SCOPUS 정보 검색 플랫폼

Volumn 4, Issue 9, 2009, Pages 1469-1479

Docking studies of structurally diverse antimalarial drugs targeting PfATP6: No correlation between in silico binding affinity and in vitro antimalarial activity

(5) Garah, Fatima Bousejra El a Stigliani, Jean Luc a Coslédan, Frédéric b Meunier, Bernard b Robert, Anne a

a LCC LABORATOIRE DE CHIMIE DE COORDINATION (France)

b Zone Industrielle de Vic de Graves (France)

Author keywords

Antimalarial agents; Artemisinin; Enzymes; Inhibitors; Molecular modeling

Indexed keywords

ADAMANTANE; ANTIMALARIAL AGENT; ARTEMISININ; ARTEMISININ DERIVATIVE; CHLOROQUINE; CYCLOPIAZONIC ACID; DOCKING PROTEIN; LIGAND; MEFLOQUINE; OUABAIN; PEROXIDE; PLASMODIUM FALCIPARUM SARCOPLASMIC RETICULUM CALCIUM TRANSPORTING ADENOSINE TRIPHOSPHATASE; QUININE; QUINOLINE; SARCOPLASMIC RETICULUM CALCIUM TRANSPORTING ADENOSINE TRIPHOSPHATASE; SARCOPLASMIC RETICULUM CALCIUM TRANSPORTING ADENOSINE TRIPHOSPHATASE 1A; SILICON; THAPSIGARGIN; UNCLASSIFIED DRUG;

ALKYLATION; ANTIMALARIAL ACTIVITY; ARTEMISIA ANNUA; ARTICLE; BINDING AFFINITY; CONFORMATION; CONFORMATIONAL TRANSITION; CRYSTAL STRUCTURE; DRUG TARGETING; IN VITRO STUDY; MODEL; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; PROTEIN STRUCTURE; RABBIT; VALIDATION PROCESS;

ANIMALS; ANTIMALARIALS; ARTEMISININS; CALCIUM-TRANSPORTING ATPASES; COMPUTER SIMULATION; ENZYME INHIBITORS; PLASMODIUM FALCIPARUM; PROTEIN BINDING; QUINOLINES; SESQUITERPENES;

EID: 69749102711 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200900200 Document Type: Article

Times cited : (38)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.