Strategies for the design of selective protein kinase inhibitors

Mini-Reviews in Medicinal Chemistry

Volumn 8, Issue 12, 2008, Pages 1291-1297

  Sawa, Masaaki ^a  

^a 1 5 5 Minatojima Minamimachi   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE TRIPHOSPHATE; BINDING PROTEIN; CALCIUM CALMODULIN DEPENDENT PROTEIN KINASE; CASEIN KINASE I; CYCLIC AMP DEPENDENT PROTEIN KINASE; CYCLIC GMP DEPENDENT PROTEIN KINASE; CYCLIN DEPENDENT KINASE; DASATINIB; EPIDERMAL GROWTH FACTOR RECEPTOR; ERLOTINIB; GEFITINIB; GLYCOGEN SYNTHASE KINASE; GUANYLATE CYCLASE; IMATINIB; LAPATINIB; MITOGEN ACTIVATED PROTEIN KINASE; NILOTINIB; POTASSIUM CHANNEL HERG; PROTEIN KINASE C; PROTEIN KINASE INHIBITOR; PROTEIN TYROSINE KINASE; PYRAZOLE DERIVATIVE; SORAFENIB; SUNITINIB;

CHANNEL GATING; COMPUTER MODEL; DRUG CONFORMATION; DRUG DESIGN; DRUG PROTEIN BINDING; DRUG SAFETY; DRUG SELECTIVITY; DRUG STRUCTURE; ENZYME INHIBITION; HUMAN; HYDROPHOBICITY; REVIEW;

ADENOSINE TRIPHOSPHATE; ANIMALS; CHEMISTRY, PHARMACEUTICAL; DRUG DESIGN; ENZYME INHIBITORS; ETHER-A-GO-GO POTASSIUM CHANNELS; HUMANS; INFLAMMATION; MODELS, CHEMICAL; PHYLOGENY; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN KINASE INHIBITORS;

EID: 57149144946     PISSN: 13895575     EISSN: None     Source Type: Journal    
DOI: 10.2174/138955708786141043     Document Type: Review

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