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Volumn 17, Issue 1, 2010, Pages 69-76

Radiolabeled regulatory peptides for imaging and therapy

Author keywords

Molecular imaging; Peptides; Regulatory; Therapy

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID AC 225; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID DEXTRO PHENYLALANINE TYROSINE 3 OCTREOTIDE AC 225; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID DEXTRO PHENYLALANINE TYROSINE 3 OCTREOTIDE LU 177; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID DEXTRO PHENYLALANINE TYROSINE 3 OCTREOTIDE Y 90; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID LU 177; BISMUTH 212; BISMUTH 213; COPPER 64; GALLIUM; GALLIUM 66; GALLIUM 67; GALLIUM 68; LUTETIUM 177; OCTREOTIDE; OCTREOTIDE[DEXTRO PHENYLALANYLCYSTEINYLPHENYLANINE DEXTRO TRYPTOPHYLLYSYLTHREONYLCYSTEINYLTHREONINE OL]; PEPTIDE; PEPTIDE RECEPTOR; RADIOISOTOPE; RADIOLABELED REGULATORY PEPTIDE; RADIOPHARMACEUTICAL AGENT; RHENIUM 186; RHENIUM 188; SOMATOSTATIN DERIVATIVE; TECHNETIUM 99M; TYROSINE 3 OCTREOTATE[DEXTRO PHENYLALANYLCYSTEINYLTYROSINE DEXTRO TRYPTOPHYLLYSYLTHREONYLCYSTEINYLTHREONINE]; TYROSINE 3 OCTREOTIDE[DEXTRO PHENYLALANYLCYSTEINYLTYROSINE DEXTRO TRYPTOPHYLLYSYLTHREONYLCYSTEINYLTHREONINE OL]; UNCLASSIFIED DRUG; UNINDEXED DRUG; YTTRIUM 86; YTTRIUM 90;

EID: 75149157017     PISSN: 1752296X     EISSN: None     Source Type: Journal    
DOI: 10.1097/MED.0b013e32833392ac     Document Type: Review
Times cited : (22)

References (29)
  • 1
    • 67651111779 scopus 로고    scopus 로고
    • Tumor imaging and therapy using radiolabeled somatostatin analogues
    • Jong MD, Breeman WAP, Kwekkeboom DJ, et al. Tumor imaging and therapy using radiolabeled somatostatin analogues. Acc Chem Res 2009; 42:873-880.
    • (2009) Acc Chem Res , vol.42 , pp. 873-880
    • Jong, M.D.1    Breeman, W.A.P.2    Kwekkeboom, D.J.3
  • 2
    • 57349195981 scopus 로고    scopus 로고
    • Peptide-based probes for cancer imaging
    • Reubi JC, Maecke HR. Peptide-based probes for cancer imaging. J Nucl Med 2008; 49:1735-1738.
    • (2008) J Nucl Med , vol.49 , pp. 1735-1738
    • Reubi, J.C.1    Maecke, H.R.2
  • 3
    • 41649083838 scopus 로고    scopus 로고
    • Targeted tumor diagnosis and therapy with peptide hormones as radiopharmaceuticals
    • Khan IU, Beck-Sickinger AG. Targeted tumor diagnosis and therapy with peptide hormones as radiopharmaceuticals. Anticancer Agents Med Chem 2008; 8:186-199.
    • (2008) Anticancer Agents Med Chem , vol.8 , pp. 186-199
    • Khan, I.U.1    Beck-Sickinger, A.G.2
  • 4
    • 50349089716 scopus 로고    scopus 로고
    • Preclinical evaluation of the a-particle generator nuclide 225Ac for somatostatin receptor radiotherapy of neuroendocrine tumors
    • Miederer M, Henriksen G, Alke A, et al. Preclinical evaluation of the a-particle generator nuclide 225Ac for somatostatin receptor radiotherapy of neuroendocrine tumors. Clin Cancer Res 2008; 14:3555-3561.
