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Volumn 2, Issue 10, 2007, Pages 1414-1417

Naphthyl tetronic acids as multi-target inhibitors of bacterial peptidoglycan biosynthesis

(16) Mansour, Tarek S a Caufield, Craig E b Rasmussen, Beth a Chopra, Rajiv b Krishnamurthy, Girija a Morris, Koi M b Svenson, Kristine b Bard, Joel b Smeltzer, Claudia a Naughton, Shaughnessy b Antane, Schuyler b Yang, Youjun a Severin, Anatoly a Quagliato, Dominick b Petersen, Peter J a Singh, Guy a

a WYETH RESEARCH (United States)

b PFIZER INC (United States)

Author keywords

Antibiotics; Furanones; Inhibitors; Naphthyl tetronic acids; Pulvinones

Indexed keywords

ANTIINFECTIVE AGENT; FURAN DERIVATIVE; PEPTIDOGLYCAN; TETRONIC ACID; UNCLASSIFIED DRUG;

ARTICLE; BACTERIUM; BIOSYNTHESIS; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECT; METABOLISM; MICROBIOLOGICAL EXAMINATION; SYNTHESIS;

ANTI-BACTERIAL AGENTS; BACTERIA; FURANS; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR; PEPTIDOGLYCAN;

EID: 42149141235 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200700094 Document Type: Article

Times cited : (42)

References (35)

1
- 22144465528
- S. Stefani, Curr. Med. Chem.: Anti-Infect. Agents 2005, 4, 235-257.
- (2005) Curr. Med. Chem.: Anti-Infect. Agents , vol.4 , pp. 235-257
- Stefani, S.¹

2
- 0242291985
- S. J. Projan, Curr. Opin. Microbiol. 2003, 6, 427-430.
- (2003) Curr. Opin. Microbiol , vol.6 , pp. 427-430
- Projan, S.J.¹

3
- 33845903833
- D. J. Payne, M. N. Gwynn, D. J. Holmes, D. L. Pompliano, Nat. Rev. Drug Discovery 2007, 6, 29-40.
- (2007) Nat. Rev. Drug Discovery , vol.6 , pp. 29-40
- Payne, D.J.¹ Gwynn, M.N.² Holmes, D.J.³ Pompliano, D.L.⁴

4
- 0042908666
- ASM Press, Washington DC
- C. Walsh, Antibiotics, Actions, Origins, Resistance, ASM Press, Washington DC, 2003.
- (2003) Antibiotics, Actions, Origins, Resistance
- Walsh, C.¹

5
- 0037223505
- A. El Zoeiby, F. Sanschagrin, R. C. Levesque, Mol. Microbiol. 2003, 47, 1-12.
- (2003) Mol. Microbiol , vol.47 , pp. 1-12
- El Zoeiby, A.¹ Sanschagrin, F.² Levesque, R.C.³

6
- 0034812451
- A. L. Koch, Antimicrob. Agents Chemother. 2001, 45, 2671-2675.
- (2001) Antimicrob. Agents Chemother , vol.45 , pp. 2671-2675
- Koch, A.L.¹

7
- 0142074781
- S. Utaida, P. M. Dunman, D. Macapagal, D. Murphy, S. J. Projan, V. K. Singh, R. K. Jayaswal, B. J. Wilkinson, Microbiology 2003, 149, 2719-2732.
- (2003) Microbiology , vol.149 , pp. 2719-2732
- Utaida, S.¹ Dunman, P.M.² Macapagal, D.³ Murphy, D.⁴ Projan, S.J.⁵ Singh, V.K.⁶ Jayaswal, R.K.⁷ Wilkinson, B.J.⁸

8
- 22144498106
- B. J. Wilkinson, A. Muthaiyan and R. K. Jayaswal, Curr. Med. Chem.: Anti-Infect. Agents 2005, 4, 259-276.
- (2005) Curr. Med. Chem.: Anti-Infect. Agents , vol.4 , pp. 259-276
- Wilkinson, B.J.¹ Muthaiyan, A.² Jayaswal, R.K.³

9
- 33748764203
- A. Bachelier, R. Mayer, C. D. Klein, Bioorg. Med. Chem. Lett. 2006, 16, 5605-5609.
- (2006) Bioorg. Med. Chem. Lett , vol.16 , pp. 5605-5609
- Bachelier, A.¹ Mayer, R.² Klein, C.D.³

10
- 17144418885
- S. Eschenburg, M. A. Priestman, F. A. Abdul-Latif, C. Delchaume, F. Fassy, E. Schoenbrum, J. Biol. Chem. 2005, 280, 14070-14075.
- (2005) J. Biol. Chem , vol.280 , pp. 14070-14075
- Eschenburg, S.¹ Priestman, M.A.² Abdul-Latif, F.A.³ Delchaume, C.⁴ Fassy, F.⁵ Schoenbrum, E.⁶

