Solid-phase peptide library synthesis on HiCore resin for screening substrate specificity of Brk protein tyrosine kinase

Journal of Combinatorial Chemistry

Volumn 10, Issue 1, 2008, Pages 20-23

  Shin, Dong Sik ^a   Kim, Yun Gon ^a   Kim, Eun Mi ^a   Kim, Mira ^a   Park, Hyung Yeon ^b   Kim, June Hyung ^c   Lee, Bon Su ^b   Kim, Byung Gee ^a   Lee, Yoon Sik ^a  

^a Seoul National University   (South Korea)

^b Inha University   (South Korea)

^c Dong A University   (South Korea)

Author keywords

[No Author keywords available]

Indexed keywords

CROSS LINKING REAGENT; PEPTIDE; PEPTIDE LIBRARY; PROTEIN TYROSINE KINASE; PTK6 PROTEIN, HUMAN; RESIN; TUMOR PROTEIN; UNCLASSIFIED DRUG;

ARTICLE; CHEMISTRY; COMBINATORIAL CHEMISTRY; DRUG DESIGN; ENZYME SPECIFICITY; MASS SPECTROMETRY; SYNTHESIS;

COMBINATORIAL CHEMISTRY TECHNIQUES; CROSS-LINKING REAGENTS; DRUG DESIGN; NEOPLASM PROTEINS; PEPTIDE LIBRARY; PEPTIDES; PROTEIN-TYROSINE KINASES; RESINS, SYNTHETIC; SPECTROMETRY, MASS, MATRIX-ASSISTED LASER DESORPTION-IONIZATION; SUBSTRATE SPECIFICITY;

EID: 38849181530     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc7001217     Document Type: Article

References (34)

1. Lam, K. S.; Salmon, S. E.; Hersh, E. M.; Hruby, V. J.; Kazmierski, W. M.; Knapp, R. J. Nature 1991, 354, 82-84.
2. Houghten, R. A. Proc. Natl. Acad. Sci. U.S.A. 1984, 82, 5131-5135.
3. (a) Lau, D. H.; Guo, L.; Liu, R.; Song, A.; Shao, C.; Lam, K. S Biotechnol. Lett. 2002, 24, 497-500.
4. (b) St. Hilaire, P. M.; Alvesv, L. C.; Herrera, F.; Renil, M.; Sanderson, S. J.; Mottram, J. C.; Coombs, G. H.; Juliano, M. A.; Juliano, L.; Arevalo, J.; Meldal, M. J. Med. Chem. 2002, 45, 1971-1982.
5. (c) Verdoliva, A.; Marasco, D.; De Capua, A.; Saporito, A.; Bellofiore, P.; Manfredi, V.; Fattorusso, R.; Pedone, C.; Ruvo, M. ChemBioChem 2005, 6, 1242-1253.
6. (d) Shin, D. S.; Kim, D. H.; Chung, W. J.; Lee, Y. S. J. Biochem. Mol. Biol. 2005, 38, 517-525.
7. (a) Laursen, R. A. Eur. J. Biochem. 1971, 20, 89-102.
8. (b) Matsueda, G. R.; Haber, E.; Margolies, M. N. Biochemistry 1981, 20, 2571-2580.
9. (c) Fields, C. G.; VanDrisse, V. L.; Fields, G. B. Pept. Res. 1993, 6, 39-47.
10. (a) Youngquist, R. S.; Fuentes, G. R.; Lacey, M. P.; Keough, T. J. Am. Chem. Soc. 1995, 117, 3900-3906.
11. (b) Wang, X.; Peng, L.; Liu, R.; Gill, S. S.; Lam, K. S. J. Comb. Chem. 2005, 7, 197-209.
12. (a) Spetzler, J. C.; Westphal, V.; Winther, J. R.; Meldal, M. J. Pept. Sci. 1998, 4, 128-137.
13. (b) Song, A.; Zhang, J.; Lebrilla, C. B.; Lam, K. S. J. Am. Chem. Soc. 2003, 125, 6180-6188.
14. (c) Ying, L.; Liu, R.; Zhang, J.; Lam, K.; Lebrilla, C. B.; Gervay-Hague, J. J. Comb. Chem. 2005, 7, 372-384.
15. Franz, A. H.; Liu, R.; Song, A.; Lam, K. S.; Lebrilla, C. B. J. Comb. Chem. 2003, 5, 125-137.
16. (a) Kim, H.; Cho, J. K.; Chung, W. J.; Lee, Y. S. Org. Lett. 2004, 6, 3273-3276.
17. (b) HiCore® resin is commercially available from BeadTechlnc (www.beadtech.co.kr).
18. Kim, D. H.; Lee, H. Y.; Kim, H.; Kim, H.; Lee, Y. S.; Park, S. B. J. Comb. Chem. 2006, 8, 280-285.
19. (a) Shin, J. S.; Kim, B. G.; Kim, D. H.; Lee, Y. S Anal. Biochem. 1996, 236, 9-13.
20. (b) Lee, Y. S.; Kim, D. H. In Peptide 1996; Ramage, R., Epton, R., Eds.; Mayflower Scientific: Birmingham, U.K., 1997; pp 571-572.
21. Kaiser, E.; Colescott, R. L.; Bossinger, C. D.; Cook, P. I. Anal. Biochem. 1970, 34, 595-598.
22. Bunin, B. A. The Combinatorial Index; Academic Press: San Diego, 1998; pp 219-220.
23. Ullrich, A.; Schlessinger, J. Cell 1990, 61, 203-212.
24. (a) Harvey, A. J.; Crompton, M. R. Anti-Cancer Drugs 2004, 15, 107-111.
25. (b) Kasprzycka, M.; Majewski, M.; Wang, Z. J.; Ptasznik, A; Wysocka, M.; Zhang, Q.; Marzec, M.; Gimotty, P.; Crompton, M. R.; Wasik, M. A. Am. J. Pathol. 2006, 168, 1631-1641.
26. (a) Martin, S. E.; Peterson, B. J. Pept. Sci. 2002, 8, 227-233.
27. (b) Kim, Y. G.; Shin, D. S.; Kim, E. M.; Park, H. Y.; Lee, C. S.; Kim, J. H.; Lee, B. S.; Lee, Y. S.; Kim, B. G. Angew. Chem., Int. Ed. 2007, 46, 5408-5411.
28. (a) Crooks, G. E.; Hon, G.; Chandonia, J.-M.; Brenner, S. E Genome Res. 2004, 14, 1188-1190.
29. (b) Fujii, K.; Zhu, G.; Liu, Y.; Hallam, J.; Chen, L.; Herrero, J.; Shaw, S. Proc. Natl. Acad. Sci. U.S.A. 2004, 101, 13744-13749.
30. Qiu, H.; Miller, W. T. Oncogene 2004, 23, 2216-2223.
31. Songyang, Z.; Cantley, L. C. Trends Biochem. Sci. 1995, 20, 470-475.
32. (a) Lou, Q.; Wu, J.; Salmon, S. E.; Lam, K. S. Lett. Pept. Sci. 1995, 2, 289-296.
33. (b) Lou, Q.; Leftwich, M. E.; Lam, K. S. Bioorg. Med. Chem. 1996, 4, 677-682.
34. Kreegipuu, A.; Blom, N.; Järv, S. J. FEBS Lett. 1998, 430, 45-50.