    • (2008) Clin Cancer Res , vol.14 , pp. 3555-3561
    • Miederer, M.1    Henriksen, G.2    Alke, A.3
  • 5
    • 43749091955 scopus 로고    scopus 로고
    • Treatment with the radiolabeled somatostatin analog [177Lu-DOTA0, Tyr3]octreotate: Toxicity, efficacy, and survival
    • Kwekkeboom DJ, de Herder WW, Kam BL, et al. Treatment with the radiolabeled somatostatin analog [177Lu-DOTA0, Tyr3]octreotate: toxicity, efficacy, and survival. J Clin Oncol 2008; 26:2124-2130.
    • (2008) J Clin Oncol , vol.26 , pp. 2124-2130
    • Kwekkeboom, D.J.1    De Herder, W.W.2    Kam, B.L.3
  • 6
    • 65349111443 scopus 로고    scopus 로고
    • Outcome of treating advanced neuroendocrine tumors with radiolabeled somatostatin analogues
    • Muros MA, Varsavsky M, Rozas PI, et al. Outcome of treating advanced neuroendocrine tumors with radiolabeled somatostatin analogues. Clin Transl Oncol 2009; 11:48-53.
    • (2009) Clin Transl Oncol , vol.11 , pp. 48-53
    • Muros, M.A.1    Varsavsky, M.2    Rozas, P.I.3
  • 7
    • 57349185212 scopus 로고    scopus 로고
    • Preparation and biological evaluation of 64Cu-CB-TE2A-sst2-ANT, a somatostatin antagonist for PET imaging of somatostatin receptor-positive tumors
    • Wadas TJ, Eiblmaier M, Zheleznyak A, et al. Preparation and biological evaluation of 64Cu-CB-TE2A-sst2-ANT, a somatostatin antagonist for PET imaging of somatostatin receptor-positive tumors. J Nucl Med 2008; 49:1819-1827.
    • (2008) J Nucl Med , vol.49 , pp. 1819-1827
    • Wadas, T.J.1    Eiblmaier, M.2    Zheleznyak, A.3
  • 8
    • 46849089935 scopus 로고    scopus 로고
    • Design and in vitro characterization of highly sst2-selective somatostatin antagonists suitable for radiotargeting
    • Cescato R, Erchegyi J, Waser B, et al. Design and in vitro characterization of highly sst2-selective somatostatin antagonists suitable for radiotargeting. J Med Chem 2008; 51:4030-4037.
    • (2008) J Med Chem , vol.51 , pp. 4030-4037
    • Cescato, R.1    Erchegyi, J.2    Waser, B.3
  • 9
    • 38949198118 scopus 로고    scopus 로고
    • Bombesin receptor antagonists may be preferable to agonists for tumor targeting
    • Cescato R, Maina T, Nock B, et al. Bombesin receptor antagonists may be preferable to agonists for tumor targeting. J Nucl Med 2008; 49:318-326.
    • (2008) J Nucl Med , vol.49 , pp. 318-326
    • Cescato, R.1    Maina, T.2    Nock, B.3
  • 10
    • 41149176081 scopus 로고    scopus 로고
    • Mammalian bombesin receptors: Nomenclature, distribution, pharmacology, signaling, and functions in normal and disease states
    • Jensen RT, Battey JF, Spindel ER, et al. Mammalian bombesin receptors: nomenclature, distribution, pharmacology, signaling, and functions in normal and disease states. Pharmacol Rev 2008; 60:1-42.
    • (2008) Pharmacol Rev , vol.60 , pp. 1-42
    • Jensen, R.T.1    Battey, J.F.2    Spindel, E.R.3
  • 11
    • 60449087638 scopus 로고    scopus 로고
    • In vitro binding evaluation of 177Lu AMBA, a novel 177Lu-labeled GRP-R agonist for systemic radiotherapy in human tissues
    • Thomas R, Chen J, Roudier MM, et al. In vitro binding evaluation of 177Lu AMBA, a novel 177Lu-labeled GRP-R agonist for systemic radiotherapy in human tissues. Clin Exp Metastasis 2009; 26:105-119.
