In vitro binding evaluation of 177Lu-AMBA, a novel 177Lu-labeled GRP-R agonist for systemic radiotherapy in human tissues

Clinical and Experimental Metastasis

Volumn 26, Issue 2, 2009, Pages 105-119

  Thomas, Regi ^a   Chen, Jianqing ^a   Roudier, Martine M ^b,c,d   Vessella, Robert L ^b,e   Lantry, Laura E ^a   Nunn, Adrian D ^a  

^a Bracco Research USA   (United States)

^b UNIVERSITY OF WASHINGTON SCHOOL OF MEDICINE   (United States)

^c UNIVERSITY OF WASHINGTON   (United States)

^d AMGEN INC   (United States)

^e VA Puget Sound   (United States)

Author keywords

177Lu AMBA; Bombesin; Gastrin releasing peptide receptor; Hormone refractory prostate cancer; Metastasis

Indexed keywords

BOMBESIN; GASTRIN RELEASING PEPTIDE; GASTRIN RELEASING PEPTIDE RECEPTOR; IODINE 125; LUTETIUM 177; PEPTIDE; RADIOLIGAND; RECEPTOR SUBTYPE;

ANIMAL CELL; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BREAST CANCER; DRUG BINDING SITE; DRUG RECEPTOR BINDING; DRUG TARGETING; HUMAN; HUMAN CELL; HUMAN TISSUE; IN VITRO STUDY; METASTASIS; NONHUMAN; PROSTATE CANCER;

ADULT; AGED; AGED, 80 AND OVER; AUTORADIOGRAPHY; BINDING SITES; BINDING, COMPETITIVE; BOMBESIN; BREAST NEOPLASMS; FEMALE; HUMANS; MALE; MIDDLE AGED; NEOPLASM METASTASIS; OLIGOPEPTIDES; ORGAN SPECIFICITY; PROSTATIC NEOPLASMS; RADIOPHARMACEUTICALS; RECEPTORS, BOMBESIN; YOUNG ADULT;

EID: 60449087638     PISSN: 02620898     EISSN: 15737276     Source Type: Journal    
DOI: 10.1007/s10585-008-9220-0     Document Type: Article

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