메뉴 건너뛰기




Volumn 591, Issue 1-3, 2008, Pages 132-135

Effects of URB597 as an inhibitor of fatty acid amide hydrolase on modulation of nociception in a rat model of cholestasis

Author keywords

(Rat); Antinociception; Cholestasis; Endocannabinoid; Fatty acid amide hydrolase

Indexed keywords

1 (2,4 DICHLOROPHENYL) 5 (4 IODOPHENYL) 4 METHYL N (1 PIPERIDYL) 1H PYRAZOLE 3 CARBOXAMIDE; 5 (4 CHLORO 3 METHYLPHENYL) 1 (4 METHYLBENZYL) N (1,3,3 TRIMETHYLBICYCLO[2.2.1]HEPTAN 2 YL) 3 PYRAZOLECARBOXAMIDE; CANNABINOID 1 RECEPTOR ANTAGONIST; CANNABINOID CB2 RECEPTOR ANTAGONIST; CYCLOHEXYLCARBAMIC ACID 3' CARBAMOYLBIPHENYL 3 YL ESTER; DRUG VEHICLE; ENDOCANNABINOID; ENDOCANNABINOID INHIBITOR; FATTY ACID AMIDASE INHIBITOR; OPIATE RECEPTOR; UNCLASSIFIED DRUG;

EID: 48749116524     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2008.06.061     Document Type: Article
Times cited : (15)