11
- 14844347076
- S. Mizyed, A. Oddone, B. Byczynski, D. W. Hughes, P. J. Berti, Biochemistry 2005, 44, 4011-4017.
- (2005) Biochemistry , vol.44 , pp. 4011-4017
- Mizyed, S.¹ Oddone, A.² Byczynski, B.³ Hughes, D.W.⁴ Berti, P.J.⁵

12
- 0037430432
- J. J. Bronson, K. DenBleyker, L. Kenneth, P. J. Falk, R. A. Mate, H. T. Ho, M. J. Pucci, L. B. Snyder, Bioorg. Med. Chem. Lett. 2003, 13, 873-875.
- (2003) Bioorg. Med. Chem. Lett , vol.13 , pp. 873-875
- Bronson, J.J.¹ DenBleyker, K.² Kenneth, L.³ Falk, P.J.⁴ Mate, R.A.⁵ Ho, H.T.⁶ Pucci, M.J.⁷ Snyder, L.B.⁸

13
- 0034678644
- C. J. Andres, J. J. Bronson, S. V. D'Andrea, M. S. Deshpande, S. Milind, P. J. Falk, K. A. Grant-Young, W. E. Harte, H. T. Ho, P. F. Misco, J. G. Robertson, D. Stock, Y. Sun, A. W. Walsh, Bioorg. Med. Chem. Lett. 2000, 10, 715-717.
- (2000) Bioorg. Med. Chem. Lett , vol.10 , pp. 715-717
- Andres, C.J.¹ Bronson, J.J.² D'Andrea, S.V.³ Deshpande, M.S.⁴ Milind, S.⁵ Falk, P.J.⁶ Grant-Young, K.A.⁷ Harte, W.E.⁸ Ho, H.T.⁹ Misco, P.F.¹⁰ Robertson, J.G.¹¹ Stock, D.¹² Sun, Y.¹³ Walsh, A.W.¹⁴

14
- 10744223112
- Z. Li, G. D. Francisco, W. Hu, P. Labthavikul, P. J. Petersen, A. Severin, G. Singh, Y. Yang, B. A. Rasumessen, Y. I. Lin, J. S. Skotnicki, T. S. Mansour, Bioorg. Med. Chem. Lett. 2003, 13, 2591-2594.
- (2003) Bioorg. Med. Chem. Lett , vol.13 , pp. 2591-2594
- Li, Z.¹ Francisco, G.D.² Hu, W.³ Labthavikul, P.⁴ Petersen, P.J.⁵ Severin, A.⁶ Singh, G.⁷ Yang, Y.⁸ Rasumessen, B.A.⁹ Lin, Y.I.¹⁰ Skotnicki, J.S.¹¹ Mansour, T.S.¹²

15
- 0035833985
- S. Marmor, C. P. Petersen, F. Reck, W. Yang, N. Gao, S. L. Fisher, Biochemistry 2001, 40, 12207-12214.
- (2001) Biochemistry , vol.40 , pp. 12207-12214
- Marmor, S.¹ Petersen, C.P.² Reck, F.³ Yang, W.⁴ Gao, N.⁵ Fisher, S.L.⁶

16
- 33749531892
- J. Humljan, M. Kotnik, A. Boniface, T. Solmajer, U. Urleb, D. Blanot, S. Gobec, Tetrahedron 2006, 62, 10980-10988.
- (2006) Tetrahedron , vol.62 , pp. 10980-10988
- Humljan, J.¹ Kotnik, M.² Boniface, A.³ Solmajer, T.⁴ Urleb, U.⁵ Blanot, D.⁶ Gobec, S.⁷

17
- 33745068955
- G. F. Stamper, K. L. Longenecker, E. H. Fry, G. Clarissa, A. S. Florjancic, Y. G. Gu, D. D. Anderson, C. S. Cooper, T. Zhang, R. F. Clark, Y. Cia, C. L. Black-Schaefer, L. Candace, J. O. McCall, C. G. Lerner, P. J. Hajduk, B. A. Beutel, V. S. Stoll, Chem. Biol. Drug Des. 2006, 67, 58-65.
- (2006) Chem. Biol. Drug Des , vol.67 , pp. 58-65
- Stamper, G.F.¹ Longenecker, K.L.² Fry, E.H.³ Clarissa, G.⁴ Florjancic, A.S.⁵ Gu, Y.G.⁶ Anderson, D.D.⁷ Cooper, C.S.⁸ Zhang, T.⁹ Clark, R.F.¹⁰ Cia, Y.¹¹ Black-Schaefer, C.L.¹² Candace, L.¹³ McCall, J.O.¹⁴ Lerner, C.G.¹⁵ Hajduk, P.J.¹⁶ Beutel, B.A.¹⁷ Stoll, V.S.¹⁸

