Erratum to "Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template" [Bioorg. Med. Chem. 16 (2008) 2974-2983] (DOI:10.1016/j.bmc.2007.12.047);Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template

Bioorganic and Medicinal Chemistry

Volumn 16, Issue 6, 2008, Pages 2974-2983

  Spencer, John ^a   Gaffen, John ^a   Griffin, Eric ^a   Harper, Elaine A ^a   Linney, Ian D ^a   McDonald, Iain M ^a   Roberts, Sonia P ^a   Shaxted, Mark E ^a   Adatia, Trushar ^b   Bashall, Alan ^b  

^a James Black Foundation   (United Kingdom)

^b LONDON METROPOLITAN UNIVERSITY   (United Kingdom)

Author keywords

Antagonist; Benzotriazepine; CCK; CCK2; Gastrin

Indexed keywords

1H 1,3,5 BENZOTRIAZEPINE 2,4 (3H,5H)DIONE; 2 [1 CYCLOHEPTYL 2,4 DIOXO 5 (2 OXO 2 PYRROLIDIN 1 YL ETHYL) 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N 3 TOLYL ACETAMIDE; 2 [1 CYCLOHEPTYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N 3 TOLYL ACETAMIDE; 2 [1 CYCLOHEPTYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N [3 (5 OXO 2,5 DIHYDRO[1,2,4]OXADIAZOL 3 YL)PHENYL]ACETAMIDE; 2 [1 CYCLOHEXYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N (3 METHYLAMINO PHENYL)ACETAMIDE; 2 [1 CYCLOHEXYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N [3 (2 METHYL THIAZOL 4 YL)PHENYL]ACETAMIDE; 2 [1 CYCLOHEXYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N [3 (5 OXO 2,5 DIHYDRO[1,2,4]OXADIAZOL 3 YL)PHENYL]ACETAMIDE; 2 [1 CYCLOHEXYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N [3 [METHYL(2H TETRAZOL 5 YL)AMINO]PHENYL]ACETAMIDE; 2 [2,4 DIOXO 1 (2 OXO 2 PYRROLIDIN 1 YL ETHYL) 5 PHENYL 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N PHENYL ACETAMIDE; 3 [2 (2,4 DIOXO 1 (2 OXO 2 PYRROLIDIN 1 YL ETHYL) 5 PHENYL 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL)ACETYLAMINO]BENZOIC ACID; 3 [3[ 2 [1 CYCLOHEXYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]ACETYLAMINO]PHENYL]PROPIONIC ACID; 4 [1 CYCLOHEXYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]N [3 (5 OXO 2,5 DIHYDRO[1,2,4]OXADIAZOL 3 YL)PHENYL]BUTYRAMIDE; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ B RECEPTOR ANTAGONIST; CHOLECYSTOKININ RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG; [3[ 2 [1 CYCLOHEPTYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]ACETYLAMINO]PHENYLSULFANYL]ACETIC ACID; [3[ 2 [1 CYCLOHEPTYL 5 (3,3 DIMETHYL 2 OXO BUTYL) 2,4 DIOXO 1,2,4,5 TETRAHYDRO 1,3,5 BENZOTRIAZEPIN 3 YL]ACETYLAMINO]PHENYL]ACETIC ACID; BENZAZEPINE DERIVATIVE; CHOLECYSTOKININ B RECEPTOR; TRIAZINE DERIVATIVE;

ANALYTIC METHOD; ARTICLE; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ANIMAL; CHEMISTRY; DRUG ANTAGONISM; HUMAN; PROTEIN BINDING; STRUCTURE ACTIVITY RELATION;

ANIMALS; BENZAZEPINES; HUMANS; PROTEIN BINDING; RECEPTOR, CHOLECYSTOKININ B; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZINES;

EID: 40949147712     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2008.05.070     Document Type: Erratum

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