References (36)
  • 2
    • 0028115962 scopus 로고
    • Cholestasis in the male rat is associated with naloxone-reversible antinociception
    • Bergasa N.V., Alling D.W., Vergalla J., and Jones E.A. Cholestasis in the male rat is associated with naloxone-reversible antinociception. J. Hepatol. 20 (1994) 85-90
    • (1994) J. Hepatol. , vol.20 , pp. 85-90
    • Bergasa, N.V.1    Alling, D.W.2    Vergalla, J.3    Jones, E.A.4
  • 3
    • 9744279017 scopus 로고    scopus 로고
    • Cannabinoid/opioid crosstalk in the central nervous system
    • Corchero J., Manzanares J., and Fuentes J.A. Cannabinoid/opioid crosstalk in the central nervous system. Crit. Rev. Neurobiol. 16 (2004) 159-172
    • (2004) Crit. Rev. Neurobiol. , vol.16 , pp. 159-172
    • Corchero, J.1    Manzanares, J.2    Fuentes, J.A.3
  • 5
    • 0031911236 scopus 로고    scopus 로고
    • Endogenous nitric oxide modulates naloxone-precipitated withdrawal signs in a mouse model with acute cholestasis
    • Dehpour A.R., Akbarloo N., and Ghafourifar P. Endogenous nitric oxide modulates naloxone-precipitated withdrawal signs in a mouse model with acute cholestasis. Behav. Pharmacol. 9 (1998) 77-80
    • (1998) Behav. Pharmacol. , vol.9 , pp. 77-80
    • Dehpour, A.R.1    Akbarloo, N.2    Ghafourifar, P.3
  • 7
    • 0033812314 scopus 로고    scopus 로고
    • The effect of the serotonergic system on opioid withdrawal-like syndrome in a mouse model of cholestasis
    • Dehpour A.R., Sadeghipour H.R., Nowroozi A., and Akbarloo N. The effect of the serotonergic system on opioid withdrawal-like syndrome in a mouse model of cholestasis. Hum. Psychopharmacol. 15 (2000) 423-428
    • (2000) Hum. Psychopharmacol. , vol.15 , pp. 423-428
    • Dehpour, A.R.1    Sadeghipour, H.R.2    Nowroozi, A.3    Akbarloo, N.4
  • 10
    • 15744385109 scopus 로고    scopus 로고
    • Characterization of the fatty acid amide hydrolase inhibitor cyclohexyl carbamic acid 3-carbamoyl-biphenyl-3-yl ester (URB597): effects on anandamide and oleoylethanolamide deactivation
    • Fegley D., Gaetani S., Duranti A., Tontini A., Mor M., Tarzia G., and Piomelli D. Characterization of the fatty acid amide hydrolase inhibitor cyclohexyl carbamic acid 3-carbamoyl-biphenyl-3-yl ester (URB597): effects on anandamide and oleoylethanolamide deactivation. J. Pharmacol. Exp. Ther. 313 (2005) 352-358
    • (2005) J. Pharmacol. Exp. Ther. , vol.313 , pp. 352-358
    • Fegley, D.1    Gaetani, S.2    Duranti, A.3    Tontini, A.4    Mor, M.5    Tarzia, G.6    Piomelli, D.7
  • 11
    • 0141453951 scopus 로고    scopus 로고
    • The cannabinoid agonist WIN 55, 212-2 increases nociception threshold in cholestatic rats: implications for the treatment of the pruritus of cholestasis
    • Gingold A.R., and Bergasa N.V. The cannabinoid agonist WIN 55, 212-2 increases nociception threshold in cholestatic rats: implications for the treatment of the pruritus of cholestasis. Life Sci. 73 (2003) 2741-2747
    • (2003) Life Sci. , vol.73 , pp. 2741-2747
    • Gingold, A.R.1    Bergasa, N.V.2
  • 12
    • 33845320132 scopus 로고    scopus 로고
    • Modulation of cholestasis-induced antinociception in rats by two NMDA receptor antagonists: MK-801 and magnesium sulfate
    • Hasanein P., Parviz M., Keshavarz M., Javanmardi K., Allahtavakoli M., and Ghaseminejad M. Modulation of cholestasis-induced antinociception in rats by two NMDA receptor antagonists: MK-801 and magnesium sulfate. Eur. J. Pharmacol. 554 (2007) 123-127
    • (2007) Eur. J. Pharmacol. , vol.554 , pp. 123-127
    • Hasanein, P.1    Parviz, M.2    Keshavarz, M.3    Javanmardi, K.4    Allahtavakoli, M.5    Ghaseminejad, M.6
  • 14
    • 0037207078 scopus 로고    scopus 로고
    • Spinal and peripheral mechanisms of cannabinoid antinociception: behavioral, neurophysiological and neuroanatomical perspectives
    • Hohmann A.G. Spinal and peripheral mechanisms of cannabinoid antinociception: behavioral, neurophysiological and neuroanatomical perspectives. Chem. Phys. Lipids 121 (2002) 173-190
    • (2002) Chem. Phys. Lipids , vol.121 , pp. 173-190
    • Hohmann, A.G.1
  • 15
    • 33845344400 scopus 로고    scopus 로고
    • An endocannabinoid mechanism for stress-induced analgesia
    • Hohmann A.G., and Suplita R.L. An endocannabinoid mechanism for stress-induced analgesia. AAPS J. 8 (2006) E693-E708
    • (2006) AAPS J. , vol.8
    • Hohmann, A.G.1    Suplita, R.L.2
  • 17
    • 22544467758 scopus 로고    scopus 로고
    • Involvement of N-methyl-d-aspartate receptors and nitric oxide in the rostral ventromedial medulla in modulating morphine pain-inhibitory signals from the periaqueductal grey matter in rats
    • Javanmardi K., Parviz M., Sadr S.S., Keshavarz M., Minaii B., and Dehpour A.R. Involvement of N-methyl-d-aspartate receptors and nitric oxide in the rostral ventromedial medulla in modulating morphine pain-inhibitory signals from the periaqueductal grey matter in rats. Clin. Exp. Pharmacol. Physiol. 32 (2005) 585-589
    • (2005) Clin. Exp. Pharmacol. Physiol. , vol.32 , pp. 585-589
    • Javanmardi, K.1    Parviz, M.2    Sadr, S.S.3    Keshavarz, M.4    Minaii, B.5    Dehpour, A.R.6
  • 19
    • 35648999552 scopus 로고    scopus 로고
    • Endocannabinoid metabolism and uptake: novel targets for neuropathic and inflammatory pain
