Trans-channel interactions in batrachotoxin-modified rat skeletal muscle sodium channels: Kinetic analysis of mutual inhibition between μ-conotoxin GIIIA derivatives and amine blockers

Biophysical Journal

Volumn 95, Issue 9, 2008, Pages 4266-4276

  Ma, Quanli ^a   Pavlov, Evgeny ^a   Britvina, Tatiana ^a   Zamponi, Gerald W ^a   French, Robert J ^a  

^a UNIVERSITY OF CALGARY   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE; BATRACHOTOXIN; CONOTOXIN; CONOTOXIN G3; LIGAND; QUATERNARY AMMONIUM DERIVATIVE; SODIUM CHANNEL; SODIUM CHANNEL BLOCKING AGENT; TETRAPROPYLAMMONIUM; UNCLASSIFIED DRUG;

ANIMAL; ARTICLE; BINDING COMPETITION; CHEMISTRY; DRUG ANTAGONISM; DRUG EFFECT; KINETICS; METABOLISM; PROTEIN BINDING; RAT; SKELETAL MUSCLE;

AMINES; ANIMALS; BATRACHOTOXINS; BINDING, COMPETITIVE; CONOTOXINS; KINETICS; LIGANDS; MUSCLE, SKELETAL; PROTEIN BINDING; QUATERNARY AMMONIUM COMPOUNDS; RATS; SODIUM CHANNEL BLOCKERS; SODIUM CHANNELS;

EID: 58149161250     PISSN: 00063495     EISSN: 15420086     Source Type: Journal    
DOI: 10.1529/biophysj.108.138271     Document Type: Article

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