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Volumn 44, Issue 4, 2009, Pages 1457-1462

Synthesis of chlorovinyl sulfones as structural analogs of chalcones and their antiplasmodial activities

(6) Dominguez, Jose N a Leon, Caritza b Rodrigues, Juan a Gamboa de Dominguez, Neira a Gut, Jiri c Rosenthal, Philip J c

a UNIVERSIDAD CENTRAL DE VENEZUELA (Venezuela)

b Universidad Pedagogica Experimental Libertador (Venezuela)

c UNIVERSITY OF CALIFORNIA (United States)

Author keywords

Antimalarial activity; Chalcones; Chlorovinyl sulfones; Synthesis

Indexed keywords

2 PHENYL 1 CHLOROETHENYLPHENYLSULFONE; [2 (1' NAPHTHYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (2' CHLOROPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (2' CHLOROQUINOLIN 3' YL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (2' NAPHTHYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (2',4' DICHLOROPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (2',4',5' TRIMETHOXYPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (2',4',6' TRIMETHOXYPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (3',4' DICHLOROPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (3',4' METHYLENDIOXYPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (3',4',5' TRIMETHOXYPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (4' CHLOROPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (4' CYANOPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (4' FLUOROPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (4' METHOXYPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; [2 (4' NITROPHENYL) 1 CHLORO]ETHENYLPHENYLSULFONE; ANTIMALARIAL AGENT; CHALCONE DERIVATIVE; CHLOROQUINE; HEMOGLOBIN; HEMOZOIN; SULFONE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMALARIAL ACTIVITY; ARTICLE; CLAISEN CONDENSATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISEASE COURSE; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; EXPERIMENTAL INFECTION; EXPERIMENTAL MOUSE; FLOW CYTOMETRY; HYDROLYSIS; IC 50; MALARIA; MOUSE; NONHUMAN; PARASITE CULTIVATION; PLASMODIUM BERGHEI; PLASMODIUM BERGHEI INFECTION; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTIMALARIALS; CHALCONE; HEMEPROTEINS; HEMOGLOBINS; HUMANS; HYDROLYSIS; MALARIA; MICE; PLASMODIUM BERGHEI; PLASMODIUM FALCIPARUM; SULFONES;

EID: 61449255268 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2008.09.044 Document Type: Article

Times cited : (37)

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