    • Jhaveri M.D., Richardson D., and Chapman V. Endocannabinoid metabolism and uptake: novel targets for neuropathic and inflammatory pain. Br. J. Pharmacol. 152 (2007) 624-632
    • (2007) Br. J. Pharmacol. , vol.152 , pp. 624-632
    • Jhaveri, M.D.1    Richardson, D.2    Chapman, V.3
  • 21
    • 4644354869 scopus 로고    scopus 로고
    • Reversible inhibitors of fatty acid amide hydrolase that promote analgesia: evidence for an unprecedented combination of potency and selectivity
    • Lichtman A.H., Leung D., Shelton C.C., Saghatelian A., Hardouin C., Boger D.L., and Cravatt B.F. Reversible inhibitors of fatty acid amide hydrolase that promote analgesia: evidence for an unprecedented combination of potency and selectivity. J. Pharmacol. Exp. Ther. 311 (2004) 441-448
    • (2004) J. Pharmacol. Exp. Ther. , vol.311 , pp. 441-448
    • Lichtman, A.H.1    Leung, D.2    Shelton, C.C.3    Saghatelian, A.4    Hardouin, C.5    Boger, D.L.6    Cravatt, B.F.7
  • 22
    • 0025325535 scopus 로고
    • Structure of a cannabinoid receptor and functional expression of the cloned cDNA
    • Matsuda L.A., Lolait S.J., Brownstein M.J., Young A.C., and Bonner T.I. Structure of a cannabinoid receptor and functional expression of the cloned cDNA. Nature 346 (1990) 561-564
    • (1990) Nature , vol.346 , pp. 561-564
    • Matsuda, L.A.1    Lolait, S.J.2    Brownstein, M.J.3    Young, A.C.4    Bonner, T.I.5
  • 23
    • 22244484464 scopus 로고    scopus 로고
    • Structure and function of fatty acid amide hydrolase
    • McKinney M.K., and Cravatt B.F. Structure and function of fatty acid amide hydrolase. Annu. Rev. Biochem. 74 (2005) 411-432
    • (2005) Annu. Rev. Biochem. , vol.74 , pp. 411-432
    • McKinney, M.K.1    Cravatt, B.F.2
  • 24
    • 0035838275 scopus 로고    scopus 로고
    • CB1 receptor mediated analgesia from the Nucleus Reticularis Gigantocellularis pars alpha is activated in an animal model of neuropathic pain
    • Monhemius R., Azami J., Green D.L., and Roberts M.H. CB1 receptor mediated analgesia from the Nucleus Reticularis Gigantocellularis pars alpha is activated in an animal model of neuropathic pain. Brain Res. 908 (2001) 67-74
    • (2001) Brain Res. , vol.908 , pp. 67-74
    • Monhemius, R.1    Azami, J.2    Green, D.L.3    Roberts, M.H.4
  • 27
    • 33746880309 scopus 로고    scopus 로고
    • Endogenous opioid-mediated antinociception in cholestatic mice is peripherally, not centrally, mediated
    • Nelson L., Vergnolle N., D'Mello C., Chapman K., Le T., and Swain M.G. Endogenous opioid-mediated antinociception in cholestatic mice is peripherally, not centrally, mediated. J. Hepatol. 44 (2006) 1141-1149
    • (2006) J. Hepatol. , vol.44 , pp. 1141-1149
    • Nelson, L.1    Vergnolle, N.2    D'Mello, C.3    Chapman, K.4    Le, T.5    Swain, M.G.6
  • 28
    • 0036183282 scopus 로고    scopus 로고
    • Modulation of cholestasis-induced antinociception by CCK receptor agonists and antagonists
    • Rastegar H., Homayoun H., Afifi M., Rezayat M., and Dehpour A.R. Modulation of cholestasis-induced antinociception by CCK receptor agonists and antagonists. Eur. Neuropsychopharmacol. 12 (2002) 111-118
    • (2002) Eur. Neuropsychopharmacol. , vol.12 , pp. 111-118
    • Rastegar, H.1    Homayoun, H.2    Afifi, M.3    Rezayat, M.4    Dehpour, A.R.5
  • 30
    • 0032056333 scopus 로고    scopus 로고
    • Characterization of delta9-tetrahydrocannabinol and anandamide antinociception in nonarthritic and arthritic rats
    • Smith F.L., Fujimori K., Lowe J., and Welch S.P. Characterization of delta9-tetrahydrocannabinol and anandamide antinociception in nonarthritic and arthritic rats. Pharmacol. Biochem. Behav. 60 (1998) 183-191
    • (1998) Pharmacol. Biochem. Behav. , vol.60 , pp. 183-191
    • Smith, F.L.1    Fujimori, K.2    Lowe, J.3    Welch, S.P.4
  • 32
    • 0028204163 scopus 로고
    • Adrenal secretion of BAM-22P, a potent opioid peptide, is enhanced in rats with acute cholestasis
    • Swain M.G., MacArthur L., Vergalla J., and Jones E.A. Adrenal secretion of BAM-22P, a potent opioid peptide, is enhanced in rats with acute cholestasis. Am. J. Physiol. 266 (1994) G201-G205
    • (1994) Am. J. Physiol. , vol.266
    • Swain, M.G.1    MacArthur, L.2    Vergalla, J.3    Jones, E.A.4
  • 33
    • 0024211842 scopus 로고
    • Opioid peptides and primary biliary cirrhosis
    • Thornton J.R., and Losowsky M.S. Opioid peptides and primary biliary cirrhosis. BMJ 297 (1988) 1501-1504
    • (1988) BMJ , vol.297 , pp. 1501-1504
    • Thornton, J.R.1    Losowsky, M.S.2
  • 34
    • 0024494152 scopus 로고
    • Methionine enkephalin is increased in plasma in acute liver disease and is present in bile and urine
    • Thornton J.R., and Losowsky M.S. Methionine enkephalin is increased in plasma in acute liver disease and is present in bile and urine. J. Hepatol. 8 (1989) 53-59
    • (1989) J. Hepatol. , vol.8 , pp. 53-59
    • Thornton, J.R.1    Losowsky, M.S.2
  • 36
    • 0033458086 scopus 로고    scopus 로고
    • Synergistic interactions of endogenous opioids and cannabinoid systems
    • Welch S.P., and Eads M. Synergistic interactions of endogenous opioids and cannabinoid systems. Brain Res. 848 (1999) 183-190
    • (1999) Brain Res. , vol.848 , pp. 183-190
    • Welch, S.P.1    Eads, M.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.