-
6
-
-
0033576619
-
-
Hoekstra W.J., Maryanoff B.E., Damiano B.P., Andrade-Gordon P., Cohen J.H., Costanzo M.J., Haertlein B.J., Hecker L.R., Hulshizer B.L., Kauffman J.A., Keane P., McComsey D.F., Mitchell J.A., Scott L., Shah R.D., and Yabut S.C. J. Med. Chem. 42 (1999) 5254
-
(1999)
J. Med. Chem.
, vol.42
, pp. 5254
-
-
Hoekstra, W.J.1
Maryanoff, B.E.2
Damiano, B.P.3
Andrade-Gordon, P.4
Cohen, J.H.5
Costanzo, M.J.6
Haertlein, B.J.7
Hecker, L.R.8
Hulshizer, B.L.9
Kauffman, J.A.10
Keane, P.11
McComsey, D.F.12
Mitchell, J.A.13
Scott, L.14
Shah, R.D.15
Yabut, S.C.16
-
7
-
-
0035829179
-
-
Lawson E.C., Hoekstra W.J., Addo M.F., Andrade-Gordon P., Damiano B.P., Kauffman J.A., Mitchell J.A., and Maryanoff B.E. Bioorg. Med. Chem. Lett. 11 (2001) 2619
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.11
, pp. 2619
-
-
Lawson, E.C.1
Hoekstra, W.J.2
Addo, M.F.3
Andrade-Gordon, P.4
Damiano, B.P.5
Kauffman, J.A.6
Mitchell, J.A.7
Maryanoff, B.E.8
-
8
-
-
0035887114
-
-
Damiano B.P., Mitchell J.A., Giardino E., Corcoran T., Haertlein B.J., de Garavilla L., Kauffman J.A., Hoekstra W.J., Maryanoff B.E., and Andrade-Gordon P. Thromb. Res. 104 (2001) 113
-
(2001)
Thromb. Res.
, vol.104
, pp. 113
-
-
Damiano, B.P.1
Mitchell, J.A.2
Giardino, E.3
Corcoran, T.4
Haertlein, B.J.5
de Garavilla, L.6
Kauffman, J.A.7
Hoekstra, W.J.8
Maryanoff, B.E.9
Andrade-Gordon, P.10
-
9
-
-
3042826704
-
-
Hanson J., de Leval X., David J.-L., Supuran C., Pirotte B., and Dogné J.-M. Curr. Med. Chem. Cardiovasc. Hematol. Agents 2 (2004) 157
-
(2004)
Curr. Med. Chem. Cardiovasc. Hematol. Agents
, vol.2
, pp. 157
-
-
Hanson, J.1
de Leval, X.2
David, J.-L.3
Supuran, C.4
Pirotte, B.5
Dogné, J.-M.6
-
10
-
-
18244390513
-
-
Meissner R.S., Perkins J.J., Duong L.T., Hartman G.D., Hoffman W.F., Huff J.R., Ihle N.C., Leu C.-T., Nagy R.M., Naylor-Olsen A., Rodan G.A., Rodan S.B., Whitman D.B., Wesolowski G.A., and Duggan M.E. Bioorg. Med. Chem. Lett. 12 (2002) 25
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 25
-
-
Meissner, R.S.1
Perkins, J.J.2
Duong, L.T.3
Hartman, G.D.4
Hoffman, W.F.5
Huff, J.R.6
Ihle, N.C.7
Leu, C.-T.8
Nagy, R.M.9
Naylor-Olsen, A.10
Rodan, G.A.11
Rodan, S.B.12
Whitman, D.B.13
Wesolowski, G.A.14
Duggan, M.E.15
-
11
-
-
33845619375
-
-
Yan S., Larson G., Wu J.Z., Appleby T., Ding Y., Hamatake R., Hong Z., and Yao N. Bioorg. Med. Chem. Lett. 17 (2007) 63
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 63
-
-
Yan, S.1
Larson, G.2
Wu, J.Z.3
Appleby, T.4
Ding, Y.5
Hamatake, R.6
Hong, Z.7
Yao, N.8
-
12
-
-
18244374489
-
-
Lin L.S., Kopka I.E., Mumford R.A., Magriotis P.A., Lanza Jr. T., Durette P.L., Kamenecka T., Young D.N., de Laszlo S.E., McCauley E., Van Riper G., Kidambi U., Egger L.A., Tong X., Lyons K., Vincent S., Stearns R., Colletti A., Teffera Y., Fenyk-Melody J., Schmidt J.A., MacCoss M., and Hagmanna W.K. Bioorg. Med. Chem. Lett. 12 (2002) 611
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 611
-
-
Lin, L.S.1
Kopka, I.E.2
Mumford, R.A.3
Magriotis, P.A.4
Lanza Jr., T.5
Durette, P.L.6
Kamenecka, T.7
Young, D.N.8
de Laszlo, S.E.9
McCauley, E.10
Van Riper, G.11
Kidambi, U.12
Egger, L.A.13
Tong, X.14
Lyons, K.15
Vincent, S.16
Stearns, R.17
Colletti, A.18
Teffera, Y.19
Fenyk-Melody, J.20
Schmidt, J.A.21
MacCoss, M.22
Hagmanna, W.K.23
more..
