Synthesis and biological activity of 1-alkylcarbonylmethyl analogues of YM022

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 1, 1996, Pages 51-54

  Semple, Graeme ^a   Ryder, Hamish ^a   Kendrick, David A ^a   Szelke, Michael ^a   Ohta, Mitsuaki ^b   Satoh, Masato ^b   Nishida, Akito ^b   Akuzawa, Shinobu ^b   Miyata, Keiji ^b  

^a Chilworth Research Centre   (United Kingdom)

^b Yamanouchi Inst Drug Discov Res   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2,3 DIHYDRO 1 METHYL 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL) 3 (3 METHYLPHENYL)UREA; 1 [1 (TERT BUTYLCARBONYLMETHYL) 2,3 DIHYDRO 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL] 3 (3 METHYLPHENYL)UREA; 1 [2,3 DIHYDRO 1 (2' METHYLPHENACYL) 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL] 3 (3 METHYLPHENYL)UREA; BENZODIAZEPINE DERIVATIVE; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ B RECEPTOR; CHOLECYSTOKININ OCTAPEPTIDE; DEVAZEPIDE; GASTRIN ANTAGONIST; GASTRIN RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; ENANTIOMER; INTRAGASTRIC DRUG ADMINISTRATION; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN; PANCREAS; STOMACH ACID SECRETION; STRUCTURE ACTIVITY RELATION;

ANIMALIA;

EID: 0030063935     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(95)00556-9     Document Type: Article

References (11)

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