Synthesis and antimycobacterial activity of 5-formylaminopyrimidines; analogs of antibacterial purines

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 12, 2009, Pages 3297-3299

  Brændvang, Morten ^a   Charnock, Colin ^b   Gundersen, Lise Lotte ^a  

^a UNIVERSITY OF OSLO   (Norway)

^b OSLO METROPOLITAN UNIVERSITY   (Norway)

Author keywords

Antimycobacterial; Pyrimidine; Ring opening; Tuberculosis

Indexed keywords

5 FORMYLAMINOPYRIMIDINE DERIVATIVE; AMINE; PURINE DERIVATIVE; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; DRUG CYTOTOXICITY; DRUG SCREENING; DRUG SYNTHESIS; ESCHERICHIA COLI; IC 50; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; RING OPENING; STAPHYLOCOCCUS AUREUS;

ANTI-BACTERIAL AGENTS; DOSE-RESPONSE RELATIONSHIP, DRUG; MYCOBACTERIUM TUBERCULOSIS; PURINES; PYRIMIDINES; STRUCTURE-ACTIVITY RELATIONSHIP;

MYCOBACTERIUM TUBERCULOSIS;

EID: 65749085114     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.04.082     Document Type: Article

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