    • (2009) Clin Exp Metastasis , vol.26 , pp. 105-119
    • Thomas, R.1    Chen, J.2    Roudier, M.M.3
  • 12
    • 67651151216 scopus 로고    scopus 로고
    • True radiotracers: Cu-64 targeting vectors based upon bombesin peptide
    • Hoffman TJ, Smith CJ. True radiotracers: Cu-64 targeting vectors based upon bombesin peptide. Nucl Med Biol 2009; 36:579-585.
    • (2009) Nucl Med Biol , vol.36 , pp. 579-585
    • Hoffman, T.J.1    Smith, C.J.2
  • 13
    • 59649105956 scopus 로고    scopus 로고
    • In vitro and in vivo analysis of [64Cu-NO2A-8-Aoc-BBN(7-14)NH2]: A site-directed radiopharmaceutical for positron-emission tomography imaging of T-47D human breast cancer tumors
    • Prasanphanich AF, Retzloff L, Lane SR, et al. In vitro and in vivo analysis of [64Cu-NO2A-8-Aoc-BBN(7-14)NH2]: a site-directed radiopharmaceutical for positron-emission tomography imaging of T-47D human breast cancer tumors. Nucl Med Biol 2009; 36:171-181.
    • (2009) Nucl Med Biol , vol.36 , pp. 171-181
    • Prasanphanich, A.F.1    Retzloff, L.2    Lane, S.R.3
  • 14
    • 33747105269 scopus 로고    scopus 로고
    • 177Lu-AMBA: Synthesis and characterization of a selective 177Lu-labeled GRP-R agonist for systemic radiotherapy of prostate cancer
    • Lantry LE, Cappelletti E, Maddalena ME, et al. 177Lu-AMBA: synthesis and characterization of a selective 177Lu-labeled GRP-R agonist for systemic radiotherapy of prostate cancer. J Nucl Med 2006; 47:1144-1152.
    • (2006) J Nucl Med , vol.47 , pp. 1144-1152
    • Lantry, L.E.1    Cappelletti, E.2    Maddalena, M.E.3
  • 15
    • 56649115222 scopus 로고    scopus 로고
    • Novel glycated [99mTc(CO) 3]-labeled bombesin analogues for improved targeting of gastrin-releasing peptide receptor-positive tumors
    • Schweinsberg C, Maes V, Brans L, et al. Novel glycated [99mTc(CO)3]-labeled bombesin analogues for improved targeting of gastrin-releasing peptide receptor-positive tumors. Bioconjugate Chem 2008; 19:2432-2439.
    • (2008) Bioconjugate Chem , vol.19 , pp. 2432-2439
    • Schweinsberg, C.1    Maes, V.2    Brans, L.3
  • 16
    • 44149100050 scopus 로고    scopus 로고
    • 203Pb-labeled a-melanocyte-stimulating hormone peptide as an imaging probe for melanoma detection
    • Miao Y, Figueroa SD, Fisher DR, et al. 203Pb-labeled a-melanocyte- stimulating hormone peptide as an imaging probe for melanoma detection. J Nucl Med 2008; 49:823-829.
    • (2008) J Nucl Med , vol.49 , pp. 823-829
    • Miao, Y.1    Figueroa, S.D.2    Fisher, D.R.3
  • 17
    • 67349235942 scopus 로고    scopus 로고
    • Development of high-specificactivity 68Ga-labeled DOTA-rhenium-cyclized a-MSH peptide analog to target MC1 receptors overexpressed by melanoma tumors
    • Cantorias MV, Figueroa SD, Quinn TP, et al. Development of high-specificactivity 68Ga-labeled DOTA-rhenium-cyclized a-MSH peptide analog to target MC1 receptors overexpressed by melanoma tumors. Nucl Med Biol 2009; 36:505-513.
