polymorphism in humans. Br J Clin Pharmacol 55(1):51-61.
    • (2003) Br J Clin Pharmacol , vol.55 , Issue.1 , pp. 51-61
    • Kirchheiner, J.1    Meineke, I.2    Steinbach, N.3    Meisel, C.4    Roots, I.5    Brockmoller, J.6
  • 26
    • 0035417251 scopus 로고    scopus 로고
    • Determination of endocrine-disrupting phenolic compounds and estrogens in surface and drinking water by HRGC-(NCI)-MS in the picogram per liter range
    • Kuch HM, Ballschmiter K. (2001). Determination of endocrine-disrupting phenolic compounds and estrogens in surface and drinking water by HRGC-(NCI)-MS in the picogram per liter range. Environ Sci Technol 35(15):3201-3206
    • (2001) Environ Sci Technol , vol.35 , Issue.15 , pp. 3201-3206
    • Kuch, H.M.1    Ballschmiter, K.2
  • 27
    • 34748895120 scopus 로고    scopus 로고
    • Prediction of metabolic clearance of bisphenol A (4,4″-dihydroxy-2, 2-diphenylpropane) using cryopreserved human hepatocytes
    • Kuester RK, Sipes IG. (2007). Prediction of metabolic clearance of bisphenol A (4,4″-dihydroxy-2,2-diphenylpropane) using cryopreserved human hepatocytes. Drug Metab Dispos 35(10):1910-1915
    • (2007) Drug Metab Dispos , vol.35 , Issue.10 , pp. 1910-1915
    • Kuester, R.K.1    Sipes, I.G.2
  • 28
    • 0034069492 scopus 로고    scopus 로고
    • Estrogenic activity of octylphenol, nonylphenol, bisphenol A and methoxychlor in rats
    • Laws SC, Carey SA, Ferrell JM, Bodman GJ, Cooper RL. (2000). Estrogenic activity of octylphenol, nonylphenol, bisphenol A and methoxychlor in rats. Toxicol Sci 54(1):154-167
    • (2000) Toxicol Sci , vol.54 , Issue.1 , pp. 154-167
    • Laws, S.C.1    Carey, S.A.2    Ferrell, J.M.3    Bodman, G.J.4    Cooper, R.L.5
  • 30
    • 33846430542 scopus 로고    scopus 로고
    • Inhibitory potential of nonsteroidal anti-inflammatory drugs on UDPglucuronosyltransferase 2B7 in human liver microsomes
    • Mano Y, Usui T, Kamimura H. (2007). Inhibitory potential of nonsteroidal anti-inflammatory drugs on UDPglucuronosyltransferase 2B7 in human liver microsomes. Eur J Clin Pharmacol 63(2):211-216
    • (2007) Eur J Clin Pharmacol , vol.63 , Issue.2 , pp. 211-216
    • Mano, Y.1    Usui, T.2    Kamimura, H.3
  • 31
    • 0035102123 scopus 로고    scopus 로고
    • Vitro and in vivo interactions of bisphenol A and its metabolite, bisphenol A glucuronide, with estrogen receptors alpha and beta
    • Matthews JB, Twomey K, Zacharewski TR. (2001). In vitro and in vivo interactions of bisphenol A and its metabolite, bisphenol A glucuronide, with estrogen receptors alpha and beta. Chem Res Toxicol 14(2):149-157
    • (2001) Chem Res Toxicol , vol.14 , Issue.2 , pp. 149-157
    • Matthews, J.B.1    Twomey, K.2    Zacharewski, T.R.3
  • 32
    • 0027408461 scopus 로고
    • Bioavailability of controlled release carbamazepine estimated by mixed effect modelling
    • Miller R, Ludden TM. (1993). Bioavailability of controlled release carbamazepine estimated by mixed effect modelling. Eur J Clin Pharmacol 44(3):231-235
    • (1993) Eur J Clin Pharmacol , vol.44 , Issue.3 , pp. 231-235
    • Miller, R.1    Ludden, T.M.2
  • 33
    • 0034748451 scopus 로고    scopus 로고
