메뉴 건너뛰기




Volumn 35, Issue 4, 2008, Pages 393-400

[64Cu]diacetyl-bis(N4-methyl-thiosemicarbazone) - a radiotracer for tumor hypoxia

Author keywords

Cu ATSM; Hypoxia; PET; Tumor

Indexed keywords

DIACETYL BIS(N4 METHYL THIOSEMICARBAZONE) CU 64; TRACER; TUMOR MARKER;

EID: 43049165789     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2008.02.002     Document Type: Review
Times cited : (35)

References (30)
  • 2
    • 0242417596 scopus 로고    scopus 로고
    • Assessing tumor hypoxia in cervical cancer by positron emission tomography with 60Cu-ATSM: relationship to therapeutic response-a preliminary report
    • F. Dehdashti P.W. Grigsby M.A. Mintun J.S. Lewis B.A. Siegel M.J. Welch Assessing tumor hypoxia in cervical cancer by positron emission tomography with 60Cu-ATSM: relationship to therapeutic response-a preliminary report Int J Radiat Oncol Biol Phys 55 5 2003 1233 1238
    • (2003) Int J Radiat Oncol Biol Phys , vol.55 , Issue.5 , pp. 1233-1238
    • Dehdashti, F.1    Grigsby, P.W.2    Mintun, M.A.3    Lewis, J.S.4    Siegel, B.A.5    Welch, M.J.6
  • 4
    • 11144265734 scopus 로고    scopus 로고
    • Current imaging paradigms in radiation oncology
    • S. Apisarnthanarax K.S. Chao Current imaging paradigms in radiation oncology Radiat Res 163 1 2005 1 25
    • (2005) Radiat Res , vol.163 , Issue.1 , pp. 1-25
    • Apisarnthanarax, S.1    Chao, K.S.2
  • 5
    • 0024998672 scopus 로고
    • 62Cu-labelling of human serum albumin-dithiosemicarbazone (HSA-DTS) conjugate for regional plasma volume measurement: application of new 62Zn/62Cu generator system
    • Y. Fujibayashi K. Matsumoto Y. Arano Y. Yonekura J. Konishi A. Yokoyama 62Cu-labelling of human serum albumin-dithiosemicarbazone (HSA-DTS) conjugate for regional plasma volume measurement: application of new 62Zn/62Cu generator system Chem Pharm Bull 38 1990 1946
    • (1990) Chem Pharm Bull , vol.38 , pp. 1946
    • Fujibayashi, Y.1    Matsumoto, K.2    Arano, Y.3    Yonekura, Y.4    Konishi, J.5    Yokoyama, A.6
  • 6
    • 44049114161 scopus 로고
    • Subcellular distribution of tissue radiocopper following intravenous administration of [67Cu]-labelled Cu-PTSM
    • I.D. Baerga R.P. Maickel M.A. Green Subcellular distribution of tissue radiocopper following intravenous administration of [67Cu]-labelled Cu-PTSM Nucl Med Biol 19 6 1992 697 701
    • (1992) Nucl Med Biol , vol.19 , Issue.6 , pp. 697-701
    • Baerga, I.D.1    Maickel, R.P.2    Green, M.A.3
  • 7
    • 0027215118 scopus 로고
    • Evaluation of copper-labelled bifunctional chelate–albumin conjugates for blood pool imaging
    • C.J. Anderson P.A. Rocque C.J. Weinheimer M.J. Welch Evaluation of copper-labelled bifunctional chelate–albumin conjugates for blood pool imaging Nucl Med Biol 20 4 1993 461 467
    • (1993) Nucl Med Biol , vol.20 , Issue.4 , pp. 461-467
    • Anderson, C.J.1    Rocque, P.A.2    Weinheimer, C.J.3    Welch, M.J.4
  • 9
    • 0041519423 scopus 로고    scopus 로고
    • Hypoxia-targeting copper bis(selenosemicarbazone) complexes: comparison with their sulfur analogues
    • Castle TC Maurer RI Sowrey FE Went MJ Reynolds CA McInnes EJ Hypoxia-targeting copper bis(selenosemicarbazone) complexes: comparison with their sulfur analogues J Am Chem Soc 125 33 2003 10040 10049
