-
1
-
-
36849035258
-
-
Reviews of cross-coupling methodology: a
-
Reviews of cross-coupling methodology: a) B. U. W. Maes, Top. Heterocycl. Chem. 2006, 1, 155-211;
-
(2006)
Top. Heterocycl. Chem
, vol.1
, pp. 155-211
-
-
Maes, B.U.W.1
-
2
-
-
20544450502
-
-
A. de Meijere, F. Diederich Eds, Wiley-VCH, Weinheim
-
b) A. de Meijere, F. Diederich (Eds.), Metal-Catalyzed Cross-Coupling Reactions, Wiley-VCH, Weinheim, 2004;
-
(2004)
Metal-Catalyzed Cross-Coupling Reactions
-
-
-
3
-
-
0036589259
-
-
c) J. Hassan, M. Sévignon, C. Gozzi, E. Schultz, M. Lemaire, Chem. Rev. 2002, 102, 1359-1470;
-
(2002)
Chem. Rev
, vol.102
, pp. 1359-1470
-
-
Hassan, J.1
Sévignon, M.2
Gozzi, C.3
Schultz, E.4
Lemaire, M.5
-
7
-
-
33745079610
-
-
b) J. S. Carey, D. Laffan, C. Thomson, M. T. Williams, Org. Biomol. Chem. 2006, 4, 2337-2347.
-
(2006)
Org. Biomol. Chem
, vol.4
, pp. 2337-2347
-
-
Carey, J.S.1
Laffan, D.2
Thomson, C.3
Williams, M.T.4
-
11
-
-
33947416063
-
-
b) K. Billingsley, K. W. Anderson, S. L. Buchwald, J. Am. Chem. Soc. 2007, 129, 3358-3366.
-
(2007)
J. Am. Chem. Soc
, vol.129
, pp. 3358-3366
-
-
Billingsley, K.1
Anderson, K.W.2
Buchwald, S.L.3
-
12
-
-
0037244546
-
-
For a review of heterocyclic boronic acids
-
For a review of heterocyclic boronic acids: E. Tyrrell, P. Brookes, Synthesis 2003, 469-483.
-
(2003)
Synthesis
, pp. 469-483
-
-
Tyrrell, E.1
Brookes, P.2
-
15
-
-
0037474677
-
-
c) A. A. Fuller, H. R. Hester, E. V. Salo, E. P. Stevens, Tetrahedron Lett. 2003, 44, 2935-2938;
-
(2003)
Tetrahedron Lett
, vol.44
, pp. 2935-2938
-
-
Fuller, A.A.1
Hester, H.R.2
Salo, E.V.3
Stevens, E.P.4
-
16
-
-
21244487916
-
-
d) M. D. Helm, J. E. Moore, A. Plant, J. P. A. Harrity, Angew. Chem. Int. Ed. 2005, 44, 3889-3892.
-
(2005)
Angew. Chem. Int. Ed
, vol.44
, pp. 3889-3892
-
-
Helm, M.D.1
Moore, J.E.2
Plant, A.3
Harrity, J.P.A.4
-
19
-
-
36849039834
-
-
Eds, F. Diederich, A. de Meijere, Wiley-VCH, Weinheim, ch. 2;
-
c) N. Miyaura in Metal-Catalyzed Cross-Coupling Reactions (Eds.: F. Diederich, A. de Meijere), Wiley-VCH, Weinheim, 2004, ch. 2;
-
(2004)
Metal-Catalyzed Cross-Coupling Reactions
-
-
Miyaura, N.1
-
21
-
-
0035821359
-
-
Reviews of lithiation of azines: a
-
Reviews of lithiation of azines: a) F. Mongin, G. Quéguiner, Tetrahedron 2001, 57, 4059-4090;
-
(2001)
Tetrahedron
, vol.57
, pp. 4059-4090
-
-
Mongin, F.1
Quéguiner, G.2
-
22
-
-
0035927228
-
-
b) A. Turck, N. Plé, F. Mongin, G. Quéguiner, Tetrahedron 2001, 57, 4489-4505.
