The fifth transmembrane domain of angiotensin II type 1 receptor participates in the formation of the ligand-binding pocket and undergoes a counterclockwise rotation upon receptor activation

Journal of Biological Chemistry

Volumn 284, Issue 46, 2009, Pages 31953-31961

  Domazet, Ivana ^a   Martin, Stéphane S ^a   Holleran, Brian J ^a   Morin, Marie Ève ^a   Lacasse, Patrick ^a   Lavigne, Pierre ^a   Escher, Emanuel ^a   Leduc, Richard ^a   Guillemette, Gaétan ^a  

^a UNIVERSITY OF SHERBROOKE   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

ACTIVATION ANALYSIS; AMMONIUM COMPOUNDS; BINDING ENERGY; CHEMICAL ACTIVATION; LIGANDS; OPTICAL RESONATORS; PROTEINS;

CONSTITUTIVELY ACTIVES; COUNTER CLOCKWISE ROTATION; COVALENT MODIFICATIONS; FREE SULFHYDRYL GROUPS; G PROTEIN COUPLED RECEPTORS; METHANETHIOSULFONATE-ETHYLAMMONIUM; RECEPTOR ACTIVATION; TRANS-MEMBRANE DOMAINS;

AMINO ACIDS;

ANGIOTENSIN 1 RECEPTOR; CYSTEINE; LYSINE; THIOMESYLIC ACID METHYL ESTER; THREONINE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; COVALENT BOND; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN DOMAIN; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN MODIFICATION; RECEPTOR BINDING;

EID: 70450225265     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M109.051839     Document Type: Article

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