    • (2003) J Am Chem Soc , vol.125 , Issue.33 , pp. 10040-10049
    • Castle, TC1    Maurer, RI2    Sowrey, FE3    Went, MJ4    Reynolds, CA5    McInnes, EJ6
  • 10
    • 0030811565 scopus 로고    scopus 로고
    • Copper-62-ATSM: a new hypoxia imaging agent with high membrane permeability and low redox potential
    • Y. Fujibayashi H. Taniuchi Y. Yonekura H. Ohtani J. Konishi A. Yokoyama Copper-62-ATSM: a new hypoxia imaging agent with high membrane permeability and low redox potential J Nucl Med 38 7 1997 1155 1160
    • (1997) J Nucl Med , vol.38 , Issue.7 , pp. 1155-1160
    • Fujibayashi, Y.1    Taniuchi, H.2    Yonekura, Y.3    Ohtani, H.4    Konishi, J.5    Yokoyama, A.6
  • 12
    • 0035043960 scopus 로고    scopus 로고
    • Tumor uptake of copper-diacetyl-bis(N(4)-methylthiosemicarbazone): effect of changes in tissue oxygenation
    • J.S. Lewis T.L. Sharp R. Laforest Y. Fujibayashi M.J. Welch Tumor uptake of copper-diacetyl-bis( N (4)-methylthiosemicarbazone): effect of changes in tissue oxygenation J Nucl Med 42 4 2001 655 661
    • (2001) J Nucl Med , vol.42 , Issue.4 , pp. 655-661
    • Lewis, J.S.1    Sharp, T.L.2    Laforest, R.3    Fujibayashi, Y.4    Welch, M.J.5
  • 13
    • 0030292909 scopus 로고    scopus 로고
    • Copper radionuclides and radiopharmaceuticals in nuclear medicine
    • P.J. Blower J.S. Lewis J. Zweit Copper radionuclides and radiopharmaceuticals in nuclear medicine Nucl Med Biol 23 1996 957 980
    • (1996) Nucl Med Biol , Issue.23 , pp. 957-980
    • Blower, P.J.1    Lewis, J.S.2    Zweit, J.3
  • 14
    • 35548962244 scopus 로고    scopus 로고
    • Cu-ATSM: a radiopharmaceutical for the PET imaging of hypoxia
    • A.L. Vavere J.S. Lewis Cu-ATSM: a radiopharmaceutical for the PET imaging of hypoxia Dalton Trans 43 2007 4983 5902
    • (2007) Dalton Trans , Issue.43 , pp. 4983-5902
    • Vavere, A.L.1    Lewis, J.S.2
  • 15
    • 0032556442 scopus 로고    scopus 로고
    • Redox-active metal complexes for imaging hypoxic tissues: structure–activity relationships in copper(II) bis(thiosemicarbazone) complexes
    • J.L.J. Dearling J.S. Lewis D.W. McCarthy M.J. Welch P.J. Blower Redox-active metal complexes for imaging hypoxic tissues: structure–activity relationships in copper(II) bis(thiosemicarbazone) complexes Chem Commun 1998 2531 2532
    • (1998) Chem Commun , pp. 2531-2532
    • Dearling, J.L.J.1    Lewis, J.S.2    McCarthy, D.W.3    Welch, M.J.4    Blower, P.J.5
  • 16
    • 33746089972 scopus 로고    scopus 로고
    • Intertumoral differences in hypoxia selectivity of the PET imaging agent 64Cu(II)-diacetyl-bis(N4-methylthiosemicarbazone)
    • H. Yuan T. Schroeder J.E. Bowsher L.W. Hedlund T. Wong M.W. Dewhirst Intertumoral differences in hypoxia selectivity of the PET imaging agent 64Cu(II)-diacetyl-bis( N 4-methylthiosemicarbazone) J Nucl Med 47 6 2006 989 998
    • (2006) J Nucl Med , vol.47 , Issue.6 , pp. 989-998
    • Yuan, H.1    Schroeder, T.2    Bowsher, J.E.3    Hedlund, L.W.4    Wong, T.5    Dewhirst, M.W.6
  • 17
    • 34247890108 scopus 로고    scopus 로고