-
13
-
-
0029984196
-
-
Georg G.I., Harriman G.C.B., Hepperle M., Clowers J.S., and Vander Velde D.G. J. Org. Chem. 61 (1996) 2664
-
(1996)
J. Org. Chem.
, vol.61
, pp. 2664
-
-
Georg, G.I.1
Harriman, G.C.B.2
Hepperle, M.3
Clowers, J.S.4
Vander Velde, D.G.5
-
17
-
-
0033615796
-
-
Zhong H.M., Cohen J.H., Abdel-Magid A.F., Kenney B.D., Maryanoff C.A., Shah R.D., Villani Jr. F.J., Zhang F., and Zhang X. Tetrahedron Lett. 40 (1999) 7721
-
(1999)
Tetrahedron Lett.
, vol.40
, pp. 7721
-
-
Zhong, H.M.1
Cohen, J.H.2
Abdel-Magid, A.F.3
Kenney, B.D.4
Maryanoff, C.A.5
Shah, R.D.6
Villani Jr., F.J.7
Zhang, F.8
Zhang, X.9
-
19
-
-
4043110495
-
-
Hsiao Y., Rivera N.R., Rosner T., Krska S.W., Njolito E., Wang F., Sun Y., Armstrong J.D., Grabowski E.J.J., Tillyer R.D., Spindler F., and Malan C. J. Am. Chem. Soc. 126 (2004) 9918
-
(2004)
J. Am. Chem. Soc.
, vol.126
, pp. 9918
-
-
Hsiao, Y.1
Rivera, N.R.2
Rosner, T.3
Krska, S.W.4
Njolito, E.5
Wang, F.6
Sun, Y.7
Armstrong, J.D.8
Grabowski, E.J.J.9
Tillyer, R.D.10
Spindler, F.11
Malan, C.12
-
20
-
-
69249174321
-
-
PCT Int. Appl. WO 097733
-
Xiao, Y.; Sun, Y.; Rosner, T.; Rivera, N. R.; Krska, S. W.; Clausen, A. M.; Armstrong, J. D.; Spindler, F.; Malan, C. PCT Int. Appl. WO 097733, 2005.
-
(2005)
-
-
Xiao, Y.1
Sun, Y.2
Rosner, T.3
Rivera, N.R.4
Krska, S.W.5
Clausen, A.M.6
Armstrong, J.D.7
Spindler, F.8
Malan, C.9
-
21
-
-
0035586875
-
-
Boesch H., Cesco-Cancian S., Hecker L.R., Hoekstra W.J., Justus M., Maryanoff C.A., Scott L., Shah R.D., Solms G., Sorgi K.L., Stefanick S.M., Thurnheer U., Villani F.J., and Walker D.G. Org. Process Res. Dev. 5 (2001) 23
-
(2001)
Org. Process Res. Dev.
, vol.5
, pp. 23
-
-
Boesch, H.1
Cesco-Cancian, S.2
Hecker, L.R.3
Hoekstra, W.J.4
Justus, M.5
Maryanoff, C.A.6
Scott, L.7
Shah, R.D.8
Solms, G.9
Sorgi, K.L.10
Stefanick, S.M.11
Thurnheer, U.12
Villani, F.J.13
Walker, D.G.14
-
22
-
-
7744233724
-
-
Kuwata S., Yamada T., Shinogi T., Yamagami N., Kitabashi F., Miyazawa T., and Watanabe H. Bull. Chem. Soc. Jpn. 52 (1979) 3326
-
(1979)
Bull. Chem. Soc. Jpn.