-
(2001)
Tetrahedron
, vol.57
, pp. 4489-4505
-
-
Turck, A.1
Plé, N.2
Mongin, F.3
Quéguiner, G.4
-
23
-
-
0012397313
-
-
a) V. Snieckus, Chem. Rev. 1990, 90, 879-933;
-
(1990)
Chem. Rev
, vol.90
, pp. 879-933
-
-
Snieckus, V.1
-
24
-
-
3242659209
-
-
b) M. C. Whisler, S. MacNeil, V. Snieckus, P. Beak, Angew. Chem. Int. Ed. 2004, 43, 2206-2225;
-
(2004)
Angew. Chem. Int. Ed
, vol.43
, pp. 2206-2225
-
-
Whisler, M.C.1
MacNeil, S.2
Snieckus, V.3
Beak, P.4
-
25
-
-
2942530950
-
-
c) R. Chinchilla, C. Nájera, M. Yus, Chem. Rev. 2004, 104, 2667-2722.
-
(2004)
Chem. Rev
, vol.104
, pp. 2667-2722
-
-
Chinchilla, R.1
Nájera, C.2
Yus, M.3
-
26
-
-
0036532565
-
-
a) A. Bouillon, J.-C. Lancelot, V. Collot, P. R. Bovy, S. Rault, Tetrahedron 2002, 58, 2885-2890;
-
(2002)
Tetrahedron
, vol.58
, pp. 2885-2890
-
-
Bouillon, A.1
Lancelot, J.-C.2
Collot, V.3
Bovy, P.R.4
Rault, S.5
-
27
-
-
0037156677
-
-
b) A. Bouillon, J.-C. Lancelot, V. Collot, P. R. Bovy, S. Rault, Tetrahedron 2002, 58, 3323-3328;
-
(2002)
Tetrahedron
, vol.58
, pp. 3323-3328
-
-
Bouillon, A.1
Lancelot, J.-C.2
Collot, V.3
Bovy, P.R.4
Rault, S.5
-
28
-
-
0037182035
-
-
c) A. Bouillon, J.-C. Lancelot, P. R. Bovy, S. Rault, Tetrahedron 2002, 58, 4369-4373;
-
(2002)
Tetrahedron
, vol.58
, pp. 4369-4373
-
-
Bouillon, A.1
Lancelot, J.-C.2
Bovy, P.R.3
Rault, S.4
-
29
-
-
0037178508
-
-
d) W. Li, D. P. Nelson, M. S. Jensen, R. S. Hoerrner, D. Cai, R. D. Larsen, P. J. Reider, J. Org. Chem. 2002, 67, 5394-5397;
-
(2002)
J. Org. Chem
, vol.67
, pp. 5394-5397
-
-
Li, W.1
Nelson, D.P.2
Jensen, M.S.3
Hoerrner, R.S.4
Cai, D.5
Larsen, R.D.6
Reider, P.J.7
-
30
-
-
0037131349
-
-
e) P. R. Parry, C. Wang, A. S. Batsanov, M. R. Bryce, B. Tarbit, J. Org. Chem. 2002, 67, 7541-7543;
-
(2002)
J. Org. Chem
, vol.67
, pp. 7541-7543
-
-
Parry, P.R.1
Wang, C.2
Batsanov, A.S.3
Bryce, M.R.4
Tarbit, B.5
-
31
-
-
0242467635
-
-
f) A. Bouillon, J.-C. Lancelot, J. Sopkova, O. de Santos, V. Collot, P. R. Bovy, S. Rault, Tetrahedron 2003, 59, 10043-10049;
-
(2003)
Tetrahedron
, vol.59
, pp. 10043-10049
-
-
Bouillon, A.1
Lancelot, J.-C.2
Sopkova, J.3
de Santos, O.4
Collot, V.5
Bovy, P.R.6
Rault, S.7
-
32
-
-
0347623383
-
-
g) A. Bouillon, A. S. Voisin, A. Robic, J.-C. Lancelot, V. Collot, S. Rault, J. Org. Chem. 2003, 68, 10178-10180;
-
(2003)
J. Org. Chem
, vol.68
, pp. 10178-10180