    • The influence of tumor oxygenation on hypoxia imaging in murine squamous cell carcinoma using [64Cu]Cu-ATSM or [18F]fluoromisonidazole positron emission tomography
    • K. Matsumoto L. Szajek M.C. Krishna J.A. Cook J. Seidel K. Grimes The influence of tumor oxygenation on hypoxia imaging in murine squamous cell carcinoma using [64Cu]Cu-ATSM or [18F]fluoromisonidazole positron emission tomography Int J Oncol 30 4 2007 873 881
    • (2007) Int J Oncol , vol.30 , Issue.4 , pp. 873-881
    • Matsumoto, K.1    Szajek, L.2    Krishna, M.C.3    Cook, J.A.4    Seidel, J.5    Grimes, K.6
  • 19
    • 0036943656 scopus 로고    scopus 로고
    • Copper bis(thiosemicarbazone) complexes as hypoxia imaging agents: structure–activity relationships
    • J.L.J. Dearling J.S. Lewis G.E.D. Mullen M.J. Welch P.J. Blower Copper bis(thiosemicarbazone) complexes as hypoxia imaging agents: structure–activity relationships J Biol Inorg Chem 7 2002 249 259
    • (2002) J Biol Inorg Chem , vol.7 , pp. 249-259
    • Dearling, J.L.J.1    Lewis, J.S.2    Mullen, G.E.D.3    Welch, M.J.4    Blower, P.J.5
  • 20
    • 22144449210 scopus 로고    scopus 로고
    • Cell line-dependent differences in uptake and retention of the hypoxia-selective nuclear imaging agent Cu-ATSM
    • P. Burgman J.A. O'Donoghue J.S. Lewis M.J. Welch J.L. Humm C. Ling Cell line-dependent differences in uptake and retention of the hypoxia-selective nuclear imaging agent Cu-ATSM Nucl Med Biol 32 2005 623 630
    • (2005) Nucl Med Biol , vol.32 , pp. 623-630
    • Burgman, P.1    O'Donoghue, J.A.2    Lewis, J.S.3    Welch, M.J.4    Humm, J.L.5    Ling, C.6
  • 21
    • 0034832606 scopus 로고    scopus 로고
    • Copper homeostasis: the role of cellular transporters
    • E. Harris Copper homeostasis: the role of cellular transporters Nutr Rev 59 2001 281 285
    • (2001) Nutr Rev , vol.59 , pp. 281-285
    • Harris, E.1
  • 22
    • 0041341920 scopus 로고    scopus 로고
    • The copper export pump nATP7B modulates the cellular pharmacology of carboplatin in ovarian carcinoma cells
    • K. Katano R. Safaei G. Samimi A. Holzer M. Rochdi S.B. Howell The copper export pump nATP7B modulates the cellular pharmacology of carboplatin in ovarian carcinoma cells Mol Pharmacol 64 2003 466 473
    • (2003) Mol Pharmacol , vol.64 , pp. 466-473
    • Katano, K.1    Safaei, R.2    Samimi, G.3    Holzer, A.4    Rochdi, M.5    Howell, S.B.6
  • 23
    • 0032923178 scopus 로고    scopus 로고
    • Comparative studies of Cu-64-ATSM and C-11-acetate in an acute myocardial infarction model: ex vivo imaging of hypoxia in rats
    • Y. Fujibayashi C.S. Cutler C.J. Anderson D.W. McCarthy L.A. Jones T. Sharp Comparative studies of Cu-64-ATSM and C-11-acetate in an acute myocardial infarction model: ex vivo imaging of hypoxia in rats Nucl Med Biol 26 1999 117 121
    • (1999) Nucl Med Biol , vol.26 , pp. 117-121
    • Fujibayashi, Y.1    Cutler, C.S.2    Anderson, C.J.3    McCarthy, D.W.4    Jones, L.A.5    Sharp, T.6
  • 24
    • 0036841704 scopus 로고    scopus 로고
    • Delineation of hypoxia in canine myocardium using PET and copper(II)-diacetyl-bis(N(4)-methylthiosemicarbazone)
    • J.S. Lewis P. Herrero T.L. Sharp J.A. Engelbach Y. Fujibayashi R. Laforest Delineation of hypoxia in canine myocardium using PET and copper(II)-diacetyl-bis( N (4)-methylthiosemicarbazone) J Nucl Med 43 11 2002 1557 1569
