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Volumn 456, Issue 4, 2008, Pages 717-720

A yeast-based phenotypic screen for aquaporin inhibitors

Author keywords

Ammonia; Aquaporin; Assay; Compound library screening; Methylamine

Indexed keywords

AQUAPORIN; AQUAPORIN 1; MERCURIC CHLORIDE; METHYLAMINE; TETRYLAMMONIUM;

EID: 43749121916     PISSN: 00316768     EISSN: 14322013     Source Type: Journal    
DOI: 10.1007/s00424-007-0383-3     Document Type: Article
Times cited : (16)

References (14)
  • 1
    • 4444221676 scopus 로고    scopus 로고
    • From structure to disease: The evolving tale of aquaporin biology
    • King LS, Kozono D, Agre P (2004) From structure to disease: the evolving tale of aquaporin biology. Nature Rev 5:687-698
    • (2004) Nature Rev , vol.5 , pp. 687-698
    • King, L.S.1    Kozono, D.2    Agre, P.3
  • 2
    • 0242573122 scopus 로고    scopus 로고
    • Aquaporin water channels: Molecular mechanisms for human diseases
    • Agre P, Kozono D (2003) Aquaporin water channels: molecular mechanisms for human diseases. FEBS Lett 555:72-78
    • (2003) FEBS Lett , vol.555 , pp. 72-78
    • Agre, P.1    Kozono, D.2
  • 3
    • 33845974063 scopus 로고    scopus 로고
    • Regulation and dysregulation of aquaporins in water balance disorders
    • Nielsen S, Kwon TH, Frøkiær J, Agre P (2007) Regulation and dysregulation of aquaporins in water balance disorders. J Intern Med 261:53-64
    • (2007) J Intern Med , vol.261 , pp. 53-64
    • Nielsen, S.1    Kwon, T.H.2    Frøkiær, J.3    Agre, P.4
  • 4
    • 0021251173 scopus 로고
    • Transport of water and urea in red blood cells
    • Macey RI (1984) Transport of water and urea in red blood cells. Am J Physiol 246:C195-C203
    • (1984) Am J Physiol , vol.246
    • MacEy, R.I.1
  • 5
    • 0027472168 scopus 로고
    • The mercury-sensitive residue at cysteine 189 in the CHIP28 water channel
    • Preston GM, Jung JS, Guggino WB, Agre P (1993) The mercury-sensitive residue at cysteine 189 in the CHIP28 water channel. J Biol Chem 268:17-20
    • (1993) J Biol Chem , vol.268 , pp. 17-20
    • Preston, G.M.1    Jung, J.S.2    Guggino, W.B.3    Agre, P.4
  • 6
    • 34047181984 scopus 로고    scopus 로고
    • Structural basis of aquaporin inhibition by mercury
    • Savage DF, Stroud RM (2007) Structural basis of aquaporin inhibition by mercury. J Mol Biol 368:607-617
    • (2007) J Mol Biol , vol.368 , pp. 607-617
    • Savage, D.F.1    Stroud, R.M.2
  • 7
    • 0037145839 scopus 로고    scopus 로고
    • New potent inhibitors of aquaporins: Silver and gold compounds inhibit aquaporins of plant and human origin
    • Niemietz CM, Tyerman SD (2002) New potent inhibitors of aquaporins: silver and gold compounds inhibit aquaporins of plant and human origin. FEBS Lett 531:443-447
    • (2002) FEBS Lett , vol.531 , pp. 443-447
    • Niemietz, C.M.1    Tyerman, S.D.2
  • 8
    • 33747889760 scopus 로고    scopus 로고
    • Expression of heterologous aquaporins for functional analysis in Saccharomyces cerevisiae
    • Pettersson N, Hagström J, Bill RM, Hohmann S (2006) Expression of heterologous aquaporins for functional analysis in Saccharomyces cerevisiae. Curr Genet 50:247-255
    • (2006) Curr Genet , vol.50 , pp. 247-255
    • Pettersson, N.1    Hagström, J.2    Bill, R.M.3    Hohmann, S.4
  • 9
    • 0025706152 scopus 로고
    • Mutations affecting TEA blockade and ion permeation in voltage-activated K+ channels
    • MacKinnon R, Yellen G (1990) Mutations affecting TEA blockade and ion permeation in voltage-activated K+ channels. Science 250:276-279
    • (1990) Science , vol.250 , pp. 276-279
    • MacKinnon, R.1    Yellen, G.2
  • 10
    • 0034014858 scopus 로고    scopus 로고
    • Inhibition of aquaporin-1 water permeability by tetraethylammonium: Involvement of the loop e pore region
    • Brooks HL, Regan JW, Yool AJ (2000) Inhibition of aquaporin-1 water permeability by tetraethylammonium: involvement of the loop E pore region. Mol Pharmacol 57:1021-1026
    • (2000) Mol Pharmacol , vol.57 , pp. 1021-1026
    • Brooks, H.L.1    Regan, J.W.2    Yool, A.J.3
  • 12
    • 31044449089 scopus 로고    scopus 로고
    • Point mutations in the aromatic/arginine region in aquaporin 1 allow passage of urea, glycerol, ammonia, and protons
    • Beitz E, Wu B, Holm LM, Schultz JE, Zeuthen T (2006) Point mutations in the aromatic/arginine region in aquaporin 1 allow passage of urea, glycerol, ammonia, and protons. Proc Natl Acad Sci USA 103:269-274
    • (2006) Proc Natl Acad Sci USA , vol.103 , pp. 269-274
    • Beitz, E.1    Wu, B.2    Holm, L.M.3    Schultz, J.E.4    Zeuthen, T.5
  • 14
    • 34548131086 scopus 로고    scopus 로고
    • Microwave-assisted ring opening of epoxides: A general route to the synthesis of 1-aminopropan-2-ols with anti malaria parasite activities
    • Robin A, Brown F, Bahamontes-Rosa N, Wu B, Beitz E, Kun JF, Flitsch SL (2007) Microwave-assisted ring opening of epoxides: a general route to the synthesis of 1-aminopropan-2-ols with anti malaria parasite activities. J Med Chem 50:4243-4249
    • (2007) J Med Chem , vol.50 , pp. 4243-4249
    • Robin, A.1    Brown, F.2    Bahamontes-Rosa, N.3    Wu, B.4    Beitz, E.5    Kun, J.F.6    Flitsch, S.L.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.