-
-
Bouillon, A.1
Voisin, A.S.2
Robic, A.3
Lancelot, J.-C.4
Collot, V.5
Rault, S.6
-
35
-
-
11844280304
-
-
j) A. E. Thompson, G. Hughes, A. S. Batsanov, M. R. Bryce, P. R. Parry, B. Tarbit, J. Org. Chem. 2005, 70, 388-390;
-
(2005)
J. Org. Chem
, vol.70
, pp. 388-390
-
-
Thompson, A.E.1
Hughes, G.2
Batsanov, A.S.3
Bryce, M.R.4
Parry, P.R.5
Tarbit, B.6
-
36
-
-
24944474804
-
-
k) H. M. Hansen, M. Lysen, M. Begtrup, J. Kristensen, Tetrahedron 2005, 61, 9955-9960;
-
(2005)
Tetrahedron
, vol.61
, pp. 9955-9960
-
-
Hansen, H.M.1
Lysen, M.2
Begtrup, M.3
Kristensen, J.4
-
37
-
-
18144379513
-
-
l) A. E. Thompson, A. S. Batsanov, M. R. Bryce, N. Saygili, P. R. Parry, B. Tarbit, Tetrahedron 2005, 61, 5131-5135;
-
(2005)
Tetrahedron
, vol.61
, pp. 5131-5135
-
-
Thompson, A.E.1
Batsanov, A.S.2
Bryce, M.R.3
Saygili, N.4
Parry, P.R.5
Tarbit, B.6
-
38
-
-
30544445259
-
-
m) T. Cailly, F. Fabis, A. Bouillon, S. Lemaître, J. Sopkova, O. de Santos, S. Rault, Synlett 2006, 53-56;
-
(2006)
Synlett
, pp. 53-56
-
-
Cailly, T.1
Fabis, F.2
Bouillon, A.3
Lemaître, S.4
Sopkova, J.5
de Santos, O.6
Rault, S.7
-
39
-
-
33750737691
-
-
n) A. S. Voisin, A. Bouillon, I. Berenguer, J.-C. Lancelot, A. Lesnard, S. Rault, Tetrahedron 2006, 62, 11734-11739;
-
(2006)
Tetrahedron
, vol.62
, pp. 11734-11739
-
-
Voisin, A.S.1
Bouillon, A.2
Berenguer, I.3
Lancelot, J.-C.4
Lesnard, A.5
Rault, S.6
-
40
-
-
33847659575
-
-
o) M. Alessi, A. L. Larkin, K. A. Ogilvie, L. A. Green, S. Lai, S. Lopez, V. Snieckus, J. Org. Chem. 2007, 72, 1588-1594.
-
(2007)
J. Org. Chem
, vol.72
, pp. 1588-1594
-
-
Alessi, M.1
Larkin, A.L.2
Ogilvie, K.A.3
Green, L.A.4
Lai, S.5
Lopez, S.6
Snieckus, V.7
-
41
-
-
30444451469
-
-
I. A. I. Mkhalid, D. Coventry, D. Albesa-Jove, A. S. Batsanov, J. A. K. Howard, R. N. Perutz, T. B. Marder, Angew. Chem. Int. Ed. 2006, 45, 489-491.
-
(2006)
Angew. Chem. Int. Ed
, vol.45
, pp. 489-491
-
-
Mkhalid, I.A.I.1
Coventry, D.2
Albesa-Jove, D.3
Batsanov, A.S.4
Howard, J.A.K.5
Perutz, R.N.6
Marder, T.B.7
-
42
-
-
0001444995
-
-
a) T. K. Liao, E. G. Podrebarac, C. C. Cheng, J. Am. Chem. Soc. 1964, 86, 1869-1870;
-
(1964)
J. Am. Chem. Soc
, vol.86
, pp. 1869-1870
-
-
Liao, T.K.1
Podrebarac, E.G.2
Cheng, C.C.3
-
43
-
-
0025650936
-
-
b) D. Peters, A.-B. Hornfield, S. Gronowitz, J. Heterocycl. Chem. 1990, 27, 2165-2173.