    • Glucuronidation of nonylphenol and octylphenol eliminates their ability to activate transcription via the estrogen receptor
    • Moffat GJ, Burns A, Van Miller J, Joiner R, Ashby J. (2001). Glucuronidation of nonylphenol and octylphenol eliminates their ability to activate transcription via the estrogen receptor. Regul Toxicol Pharmacol 34(2):182-187
    • (2001) Regul Toxicol Pharmacol , vol.34 , Issue.2 , pp. 182-187
    • Moffat, G.J.1    Burns, A.2    Van Miller, J.3    Joiner, R.4    Ashby, J.5
  • 34
    • 0022640959 scopus 로고
    • Pharmacokinetics and bioavailability of ranitidine in normal subjects and cirrhotic patients
    • Morichau-Beauchant M, Houin G, Mavier P, Alexandre C, Dhumeaux D. (1986). Pharmacokinetics and bioavailability of ranitidine in normal subjects and cirrhotic patients. Dig Dis Sci 31(2):113-118
    • (1986) Dig Dis Sci , vol.31 , Issue.2 , pp. 113-118
    • Morichau-Beauchant, M.1    Houin, G.2    Mavier, P.3    Alexandre, C.4    Dhumeaux, D.5
  • 35
    • 0024270214 scopus 로고
    • Absorption of naproxen controlled-release tablets in fasting and postprandial volunteers
    • Mroszczak E, Yee JP, Bynum L. (1988). Absorption of naproxen controlled-release tablets in fasting and postprandial volunteers. J Clin Pharmacol 28(12):1128-1131
    • (1988) J Clin Pharmacol , vol.28 , Issue.12 , pp. 1128-1131
    • Mroszczak, E.1    Yee, J.P.2    Bynum, L.3
  • 36
    • 0023737762 scopus 로고
    • Effect of magnesium hydroxide on the absorption of tolfenamic and mefenamic acids
    • Neuvonen PJ, Kivisto KT. (1988). Effect of magnesium hydroxide on the absorption of tolfenamic and mefenamic acids. Eur J Clin Pharmacol 35(5):495-501.
    • (1988) Eur J Clin Pharmacol , vol.35 , Issue.5 , pp. 495-501
    • Neuvonen, P.J.1    Kivisto, K.T.2
  • 37
    • 0347285474 scopus 로고    scopus 로고
    • Determination of bisphenol A and 4-nonylphenol in human milk using alkaline digestion and cleanup by solid-phase extraction
    • Otaka H, Yasuhara A, Morita M. (2003). Determination of bisphenol A and 4-nonylphenol in human milk using alkaline digestion and cleanup by solid-phase extraction. Anal Sci 19(12):1663-1666
    • (2003) Anal Sci , vol.19 , Issue.12 , pp. 1663-1666
    • Otaka, H.1    Yasuhara, A.2    Morita, M.3
  • 38
    • 0025179702 scopus 로고
    • Comparative metabolism of high doses of aspirin in man and rat
    • Patel DK, Notarianni LJ, Bennett PN. (1990). Comparative metabolism of high doses of aspirin in man and rat. Xenobiotica 20(8):847-854
    • (1990) Xenobiotica , vol.20 , Issue.8 , pp. 847-854
    • Patel, D.K.1    Notarianni, L.J.2    Bennett, P.N.3
  • 39
    • 0028044817 scopus 로고
    • A recombinant phenobarbital-inducible rat liver UDPglucuronosyltransferase (UDP-glucuronosyltransferase 2B1) stably expressed in V79 cells catalyzes the glucuronidation of morphine, phenols, and carboxylic acids
    • Pritchard M, Fournel-Gigleux S, Siest G, Mackenzie P, Magdalou J. (1994). A recombinant phenobarbital-inducible rat liver UDPglucuronosyltransferase (UDP-glucuronosyltransferase 2B1) stably expressed in V79 cells catalyzes the glucuronidation of morphine, phenols, and carboxylic acids. Mol Pharmacol 45(1):42-50.