    • (2002) J Nucl Med , vol.43 , Issue.11 , pp. 1557-1569
    • Lewis, J.S.1    Herrero, P.2    Sharp, T.L.3    Engelbach, J.A.4    Fujibayashi, Y.5    Laforest, R.6
  • 26
    • 20144387807 scopus 로고    scopus 로고
    • Assessment of regional tumor hypoxia using 18F-fluoromisonidazole and 64Cu(II)-diacetyl-bis(N4-methylthiosemicarbazone) positron emission tomography: comparative study featuring microPET imaging, Po2 probe measurement, autoradiography, and fluorescent microscopy in the R3327-AT and FaDu rat tumor models
    • J.A. O'Donoghue P. Zanzonico A. Pugachev B. Wen Smith-Jones S. Cai Assessment of regional tumor hypoxia using 18F-fluoromisonidazole and 64Cu(II)-diacetyl-bis( N 4-methylthiosemicarbazone) positron emission tomography: comparative study featuring microPET imaging, Po2 probe measurement, autoradiography, and fluorescent microscopy in the R3327-AT and FaDu rat tumor models Int J Radiat Oncol Biol Phys 61 5 2005 1493 1502
    • (2005) Int J Radiat Oncol Biol Phys , vol.61 , Issue.5 , pp. 1493-1502
    • O'Donoghue, J.A.1    Zanzonico, P.2    Pugachev, A.3    Wen, B.4    Smith-Jones5    Cai, S.6
  • 27
    • 20444490000 scopus 로고    scopus 로고
    • Saptial heterogeneity and oxygen dependence of glucose consumption in R3230Ac and fibrosarcomas of the Fischer 344 rat
    • T. Schroeder H. Yuan B.L. Viglianti C. Peltz S. Asopa Z. Vujaskovic Saptial heterogeneity and oxygen dependence of glucose consumption in R3230Ac and fibrosarcomas of the Fischer 344 rat Cancer Res 65 2005 5163 5171
    • (2005) Cancer Res , Issue.65 , pp. 5163-5171
    • Schroeder, T.1    Yuan, H.2    Viglianti, B.L.3    Peltz, C.4    Asopa, S.5    Vujaskovic, Z.6
  • 28
    • 0035869722 scopus 로고    scopus 로고
    • A novel approach to overcome hypoxic tumor resistance: Cu-ATSM-guided intensity-modulated radiation therapy
    • K.S. Chao W.R. Bosch S. Mutic J.S. Lewis F. Dehdashti M.A. Mintun A novel approach to overcome hypoxic tumor resistance: Cu-ATSM-guided intensity-modulated radiation therapy Int J Radiat Oncol Biol Phys 49 4 2001 1171 1182
    • (2001) Int J Radiat Oncol Biol Phys , vol.49 , Issue.4 , pp. 1171-1182
    • Chao, K.S.1    Bosch, W.R.2    Mutic, S.3    Lewis, J.S.4    Dehdashti, F.5    Mintun, M.A.6
  • 29
    • 0029955072 scopus 로고    scopus 로고
    • Pretreatment oxygenation predicts radiation response in advanced squamous cell carcinoma of the head and neck
    • M. Nordsmark M. Overgaard J. Overgaard Pretreatment oxygenation predicts radiation response in advanced squamous cell carcinoma of the head and neck Radiother Oncol 41 1 1996 31 39
    • (1996) Radiother Oncol , vol.41 , Issue.1 , pp. 31-39
    • Nordsmark, M.1    Overgaard, M.2    Overgaard, J.3
  • 30
    • 85120249087 scopus 로고    scopus 로고
    • Use of 64Cu-ATSM for identifying tumour hypoxia in squamous cell carcinoma of the head and neck
    • M. Saunders Use of 64Cu-ATSM for identifying tumour hypoxia in squamous cell carcinoma of the head and neck 2007 UCL and Mount Vernon Hospital London
    • (2007)
    • Saunders, M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.