Design, synthesis and assaying of potential aquaporin inhibitors

Handbook of Experimental Pharmacology

Volumn 190, Issue , 2009, Pages 385-402

  Flitsch, Sabine L ^a   Haddoub, Rose ^b   Rützler, Michael ^b   Robin, Aélig ^b  

^a UNIVERSITY OF MANCHESTER   (United Kingdom)

^b NONE

Author keywords

[No Author keywords available]

Indexed keywords

ACETAZOLAMIDE; AQUAPORIN; COPPER; GOLD; INHIBITOR PROTEIN; MERCURY; PHLORETIN; QUATERNARY AMMONIUM DERIVATIVE; SILVER; SULFONAMIDE; TRANSITION ELEMENT; FLUORESCENT DYE; METAL; WATER;

ASSAY; DILUTION; DRUG DESIGN; DRUG SYNTHESIS; FLUORESCENCE; MEMBRANE PERMEABILITY; NONHUMAN; PRIORITY JOURNAL; REVIEW; WATER PERMEABILITY; ANIMAL; BIOASSAY; CELL MEMBRANE PERMEABILITY; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; DRUG EFFECT; HUMAN; INDICATOR DILUTION CURVE; METABOLISM; METHODOLOGY; PROTEIN CONFORMATION; STRUCTURE ACTIVITY RELATION;

ANIMALS; AQUAPORINS; BIOLOGICAL ASSAY; CELL MEMBRANE PERMEABILITY; DRUG DESIGN; FLUORESCENT DYES; HUMANS; INDICATOR DILUTION TECHNIQUES; METALS; MOLECULAR STRUCTURE; PHLORETIN; PROTEIN CONFORMATION; QUATERNARY AMMONIUM COMPOUNDS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; WATER;

EID: 61449361441     PISSN: 01712004     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-3-540-79885-9_19     Document Type: Review

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