18
- 0037179637
- A. de Dios, L. Prieto, J. A. Martin, A. Rubio, J. Ezquerra, M. Tebbe, B. Lopez de Uralde, J. Martin, A. Sanchez, D. L. LeToruneau, J. E. McGee, C. Boylan, T. R. Parr, Jr., M. C. Smith, J. Med. Chem. 2002, 45, 4559-4570.
- (2002) J. Med. Chem , vol.45 , pp. 4559-4570
- de Dios, A.¹ Prieto, L.² Martin, J.A.³ Rubio, A.⁴ Ezquerra, J.⁵ Tebbe, M.⁶ Lopez de Uralde, B.⁷ Martin, J.⁸ Sanchez, A.⁹ LeToruneau, D.L.¹⁰ McGee, J.E.¹¹ Boylan, C.¹² Parr Jr., T.R.¹³ Smith, M.C.¹⁴

19
- 33845864229
- C. D. Klein, A. Bachelier, J. Compt.-Aided Mol. Des. 2006, 20, 621-628.
- (2006) J. Compt.-Aided Mol. Des , vol.20 , pp. 621-628
- Klein, C.D.¹ Bachelier, A.²

20
- 0037241238
- A. H. Katz, C. E. Caufield, Curr. Pharm. Des. 2003, 9, 857-866.
- (2003) Curr. Pharm. Des , vol.9 , pp. 857-866
- Katz, A.H.¹ Caufield, C.E.²

21
- 33749852183
- K. M. Comess, M. E. Schurdak, M. J. Voorbach, M. Coen, J. D. Trumbull, H. Yang, L. Gao, H. Tang, X. Cheng, C. G. Lerner, J. O. McCall, D. J. Burns, B. A. Beutel, J. Biomol. Screening 2006, 11, 743-754.
- (2006) J. Biomol. Screening , vol.11 , pp. 743-754
- Comess, K.M.¹ Schurdak, M.E.² Voorbach, M.J.³ Coen, M.⁴ Trumbull, J.D.⁵ Yang, H.⁶ Gao, L.⁷ Tang, H.⁸ Cheng, X.⁹ Lerner, C.G.¹⁰ McCall, J.O.¹¹ Burns, D.J.¹² Beutel, B.A.¹³

22
- 3843140372
- G. Deng, R.-F. Gu, S. Mamor, S. L. Fisher, H. Jahie, G. Sonyal, J. Pharm. Biomed. Anal. 2004, 35, 817-828.
- (2004) J. Pharm. Biomed. Anal , vol.35 , pp. 817-828
- Deng, G.¹ Gu, R.-F.² Mamor, S.³ Fisher, S.L.⁴ Jahie, H.⁵ Sonyal, G.⁶

23
- 0037375658
- A. El Zoeiby, M. Beaumont, E. Dubuc, F. Sanschagrin, N. Voyer, R. C. Levesque, Bioorg. Med. Chem. 2003, 11, 1583-1592.
- (2003) Bioorg. Med. Chem , vol.11 , pp. 1583-1592
- El Zoeiby, A.¹ Beaumont, M.² Dubuc, E.³ Sanschagrin, F.⁴ Voyer, N.⁵ Levesque, R.C.⁶

24
- 29944442521
- E. Z. Baum, S. M. Crespo-Carbone, D. Abbanat, B. Foleno, A. Maden, R. Goldschmidt, K. Bush, Antimicrob. Agents Chemother. 2006, 50, 230-236.
- (2006) Antimicrob. Agents Chemother , vol.50 , pp. 230-236
- Baum, E.Z.¹ Crespo-Carbone, S.M.² Abbanat, D.³ Foleno, B.⁴ Maden, A.⁵ Goldschmidt, R.⁶ Bush, K.⁷

25
- 0037463751
- M. Maletic, J. Antonic, A. Leeman, G. Santorelli, S. Waddell, Bioorg. Med. Chem. Lett. 2003, 13, 1125-1128.
- (2003) Bioorg. Med. Chem. Lett , vol.13 , pp. 1125-1128
- Maletic, M.¹ Antonic, J.² Leeman, A.³ Santorelli, G.⁴ Waddell, S.⁵