    • (2009) Nucl Med Biol , vol.36 , pp. 505-513
    • Cantorias, M.V.1    Figueroa, S.D.2    Quinn, T.P.3
  • 18
    • 67349128040 scopus 로고    scopus 로고
    • Melanoma imaging using 111In-, 86Y-and 68Ga-labeled CHX-A00-Re(Arg11) CCMSH
    • Wie L, Zhang X, Gallazzi F, et al. Melanoma imaging using 111In-, 86Y-and 68Ga-labeled CHX-A00-Re(Arg11)CCMSH. Nucl Med Biol 2009; 36:345-354.
    • (2009) Nucl Med Biol , vol.36 , pp. 345-354
    • Wie, L.1    Zhang, X.2    Gallazzi, F.3
  • 19
    • 39749136463 scopus 로고    scopus 로고
    • 111In-labeled lactam bridge-cyclized a-melanocyte stimulating hormone peptide analogues for melanoma imaging
    • Miao Y, Gallazzi F, Guo H, Quinn TP. 111In-labeled lactam bridge-cyclized a-melanocyte stimulating hormone peptide analogues for melanoma imaging. Bioconjugate Chem 2008; 19:539-547.
    • (2008) Bioconjugate Chem , vol.19 , pp. 539-547
    • Miao, Y.1    Gallazzi, F.2    Guo, H.3    Quinn, T.P.4
  • 20
    • 62549146618 scopus 로고    scopus 로고
    • Metastatic melanoma imaging with an 111In-labeled lactam bridge-cyclized a-melanocyte-stimulating hormone peptide
    • Guo H, Shenoy N, Gershman BM, et al. Metastatic melanoma imaging with an 111In-labeled lactam bridge-cyclized a-melanocyte-stimulating hormone peptide. Nucl Med Biol 2009; 36:267-276.
    • (2009) Nucl Med Biol , vol.36 , pp. 267-276
    • Guo, H.1    Shenoy, N.2    Gershman, B.M.3
  • 21
    • 40949123297 scopus 로고    scopus 로고
    • Melanoma targeting with amelanocyte stimulating hormone analogs labeled with fac-[99mTc(CO) 3]+: Effect of cyclization on tumor-seeking properties
    • Raposinho PD, Xavier C, Correia JDG, et al. Melanoma targeting with amelanocyte stimulating hormone analogs labeled with fac-[99mTc(CO)3]+: effect of cyclization on tumor-seeking properties. J Biol Inorg Chem 2008; 13:449-459.
    • (2008) J Biol Inorg Chem , vol.13 , pp. 449-459
    • Raposinho, P.D.1    Xavier, C.2    Correia, J.D.G.3
  • 22
    • 37449007128 scopus 로고    scopus 로고
    • A 99mTc(CO)3-labeled pyrazolyl-amelanocyte-stimulating hormone analog conjugate for melanoma targeting
    • Raposinho PD, Correia JDG, Alves S, et al. A 99mTc(CO)3-labeled pyrazolyl-amelanocyte-stimulating hormone analog conjugate for melanoma targeting. Nucl Med Biol 2008; 35:91-99.
    • (2008) Nucl Med Biol , vol.35 , pp. 91-99
    • Raposinho, P.D.1    Correia, J.D.G.2    Alves, S.3
  • 23
    • 66149184413 scopus 로고    scopus 로고
    • Glycosylated DOTA-a-melanocyte-stimulating hormone analogues for melanoma targeting: Influence of the site of glycosylation on in vivo biodistribution
    • Bapst JP, Calame M, Tanner H, Eberle AN. Glycosylated DOTA-a-melanocyte-stimulating hormone analogues for melanoma targeting: influence of the site of glycosylation on in vivo biodistribution. Bioconjugate Chem 2009; 20:984-993.