-
(1990)
J. Heterocycl. Chem
, vol.27
, pp. 2165-2173
-
-
Peters, D.1
Hornfield, A.-B.2
Gronowitz, S.3
-
44
-
-
1842586937
-
-
N. Saygili, A. S. Batsanov, M. R. Bryce, Org. Biomol. Chem. 2004, 2, 852-857.
-
(2004)
Org. Biomol. Chem
, vol.2
, pp. 852-857
-
-
Saygili, N.1
Batsanov, A.S.2
Bryce, M.R.3
-
46
-
-
0037182002
-
-
Functionalized pyrimidines: a V. Bonnet, F. Mongin, F. Trecourt, G. Queguiner, P. Knochel, Tetrahedron 2002, 58, 4429-4438;
-
Functionalized pyrimidines: a) V. Bonnet, F. Mongin, F. Trecourt, G. Queguiner, P. Knochel, Tetrahedron 2002, 58, 4429-4438;
-
-
-
-
47
-
-
1842690073
-
-
b) B. Gong, F. Hong, C. Kohm, S. Jenkins, J. Tulinsky, R. Bhatt, P. de Vries, J. W. Singer, P. Klein, Bioorg. Med. Chem. Lett. 2004, 14, 2303-2308;
-
(2004)
Bioorg. Med. Chem. Lett
, vol.14
, pp. 2303-2308
-
-
Gong, B.1
Hong, F.2
Kohm, C.3
Jenkins, S.4
Tulinsky, J.5
Bhatt, R.6
de Vries, P.7
Singer, J.W.8
Klein, P.9
-
48
-
-
33748463567
-
-
c) C. G. Hartung, A. C. Backes, B. Felber, A. Missio, A. Philipp, Tetrahedron 2006, 62, 10055-10064;
-
(2006)
Tetrahedron
, vol.62
, pp. 10055-10064
-
-
Hartung, C.G.1
Backes, A.C.2
Felber, B.3
Missio, A.4
Philipp, A.5
-
49
-
-
33747519108
-
-
d) R. T. Wheelhouse, S. A. Jennings, V. A. Phillips, D. Pletsas, P. M. Murphy, N. C. Garbett, J. B. Chaires, T. C. Jenkins, J. Med. Chem. 2006, 49, 5187-5198.
-
(2006)
J. Med. Chem
, vol.49
, pp. 5187-5198
-
-
Wheelhouse, R.T.1
Jennings, S.A.2
Phillips, V.A.3
Pletsas, D.4
Murphy, P.M.5
Garbett, N.C.6
Chaires, J.B.7
Jenkins, T.C.8
-
50
-
-
12144276704
-
-
For biologically significant azabiaryls: a
-
For biologically significant azabiaryls: a) T. T. Denton, X. Zhang, J. R. Cashman, J. Med. Chem. 2005, 48, 224-239;
-
(2005)
J. Med. Chem
, vol.48
, pp. 224-239
-
-
Denton, T.T.1
Zhang, X.2
Cashman, J.R.3
-
51
-
-
18344379308
-
-
b) R. A. Smith, D. L. Hertzog, M. H. Osterhout, G. H. Ladouceur, M. Korpusik, M. A. Bobko, J. H. Jones, K. Phelan, R. H. Romero, T. Hundertmark, M. L. MacDougall, J. N. Livingston, W. R. Shoen, Bioorg. Med. Chem. Lett. 2002, 12, 1303-1306.
-
(2002)