    • (1994) Mol Pharmacol , vol.45 , Issue.1 , pp. 42-50
    • Pritchard, M.1    Fournel-Gigleux, S.2    Siest, G.3    MacKenzie, P.4    Magdalou, J.5
  • 40
    • 0017363410 scopus 로고
    • Pharmacokinetics of paracetamol (acetaminophen) after intravenous and oral administration
    • Rawlins MD, Henderson DB, Hijab AR. (1977). Pharmacokinetics of paracetamol (acetaminophen) after intravenous and oral administration. Eur J Clin Pharmacol 11(4):283-286
    • (1977) Eur J Clin Pharmacol , vol.11 , Issue.4 , pp. 283-286
    • Rawlins, M.D.1    Henderson, D.B.2    Hijab, A.R.3
  • 41
    • 20744460349 scopus 로고    scopus 로고
    • Evaluation of oral and intravenous route pharmacokinetics, plasma protein binding, and uterine tissue dose metrics of bisphenol A: A physiologically based pharmacokinetic approach
    • Teeguarden JG, Waechter JM, Jr., Clewell HJ, 3rd, Covington TR, Barton HA. (2005). Evaluation of oral and intravenous route pharmacokinetics, plasma protein binding, and uterine tissue dose metrics of bisphenol A: a physiologically based pharmacokinetic approach. Toxicol Sci 85(2):823-838
    • (2005) Toxicol Sci , vol.85 , Issue.2 , pp. 823-838
    • Teeguarden, J.G.1    Waechter Jr., J.M.2    Clewell III, H.J.3    Covington, T.R.4    Barton, H.A.5
  • 42
    • 0019301958 scopus 로고
    • Influence of food on absorption of erythromycin ethyl succinate
    • Thompson PJ, Burgess KR, Marlin GE. (1980). Influence of food on absorption of erythromycin ethyl succinate. Antimicrob Agents Chemother 18(5):829-831
    • (1980) Antimicrob Agents Chemother , vol.18 , Issue.5 , pp. 829-831
    • Thompson, P.J.1    Burgess, K.R.2    Marlin, G.E.3
  • 43
    • 1842536833 scopus 로고    scopus 로고
    • Human UDPglucuronosyltransferases: Isoform selectivity and kinetics of 4-methylumbelliferone and 1-naphthol glucuronidation, effects of organic solvents, and inhibition by diclofenac and probenecid
    • Uchaipichat V, Mackenzie PI, Guo XH, Gardner-Stephen D, Galetin A, Houston JB, Miners JO. (2004). Human UDPglucuronosyltransferases: isoform selectivity and kinetics of 4-methylumbelliferone and 1-naphthol glucuronidation, effects of organic solvents, and inhibition by diclofenac and probenecid. Drug Metab Dispos 32(4):413-423
    • (2004) Drug Metab Dispos , vol.32 , Issue.4 , pp. 413-423
    • Uchaipichat, V.1    MacKenzie, P.I.2    Guo, X.H.3    Gardner-Stephen, D.4    Galetin, A.5    Houston, J.B.6    Miners, J.O.7
  • 45
    • 0033152656 scopus 로고    scopus 로고
    • Glucuronidation of the environmental oestrogen bisphenol A by an isoform of UDPglucuronosyltransferase, UGT2B1, in the rat liver
    • Yokota H, Iwano H, Endo M, Kobayashi T, Inoue H, Ikushiro S, Yuasa A. (1999). Glucuronidation of the environmental oestrogen bisphenol A by an isoform of UDPglucuronosyltransferase, UGT2B1, in the rat liver. Biochem J 340(Pt 2):405-409
    • (1999) Biochem J , vol.340 , Issue.PART 2 , pp. 405-409
    • Yokota, H.1    Iwano, H.2    Endo, M.3    Kobayashi, T.4    Inoue, H.5    Ikushiro, S.6    Yuasa, A.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.