Radiolabeled glucocorticoids as molecular probes for imaging brain glucocorticoid receptors by means of positron emission tomography (PET)

Mini-Reviews in Medicinal Chemistry

Volumn 8, Issue 7, 2008, Pages 728-739

  Steiniger, Björn ^a   Kniess, Torsten ^a   Bergmann, Ralf ^a   Pietzsch, Jens ^a   Wuest, Frank R ^a  

^a INSTITUTE OF ION BEAM PHYSICS AND MATERIALS RESEARCH   (Germany)

Author keywords

Carbon 11; Fluorine 18; Glucocorticoid receptor; PET; Radioligands

Indexed keywords

11BETA,17BETA DIHYDROXY 6 METHYL 17ALPHA (1 PROPYNYL)ANDROSTA 1,4,6 TRIEN 3 ONE; 21 FLUORO 21 DEOXYDEXAMETHASONE F 18; 21 FLUORO 21 DEOXYTRIAMCINOLONE ACETONIDE F 18; 21 FLUORODEACYLCORTIVAZOL F 18; 21 FLUOROPREDNISONE F 18; 4 FLUOROPHENYL[3,2 C]PYRAZOLO STEROID F 18; CARBON 13; CORTISONE; DEACYLCORTIVAZOL F 18; DEXAMETHASONE; FLUORINE 18; GLUCOCORTICOID; GLUCOCORTICOID RECEPTOR; HYDROCORTISONE; NIVACORTOL; PREDNISOLONE; RADIOPHARMACEUTICAL AGENT; TRACER;

BINDING AFFINITY; BLOOD BRAIN BARRIER; DRUG DESIGN; DRUG PENETRATION; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; ISOTOPE LABELING; LIGAND BINDING; LIPOPHILICITY; MOLECULAR PROBE; NEUROIMAGING; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; REVIEW; STRUCTURE ANALYSIS; ANIMAL; BRAIN; CHEMISTRY; PHYSIOLOGY; SCINTISCANNING; SYNTHESIS;

ANIMALS; BRAIN; GLUCOCORTICOIDS; MOLECULAR PROBES; POSITRON-EMISSION TOMOGRAPHY; RADIOPHARMACEUTICALS; RECEPTORS, GLUCOCORTICOID;

EID: 46749146151     PISSN: 13895575     EISSN: None     Source Type: Journal    
DOI: 10.2174/138955708784567403     Document Type: Review

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