Targeted tumor diagnosis and therapy with peptide hormones as radiopharmaceuticals
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Preclinical evaluation of the a-particle generator nuclide 225Ac for somatostatin receptor radiotherapy of neuroendocrine tumors
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Treatment with the radiolabeled somatostatin analog [177Lu-DOTA0, Tyr3]octreotate: Toxicity, efficacy, and survival
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Preparation and biological evaluation of 64Cu-CB-TE2A-sst2-ANT, a somatostatin antagonist for PET imaging of somatostatin receptor-positive tumors
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Design and in vitro characterization of highly sst2-selective somatostatin antagonists suitable for radiotargeting
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Mammalian bombesin receptors: Nomenclature, distribution, pharmacology, signaling, and functions in normal and disease states
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In vitro binding evaluation of 177Lu AMBA, a novel 177Lu-labeled GRP-R agonist for systemic radiotherapy in human tissues
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In vitro and in vivo analysis of [64Cu-NO2A-8-Aoc-BBN(7-14)NH2]: A site-directed radiopharmaceutical for positron-emission tomography imaging of T-47D human breast cancer tumors
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177Lu-AMBA: Synthesis and characterization of a selective 177Lu-labeled GRP-R agonist for systemic radiotherapy of prostate cancer
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203Pb-labeled a-melanocyte-stimulating hormone peptide as an imaging probe for melanoma detection
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Development of high-specificactivity 68Ga-labeled DOTA-rhenium-cyclized a-MSH peptide analog to target MC1 receptors overexpressed by melanoma tumors
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Metastatic melanoma imaging with an 111In-labeled lactam bridge-cyclized a-melanocyte-stimulating hormone peptide
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A 99mTc(CO)3-labeled pyrazolyl-amelanocyte-stimulating hormone analog conjugate for melanoma targeting
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Glycosylated DOTA-a-melanocyte-stimulating hormone analogues for melanoma targeting: Influence of the site of glycosylation on in vivo biodistribution
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Improving tumor uptake and pharmacokinetics of 64Cu-labeled cyclic RGD peptide dimers with Gly3 and PEG4 linkers
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Dual integrin and gastrin-releasing peptide receptor targeted tumor imaging using 18F-labeled PEGylated RGD-bombesin heterodimer 18F-FB-PEG3-Glu-RGD-BBN
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68Ga-labeled cyclic RGD dimers with Gly3 and PEG4 linkers: Promising agents for tumor integrin avb3 PET imaging
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