, vol.52
, pp. 3326
-
-
Kuwata, S.1
Yamada, T.2
Shinogi, T.3
Yamagami, N.4
Kitabashi, F.5
Miyazawa, T.6
Watanabe, H.7
-
28
-
-
22144479415
-
-
Awasthi A.K., Boys M.L., Cain-Janicki K.J., Colson P.-J., Doubleday W.W., Duran J.E., and Farid P.N. J. Org. Chem. 70 (2005) 5387
-
(2005)
J. Org. Chem.
, vol.70
, pp. 5387
-
-
Awasthi, A.K.1
Boys, M.L.2
Cain-Janicki, K.J.3
Colson, P.-J.4
Doubleday, W.W.5
Duran, J.E.6
Farid, P.N.7
-
30
-
-
0035982154
-
-
Bull S.D., Davies S.G., Fox D.J., Gianotti M., Kelly P.M., Pierres C., Savory E.D., and Smith A.D. J. Chem. Soc., Perkin Trans. 1 (2002) 1858
-
(2002)
J. Chem. Soc., Perkin Trans. 1
, pp. 1858
-
-
Bull, S.D.1
Davies, S.G.2
Fox, D.J.3
Gianotti, M.4
Kelly, P.M.5
Pierres, C.6
Savory, E.D.7
Smith, A.D.8
-
31
-
-
69249184606
-
-
PCT Int. Appl. WO 063682
-
Walther, J.; de Lange, B.; Broxterman, Q. B.; Pöchlauer, P.; van der Sluis, M.; Uiterweerd, P.; Falk, H.; Zuckerstätter, G. PCT Int. Appl. WO 063682, 2005.
-
(2005)
-
-
Walther, J.1
de Lange, B.2
Broxterman, Q.B.3
Pöchlauer, P.4
van der Sluis, M.5
Uiterweerd, P.6
Falk, H.7
Zuckerstätter, G.8
-
33
-
-
0242691679
-
-
Park S., Forró E., Grewal H., Fülöp F., and Kazlauskas R.J. Adv. Synth. Catal. 345 (2003) 986
-
(2003)
Adv. Synth. Catal.
, vol.345
, pp. 986
-
-
Park, S.1
Forró, E.2
Grewal, H.3
Fülöp, F.4
Kazlauskas, R.J.5
-
38
-
-
69249198043
-
-
PCT Int. Appl. WO 080854
-
Gröger, H.; Trauthwein, H.; Drauz, K.; Buchholz, S.; Sacherer, C.; Werner, H. PCT Int. Appl. WO 080854, 2003.
-
(2003)
-
-
Gröger, H.1
Trauthwein, H.2
Drauz, K.3
Buchholz, S.4
Sacherer, C.5
Werner, H.6
-
39
-
-
3843131805
-
-
Gröger H., Trauthwein H., Buchholz S., Drauz K., Sacherer C., Godfrin S., and Werner H. Org. Biomol. Chem. 2 (2004) 1977
-
(2004)
Org. Biomol. Chem.
, vol.2
, pp. 1977
-
-
Gröger, H.1
Trauthwein, H.2
Buchholz, S.3
Drauz, K.4
Sacherer, C.5
Godfrin, S.6
Werner, H.7
-
40
-
-
69249176341
-
-
Eur. Patent 1624052
-
Nakamatsu, T.; Kawasaki, H.; Watanabe, K.; Nakazawa, M.; Izawa, K. Eur. Patent 1624052, 2006.
-
(2006)
-
-
Nakamatsu, T.1
Kawasaki, H.2
Watanabe, K.3
Nakazawa, M.4
Izawa, K.5
-
44
-
-
47149093206
-
-
Lee J.H., Choi B.S., Chang J.H., Lee H.B., Yoon J.-Y., Lee J., and Shin H. J. Org. Chem. 72 (2007) 10261
-
(2007)
J. Org. Chem.
, vol.72
, pp. 10261
-
-
Lee, J.H.1
Choi, B.S.2
Chang, J.H.3
Lee, H.B.4
Yoon, J.-Y.5
Lee, J.6
Shin, H.7
-
47
-
-
33747829030
-
-
Lebedev A.V., Lebedeva A.B., Sheludyakov V.D., Kovaleva E.A., Ustinova O.L., and Kozhevnikov I.B. Russ. J. Gen. Chem. 75 (2005) 1113
-
(2005)
Russ. J. Gen. Chem.
, vol.75
, pp. 1113
-
-
Lebedev, A.V.1
Lebedeva, A.B.2
Sheludyakov, V.D.3
Kovaleva, E.A.4
Ustinova, O.L.5
Kozhevnikov, I.B.6
-
48
-
-
69249179379
-
-
U.S. Patent 5698579
-
Muller, G. W. U.S. Patent 5698579, 1997.
-
(1997)
-
-
Muller, G.W.1
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