26
- 31944448127
- Y. Yang, A. Severin, R. Chopra, G. Krishnamurthy, G. Singh, W. Hu, D. Keeney, K. Svenson, P. J. Petersen, P. Labthavikul, D. M. Shlaes, B. A. Rasmussen, A. A. Failli, J. S. Shumsky, K. M. Kutterer, A. Gilbert, T. S. Mansour, Antimicrob. Agents Chemother. 2006, 50, 556-564.
- (2006) Antimicrob. Agents Chemother , vol.50 , pp. 556-564
- Yang, Y.¹ Severin, A.² Chopra, R.³ Krishnamurthy, G.⁴ Singh, G.⁵ Hu, W.⁶ Keeney, D.⁷ Svenson, K.⁸ Petersen, P.J.⁹ Labthavikul, P.¹⁰ Shlaes, D.M.¹¹ Rasmussen, B.A.¹² Failli, A.A.¹³ Shumsky, J.S.¹⁴ Kutterer, K.M.¹⁵ Gilbert, A.¹⁶ Mansour, T.S.¹⁷

27
- 27744484480
- S. Antane, C. E. Caufield, W. Hu, D. Keeney, P. Labthavikul, K. Morris, S. M. Naughton, P. J. Petersen, B. A. Rasmussen, G. Singh, Y. Yang, Bioorg. Med. Chem. Lett. 2006, 16, 176-180.
- (2006) Bioorg. Med. Chem. Lett , vol.16 , pp. 176-180
- Antane, S.¹ Caufield, C.E.² Hu, W.³ Keeney, D.⁴ Labthavikul, P.⁵ Morris, K.⁶ Naughton, S.M.⁷ Petersen, P.J.⁸ Rasmussen, B.A.⁹ Singh, G.¹⁰ Yang, Y.¹¹

28
- 33845894155
- L. L. Silver, Nat. Rev. Drug Discovery 2007, 6, 41-55.
- (2007) Nat. Rev. Drug Discovery , vol.6 , pp. 41-55
- Silver, L.L.¹

29
- 0008103724
- T. Reffstrup, P. M. Boll, Phytochemistry 1979, 18, 325-326.
- (1979) Phytochemistry , vol.18 , pp. 325-326
- Reffstrup, T.¹ Boll, P.M.²

30
- 33645059318
- D. W. Knight, G. Pattenden, J. Chem. Soc. Perkin Trans. 1 1979, 84-88.
- (1979) J. Chem. Soc. Perkin Trans. 1 , pp. 84-88
- Knight, D.W.¹ Pattenden, G.²

31
- 37049092048
- A. C. Campbell, M. S. Maidment, J. H. Pick, D. F. M. Stevenson, J. Chem. Soc. Perkin Trans. 1 1985, 1567-1576.
- (1985) J. Chem. Soc. Perkin Trans. 1 , pp. 1567-1576
- Campbell, A.C.¹ Maidment, M.S.² Pick, J.H.³ Stevenson, D.F.M.⁴

32
- 84970616552
- M. Gill, M. J. Kiefel, D. A. Lally, A. Ten, Aust. J. Chem. 1990, 43, 1497-1518.
- (1990) Aust. J. Chem , vol.43 , pp. 1497-1518
- Gill, M.¹ Kiefel, M.J.² Lally, D.A.³ Ten, A.⁴

33
- 54849413926
- Antimicrobial susceptibility testing: The in vitro activities of the antibiotics were determined by the broth microdilution method as recommended by the Clinical Laboratory Standards Institute (CLSI, Methods for Dilution Antimicrobial Susceptibility Tests for Bacteria That Grow Aerobically; Approved Standards: M7-A7, 26, 7th ed, Clinical and Laboratory Standards Institute, Wayne, PA (USA, 2006) using Mueller-Hinton II broth (MHBII, BBL Cockeysville, MD, USA, Microtiter plates containing serial dilutions of each antimicrobial agent were inoculated with each organism to yield the appropriate density (105 CFUmL-1) in a final of 100 mL. The plates were incubated for 18-22 h at 35°C in ambient air. The MIC for all isolates was defined as the lowest concentration of antimicrobial agent that completely inhibits the growth of the organism as detected by the unaided eye
- -1) in a final volume of 100 mL. The plates were incubated for 18-22 h at 35°C in ambient air. The MIC for all isolates was defined as the lowest concentration of antimicrobial agent that completely inhibits the growth of the organism as detected by the unaided eye.

34
- 33750073841
- For recent reviews on tetronic acids, see: a
- For recent reviews on tetronic acids, see: a) A. L. Zografos, D. Georgiadis, Synthesis 2006, 3157-3188;
- (2006) Synthesis , pp. 3157-3188
- Zografos, A.L.¹ Georgiadis, D.²

35
- 33845734121
- b) R. Schobert, Naturwissenschaften 2006, 94, 1-11.
- (2006) Naturwissenschaften , vol.94 , pp. 1-11
- Schobert, R.¹

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