High-throughput synthesis of azide libraries suitable for direct "click" chemistry and in situ screening

Organic and Biomolecular Chemistry

Volumn 7, Issue 9, 2009, Pages 1821-1828

  Srinivasan, Rajavel ^a   Tan, Lay Pheng ^a   Wu, Hao ^a   Yang, Peng Yu ^a   Kalesh, Karunakaran A ^a   Yao, Shao Q ^a  

^a NATIONAL UNIVERSITY OF SINGAPORE   (Singapore)

Author keywords

[No Author keywords available]

Indexed keywords

BUILDING BLOCKS; CHEMICAL LIBRARIES; CHEMICAL STRATEGIES; CLICK CHEMISTRIES; DIPOLAR CYCLOADDITION; DRUG DISCOVERIES; EFFICIENT STRATEGIES; ENZYME INHIBITORS; HIGH THROUGHPUTS; HIGH-THROUGHPUT SYNTHESIS; IN-SITU; KEY COMPONENTS; PRODUCT PURITIES; RAPID SYNTHESIS;

ACETYLENE; CYCLOADDITION; GRAFTING (CHEMICAL); LIBRARIES;

SYNTHESIS (CHEMICAL);

AZIDE; ENZYME INHIBITOR; PROTEIN TYROSINE PHOSPHATASE 1B;

ARTICLE; CHEMICAL STRUCTURE; COMBINATORIAL CHEMISTRY; DRUG ANTAGONISM; DRUG SCREENING; MOLECULAR LIBRARY; SYNTHESIS;

AZIDES; COMBINATORIAL CHEMISTRY TECHNIQUES; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; MOLECULAR STRUCTURE; PROTEIN TYROSINE PHOSPHATASE, NON-RECEPTOR TYPE 1; SMALL MOLECULE LIBRARIES;

EID: 64549106489     PISSN: 14770520     EISSN: None     Source Type: Journal    
DOI: 10.1039/b902338k     Document Type: Article

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