    • (2009) Bioconjugate Chem , vol.20 , pp. 984-993
    • Bapst, J.P.1    Calame, M.2    Tanner, H.3    Eberle, A.N.4
  • 24
    • 65249138736 scopus 로고    scopus 로고
    • Improving tumor uptake and pharmacokinetics of 64Cu-labeled cyclic RGD peptide dimers with Gly3 and PEG4 linkers
    • Shi J, Kim YS, Zhai S, et al. Improving tumor uptake and pharmacokinetics of 64Cu-labeled cyclic RGD peptide dimers with Gly3 and PEG4 linkers. Bioconjugate Chem 2009; 20:750-759.
    • (2009) Bioconjugate Chem , vol.20 , pp. 750-759
    • Shi, J.1    Kim, Y.S.2    Zhai, S.3
  • 25
    • 60549098667 scopus 로고    scopus 로고
    • Dual integrin and gastrin-releasing peptide receptor targeted tumor imaging using 18F-labeled PEGylated RGD-bombesin heterodimer 18F-FB-PEG3-Glu-RGD-BBN
    • Liu Z, Yan Y, Chin FT, et al. Dual integrin and gastrin-releasing peptide receptor targeted tumor imaging using 18F-labeled PEGylated RGD-bombesin heterodimer 18F-FB-PEG3-Glu-RGD-BBN. J Med Chem 2009; 52:425-432.
    • (2009) J Med Chem , vol.52 , pp. 425-432
    • Liu, Z.1    Yan, Y.2    Chin, F.T.3
  • 26
    • 68949212307 scopus 로고    scopus 로고
    • 68Ga-labeled NOTA-RGD-BBN peptide for dual integrin and GRPR-targeted tumor imaging
    • Liu Z, Niu G, Wang F, Chen X. 68Ga-labeled NOTA-RGD-BBN peptide for dual integrin and GRPR-targeted tumor imaging. Eur J Nucl Med Mol Imaging 2009; 36:1483-1494.
    • (2009) Eur J Nucl Med Mol Imaging , vol.36 , pp. 1483-1494
    • Liu, Z.1    Niu, G.2    Wang, F.3    Chen, X.4
  • 27
    • 67349145987 scopus 로고    scopus 로고
    • 68Ga-labeled cyclic RGD dimers with Gly3 and PEG4 linkers: Promising agents for tumor integrin avb3 PET imaging
    • Liu Z, Niu G, Shi J, et al. 68Ga-labeled cyclic RGD dimers with Gly3 and PEG4 linkers: promising agents for tumor integrin avb3 PET imaging. Eur J Nucl Med Mol Imaging 2009; 36:947-957.
    • (2009) Eur J Nucl Med Mol Imaging , vol.36 , pp. 947-957
    • Liu, Z.1    Niu, G.2    Shi, J.3
  • 28
    • 67650093751 scopus 로고    scopus 로고
    • Small-animal PET of tumors with 64Cu-labeled RGDbombesin heterodimer
    • Liu Z, Li ZB, CaoQ, et al. Small-animal PET of tumors with 64Cu-labeled RGDbombesin heterodimer. J Nucl Med 2009; 50:1168-1177.
    • (2009) J Nucl Med , vol.50 , pp. 1168-1177
    • Liu, Z.1    Li, Z.B.2    Cao, Q.3
  • 29
    • 70349139674 scopus 로고    scopus 로고
    • Evaluation of a novel Arg-Gly-Asp-conjugated a-melanocyte stimulating hormone hybrid peptide for potential melanoma therapy
    • Yang J, Guo H, Gallazzi F, et al. Evaluation of a novel Arg-Gly-Asp-conjugated a-melanocyte stimulating hormone hybrid peptide for potential melanoma therapy. Bioconjugate Chem 2009; 20:1634-1642.
    • (2009) Bioconjugate Chem , vol.20 , pp. 1634-1642
    • Yang, J.1    Guo, H.2    Gallazzi, F.3


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