Bioorg. Med. Chem. Lett
, vol.12
, pp. 1303-1306
-
-
Smith, R.A.1
Hertzog, D.L.2
Osterhout, M.H.3
Ladouceur, G.H.4
Korpusik, M.5
Bobko, M.A.6
Jones, J.H.7
Phelan, K.8
Romero, R.H.9
Hundertmark, T.10
MacDougall, M.L.11
Livingston, J.N.12
Shoen, W.R.13
-
52
-
-
0037181078
-
-
S. Ding, N. S. Gray, X. Wu, Q. Ding, P. G. Schultz, J. Am. Chem. Soc. 2002, 124, 1594-1596.
-
(2002)
J. Am. Chem. Soc
, vol.124
, pp. 1594-1596
-
-
Ding, S.1
Gray, N.S.2
Wu, X.3
Ding, Q.4
Schultz, P.G.5
-
53
-
-
36849079683
-
-
Analogous lithiation/borylation procedures on 2-amino-5-bromopyridine and 1-amino-4-bromobenzene gave complex product mixtures; the corresponding boronic acid/ester derivatives could not be isolated
-
Analogous lithiation/borylation procedures on 2-amino-5-bromopyridine and 1-amino-4-bromobenzene gave complex product mixtures; the corresponding boronic acid/ester derivatives could not be isolated.
-
-
-
-
54
-
-
36849049098
-
-
The isolated yields of cross-coupled products from in situ trapping of ester 9 were lower (based on 7) than from reactions via the purified acid 8.
-
The isolated yields of cross-coupled products from in situ trapping of ester 9 were lower (based on 7) than from reactions via the purified acid 8.
-
-
-
-
55
-
-
30544445259
-
-
For example, o-cyanopyridylboronic esters are more suitable than the corresponding boronic acids: T. Cailly, F. Fabis, A. Bouillon, S. Lemaître, J. Sopkova, O. de Santos, S. Rault, Synlett 2006, 53-56.
-
For example, o-cyanopyridylboronic esters are more suitable than the corresponding boronic acids: T. Cailly, F. Fabis, A. Bouillon, S. Lemaître, J. Sopkova, O. de Santos, S. Rault, Synlett 2006, 53-56.
-
-
-
-
57
-
-
0034600318
-
-
b) A. F. Littke, C. Dai, G. C. Fu, J. Am. Chem. Soc. 2000, 122, 4020-4028.
-
(2000)
J. Am. Chem. Soc
, vol.122
, pp. 4020-4028
-
-
Littke, A.F.1
Dai, C.2
Fu, G.C.3
-
58
-
-
33745721269
-
-
N. Kudo, M. Perseghini, G. C. Fu, Angew. Chem. Int. Ed. 2006, 45, 1282-1284.
-
(2006)
Angew. Chem. Int. Ed
, vol.45
, pp. 1282-1284
-
-
Kudo, N.1
Perseghini, M.2
Fu, G.C.3
-
59
-
-
0142231050
-
-
For examples of 2-arylbenzothiazoles for biomedical applications see: V. J. Majo, J. Prabhakaran, J. J. Mann, J. S. D. Kumar, Tetrahedron Lett. 2003, 44, 8535-8537
-
For examples of 2-arylbenzothiazoles for biomedical applications see: V. J. Majo, J. Prabhakaran, J. J. Mann, J. S. D. Kumar, Tetrahedron Lett. 2003, 44, 8535-8537.
-
-
-
-
60
-
-
0036065902
-
-
For other successful Suzuki reactions with halogenated substrates containing a primary amino group see: a) ref, 10j] b F. Bracher, J. Daab, Chem. 2002, 2288-2291
-
[10j] b) F. Bracher, J. Daab, Eur. J. Org. Chem. 2002, 2288-2291.
-
-
-
-
61
-
-
33646497228
-
-
For a related cyclization see
-
For a related cyclization see: E. F. DiMauro, J. R. Vitullo, J. Org. Chem. 2006, 71, 3959-3962.
-
(2006)
J. Org. Chem
, vol.71
, pp. 3959-3962
-
-
DiMauro, E.F.1
Vitullo, J.R.2
-
63
-
-
0042910310
-
-
C. Boga, E. Del Vecchio, L. Forlani, P. E. Todesco, J. Organomet. Chem. 2000, 601, 233-236.
-
(2000)
J. Organomet. Chem
, vol.601
, pp. 233-236
-
-
Boga, C.1
Del Vecchio, E.2
Forlani, L.3
Todesco, P.E.4
-
64
-
-
36849051096
-
-
As noted by a referee, the degassing procedure does not ensure that the solvent is free of peroxide
-
As noted by a referee, the degassing procedure does not ensure that the solvent is free of peroxide.
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